Compile Data Set for Download or QSAR
Found 176 with Last Name = 'aretz' and Initial = 'cd'
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50505262(CHEMBL4559408)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Inhibition of ROMK (unknown origin)More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9N7JPubMed
TargetG protein-activated inward rectifier potassium channel 4(Homo sapiens (Human))
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50505262(CHEMBL4559408)copy SMILEScopy InChI
Affinity DataKi:  8.20nMAssay Description:Inhibition GIRK1/4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9N7JPubMed
TargetTranslocator protein(Homo sapiens (Human))TBA
LigandPNGBDBM50605928(CHEMBL5195160)copy SMILES
Affinity DataKi:  71nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B06KQPubMed
TargetTranslocator protein(Homo sapiens (Human))TBA
LigandPNGBDBM50605927(CHEMBL5172913)copy SMILES
Affinity DataKi:  271nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B06KQPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50605954(CHEMBL5194692)copy SMILES
Affinity DataKi:  1.09E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B06KQPubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50605927(CHEMBL5172913)copy SMILES
Affinity DataKi: >4.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B06KQPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50605927(CHEMBL5172913)copy SMILES
Affinity DataKi: >4.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B06KQPubMed
TargetATP-sensitive inward rectifier potassium channel 1(Rattus norvegicus (Rat))
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM350315(US10208064, Example 30)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of rat ROMK1 expressed in HEK293 cells by Tl+ flux assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9N7JPubMed
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50505266(CHEMBL4548110)copy SMILEScopy InChI
Affinity DataIC50: 6.20nMAssay Description:Inhibition of human ROMK1 expressed in CHO cells by Tl+ flux assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9N7JPubMed
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50505267(CHEMBL4563446)copy SMILEScopy InChI
Affinity DataIC50: 6.60nMAssay Description:Inhibition of human ROMK1 expressed in CHO cells by Tl+ flux assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9N7JPubMed
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50505268(CHEMBL4549009)copy SMILEScopy InChI
Affinity DataIC50: 6.60nMAssay Description:Inhibition of human ROMK1 expressed in CHO cells by Tl+ flux assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9N7JPubMed
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50505271(CHEMBL4462473)copy SMILEScopy InChI
Affinity DataIC50: 8.80nMAssay Description:Inhibition of human ROMK1 expressed in CHO cells by Tl+ flux assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9N7JPubMed
TargetATP-sensitive inward rectifier potassium channel 1(Rattus norvegicus (Rat))
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM350282(US10208064, Example 2)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of rat ROMK1 expressed in HEK293 cells by Tl+ flux assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9N7JPubMed
TargetATP-sensitive inward rectifier potassium channel 1(Rattus norvegicus (Rat))
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM350300(US10208064, Example 19)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of rat ROMK1 expressed in HEK293 cells by Tl+ flux assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9N7JPubMed
TargetATP-sensitive inward rectifier potassium channel 1(Rattus norvegicus (Rat))
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50505263(CHEMBL4586813)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of rat ROMK1 expressed in HEK293 cells by Tl+ flux assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9N7JPubMed
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50505265(CHEMBL4465260)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Inhibition of human ROMK1 expressed in CHO cells by Tl+ flux assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9N7JPubMed
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50505270(CHEMBL4447159)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Inhibition of human ROMK1 expressed in CHO cells by Tl+ flux assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9N7JPubMed
TargetATP-sensitive inward rectifier potassium channel 1(Rattus norvegicus (Rat))
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50505261(CHEMBL4456474)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:Inhibition of rat ROMK1 expressed in HEK293 cells by Tl+ flux assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9N7JPubMed
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50204280(CHEMBL3987135 | US9573961, Example 15)copy SMILEScopy InChI
Affinity DataIC50: 57nMAssay Description:Inhibition of human ROMK1 expressed in HEK293 cells by Tl+ flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9N7JPubMed
