Compile Data Set for Download or QSAR
Found 428 with Last Name = 'oliva' and Initial = 'ca'
TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50556952(CHEMBL4754487)copy SMILES
Affinity DataKi:  0.680nMAssay Description:Mixed-type inhibition of recombinant human AChE assessed as inhibition constant using acetylthiocholine iodide as substrate by Cornish-Bowden plot an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K077XJPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50556952(CHEMBL4754487)copy SMILES
Affinity DataKi:  0.940nMAssay Description:Mixed-type inhibition of recombinant human AChE assessed as dissociation constant for protein-substrate-compound complex using acetylthiocholine iodi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K077XJPubMed
TargetCyclin-C/Cyclin-dependent kinase 8(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350239(US10208056, Compound 66)copy SMILEScopy InChI
Affinity DataIC50: 0.191nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen. This is a kinase assay platform based on measuring the binding and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 8(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350249(US10208056, Compound 76)copy SMILEScopy InChI
Affinity DataIC50: 0.262nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen. This is a kinase assay platform based on measuring the binding and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 8(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350256(US10208056, Compound 83)copy SMILEScopy InChI
Affinity DataIC50: 0.278nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen. This is a kinase assay platform based on measuring the binding and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 8(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350253(US10208056, Compound 80)copy SMILEScopy InChI
Affinity DataIC50: 0.314nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen. This is a kinase assay platform based on measuring the binding and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 8(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350262(US10208056, Compound 89)copy SMILEScopy InChI
Affinity DataIC50: 0.407nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen. This is a kinase assay platform based on measuring the binding and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 8(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350240(US10208056, Compound 67)copy SMILEScopy InChI
Affinity DataIC50: 0.466nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen. This is a kinase assay platform based on measuring the binding and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350259(US10208056, Compound 86)copy SMILEScopy InChI
Affinity DataIC50: 0.480nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen). This is a kinase assay platform based on measuring the binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50556952(CHEMBL4754487)copy SMILES
Affinity DataIC50: 0.770nMAssay Description:Inhibition of recombinant human AChE using acetylthiocholineiodide as substrate preincubated for 20 mins followed by substrate addition by Ellman's m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K077XJPubMed
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350253(US10208056, Compound 80)copy SMILEScopy InChI
Affinity DataIC50: 0.770nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen). This is a kinase assay platform based on measuring the binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Spanish National Cancer Research Centre (CNIO)

Curated by ChEMBL
LigandPNGBDBM50364777(CHEMBL1952142)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMAssay Description:Inhibition of N-terminal 6-His tagged human recombinant PIM3 using PIM tide (ARKRRRHPSGPPTA) as substrate incubated for 1 hr by fluorescence based as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4P4JPubMed
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350249(US10208056, Compound 76)copy SMILEScopy InChI
Affinity DataIC50: 0.827nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen). This is a kinase assay platform based on measuring the binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Spanish National Cancer Research Centre (CNIO)

Curated by ChEMBL
LigandPNGBDBM50364777(CHEMBL1952142)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of His tagged human recombinant PIM1 using PIM tide (ARKRRRHPSGPPTA) as substrate incubated for 1 hr by fluorescence based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4P4JPubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Spanish National Cancer Research Centre (CNIO)

Curated by ChEMBL
LigandPNGBDBM50510183(CHEMBL4457634)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of N-terminal 6-His tagged human recombinant PIM3 using PIM tide (ARKRRRHPSGPPTA) as substrate incubated for 1 hr by fluorescence based as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XW4P4JPubMed
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350211(US10208056, Compound 43)copy SMILEScopy InChI
Affinity DataIC50: 1.09nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen). This is a kinase assay platform based on measuring the binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM10592(7-chloro-15-methyl-10-azatetracyclo[11.3.1.0^{2,11...)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of recombinant human AChE using acetylthiocholineiodide as substrate preincubated for 20 mins followed by substrate addition by Ellman's m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K077XJPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50556958(CHEMBL4744528)copy SMILES
Affinity DataIC50: 1.10nMAssay Description:Inhibition of recombinant human AChE using acetylthiocholineiodide as substrate preincubated for 20 mins followed by substrate addition by Ellman's m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K077XJPubMed
TargetCyclin-C/Cyclin-dependent kinase 8(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350252(US10208056, Compound 79)copy SMILEScopy InChI
Affinity DataIC50: 1.11nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen. This is a kinase assay platform based on measuring the binding and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 8(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350263(US10208056, Compound 90)copy SMILEScopy InChI
Affinity DataIC50: 1.36nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen. This is a kinase assay platform based on measuring the binding and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 8(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350265(US10208056, Compound 92)copy SMILEScopy InChI
Affinity DataIC50: 1.41nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen. This is a kinase assay platform based on measuring the binding and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350220(US10208056, Compound 52)copy SMILEScopy InChI
Affinity DataIC50: 1.41nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen). This is a kinase assay platform based on measuring the binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350202(US10208056, Compound 34)copy SMILEScopy InChI
Affinity DataIC50: 1.41nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen). This is a kinase assay platform based on measuring the binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 8(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350227(US10208056, Compound 57)copy SMILES
Affinity DataIC50: 1.41nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen. This is a kinase assay platform based on measuring the binding and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350183(US10208056, Compound 15)copy SMILEScopy InChI
Affinity DataIC50: 1.41nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen). This is a kinase assay platform based on measuring the binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350190(US10208056, Compound 22)copy SMILEScopy InChI
Affinity DataIC50: 1.41nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen). This is a kinase assay platform based on measuring the binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 8(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350220(US10208056, Compound 52)copy SMILEScopy InChI
Affinity DataIC50: 1.41nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen. This is a kinase assay platform based on measuring the binding and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 8(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350211(US10208056, Compound 43)copy SMILEScopy InChI
Affinity DataIC50: 1.41nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen. This is a kinase assay platform based on measuring the binding and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350263(US10208056, Compound 90)copy SMILEScopy InChI
Affinity DataIC50: 1.41nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen). This is a kinase assay platform based on measuring the binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350240(US10208056, Compound 67)copy SMILEScopy InChI
Affinity DataIC50: 1.41nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen). This is a kinase assay platform based on measuring the binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350239(US10208056, Compound 66)copy SMILEScopy InChI
Affinity DataIC50: 1.41nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen). This is a kinase assay platform based on measuring the binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 8(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350270(US10208056, Compound 105)copy SMILEScopy InChI
Affinity DataIC50: 1.41nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen. This is a kinase assay platform based on measuring the binding and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 8(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350268(US10208056, Compound 96)copy SMILEScopy InChI
Affinity DataIC50: 1.41nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen. This is a kinase assay platform based on measuring the binding and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 8(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350267(US10208056, Compound 95)copy SMILEScopy InChI
Affinity DataIC50: 1.41nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen. This is a kinase assay platform based on measuring the binding and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 8(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350257(US10208056, Compound 84)copy SMILEScopy InChI
Affinity DataIC50: 1.41nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen. This is a kinase assay platform based on measuring the binding and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350262(US10208056, Compound 89)copy SMILEScopy InChI
Affinity DataIC50: 1.41nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen). This is a kinase assay platform based on measuring the binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350256(US10208056, Compound 83)copy SMILEScopy InChI
Affinity DataIC50: 1.41nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen). This is a kinase assay platform based on measuring the binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50556953(CHEMBL4748114)copy SMILES
Affinity DataIC50: 1.90nMAssay Description:Inhibition of recombinant human AChE using acetylthiocholineiodide as substrate preincubated for 20 mins followed by substrate addition by Ellman's m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K077XJPubMed
TargetCyclin-C/Cyclin-dependent kinase 8(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350183(US10208056, Compound 15)copy SMILEScopy InChI
Affinity DataIC50: 1.96nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen. This is a kinase assay platform based on measuring the binding and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 8(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350190(US10208056, Compound 22)copy SMILEScopy InChI
Affinity DataIC50: 1.98nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen. This is a kinase assay platform based on measuring the binding and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 8(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350202(US10208056, Compound 34)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen. This is a kinase assay platform based on measuring the binding and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 8(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350255(US10208056, Compound 82)copy SMILEScopy InChI
Affinity DataIC50: 2.19nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen. This is a kinase assay platform based on measuring the binding and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 8(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350269(US10208056, Compound 104)copy SMILEScopy InChI
Affinity DataIC50: 2.41nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen. This is a kinase assay platform based on measuring the binding and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 8(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350169(US10208056, Compound 1)copy SMILEScopy InChI
Affinity DataIC50: 2.59nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen. This is a kinase assay platform based on measuring the binding and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 8(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350266(US10208056, Compound 94)copy SMILEScopy InChI
Affinity DataIC50: 2.65nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen. This is a kinase assay platform based on measuring the binding and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetAcetylcholinesterase(Homo sapiens (Human))TBA
LigandPNGBDBM50556954(CHEMBL4782921)copy SMILES
Affinity DataIC50: 2.90nMAssay Description:Inhibition of recombinant human AChE using acetylthiocholineiodide as substrate preincubated for 20 mins followed by substrate addition by Ellman's m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K077XJPubMed
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350182(US10208056, Compound 14)copy SMILEScopy InChI
Affinity DataIC50: 3.01nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen). This is a kinase assay platform based on measuring the binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350252(US10208056, Compound 79)copy SMILEScopy InChI
Affinity DataIC50: 3.14nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen). This is a kinase assay platform based on measuring the binding an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 8(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350241(US10208056, Compound 68)copy SMILEScopy InChI
Affinity DataIC50: 3.23nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen. This is a kinase assay platform based on measuring the binding and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
TargetCyclin-C/Cyclin-dependent kinase 8(Homo sapiens (Human))
FUNDACIÓN DEL SECTOR PÚBLICO ESTATAL CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS CARLOS III (F.S.P. CNIO)

US Patent
LigandPNGBDBM350254(US10208056, Compound 81)copy SMILEScopy InChI
Affinity DataIC50: 3.83nMAssay Description:The binding assay relies on the LanthaScreen™ Eu-Kinase Binding Assay (Invitrogen. This is a kinase assay platform based on measuring the binding and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GB266BUS Patent
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