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM290057(US9573961, Example 42)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of human ROMK1 expressed in HEK293 cells by Tl+ flux assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9N7JPubMed
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50505264(CHEMBL4544141)copy SMILEScopy InChI
Affinity DataIC50: 65nMAssay Description:Inhibition of human ROMK1 expressed in HEK293 cells by Tl+ flux assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9N7JPubMed
TargetATP-sensitive inward rectifier potassium channel 1(Homo sapiens (Human))
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50204281(CHEMBL3933749)copy SMILEScopy InChI
Affinity DataIC50: 73nMAssay Description:Inhibition of human ROMK1 expressed in HEK293 cells by Tl+ flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9N7JPubMed
LigandPNGBDBM14361((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged PDE4D3 expressed in baculovirus infected Sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
LigandPNGBDBM50561535(CHEMBL4762079)copy SMILES
Affinity DataIC50: 110nMAssay Description:Inhibition of recombinant human C-terminal His-tagged N-terminal GST-tagged PDE4B2 expressed in baculovirus infected Sf9 cells by radioligand binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J4PPubMed
LigandPNGBDBM14361((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibition of recombinant human C-terminal His-tagged N-terminal GST-tagged PDE4B2 expressed in baculovirus infected Sf9 cells by radioligand binding...More data for this Ligand-Target Pair
LigandPNGBDBM50561537(CHEMBL4783529)copy SMILES
Affinity DataIC50: 140nMAssay Description:Inhibition of recombinant human C-terminal His-tagged N-terminal GST-tagged PDE4B2 expressed in baculovirus infected Sf9 cells by radioligand binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J4PPubMed
LigandPNGBDBM50561545(CHEMBL4763078)copy SMILES
Affinity DataIC50: 210nMAssay Description:Inhibition of recombinant human C-terminal His-tagged N-terminal GST-tagged PDE4B2 expressed in baculovirus infected Sf9 cells by radioligand binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J4PPubMed
LigandPNGBDBM50561536(CHEMBL4781035)copy SMILES
Affinity DataIC50: 230nMAssay Description:Inhibition of recombinant human C-terminal His-tagged N-terminal GST-tagged PDE4B2 expressed in baculovirus infected Sf9 cells by radioligand binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J4PPubMed
TargetATP-sensitive inward rectifier potassium channel 1(Rattus norvegicus (Rat))
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50287521(CHEMBL2146753)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Inhibition of rat ROMK1 expressed in HEK293 cells by Tl+ flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9N7JPubMed
TargetATP-sensitive inward rectifier potassium channel 1(Rattus norvegicus (Rat))
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM73215(7,13-bis(4-nitrobenzyl)-1,4,10-trioxa-7,13-diazacy...)copy SMILEScopy InChI
Affinity DataIC50: 294nMAssay Description:Inhibition of rat ROMK1 expressed in HEK293 cells by Tl+ flux assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9N7JPubMed
LigandPNGBDBM50561556(CHEMBL4793481)copy SMILES
Affinity DataIC50: 410nMAssay Description:Inhibition of recombinant human C-terminal His-tagged N-terminal GST-tagged PDE4B2 expressed in baculovirus infected Sf9 cells by radioligand binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J4PPubMed
LigandPNGBDBM50561538(CHEMBL4759907)copy SMILES
Affinity DataIC50: 430nMAssay Description:Inhibition of recombinant human C-terminal His-tagged N-terminal GST-tagged PDE4B2 expressed in baculovirus infected Sf9 cells by radioligand binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J4PPubMed
LigandPNGBDBM50561548(CHEMBL4754568)copy SMILES
Affinity DataIC50: 430nMAssay Description:Inhibition of recombinant human C-terminal His-tagged N-terminal GST-tagged PDE4B2 expressed in baculovirus infected Sf9 cells by radioligand binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J4PPubMed
LigandPNGBDBM50561535(CHEMBL4762079)copy SMILES
Affinity DataIC50: 450nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged PDE4D3 expressed in baculovirus infected Sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J4PPubMed
LigandPNGBDBM50561532(CHEMBL4789557)copy SMILES
Affinity DataIC50: 480nMAssay Description:Inhibition of recombinant human C-terminal His-tagged N-terminal GST-tagged PDE4B2 expressed in baculovirus infected Sf9 cells by radioligand binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J4PPubMed
LigandPNGBDBM50561554(CHEMBL4786383)copy SMILES
Affinity DataIC50: 490nMAssay Description:Inhibition of recombinant human C-terminal His-tagged N-terminal GST-tagged PDE4B2 expressed in baculovirus infected Sf9 cells by radioligand binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J4PPubMed
LigandPNGBDBM50561534(CHEMBL4765220)copy SMILES
Affinity DataIC50: 600nMAssay Description:Inhibition of recombinant human C-terminal His-tagged N-terminal GST-tagged PDE4B2 expressed in baculovirus infected Sf9 cells by radioligand binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J4PPubMed
LigandPNGBDBM50561553(CHEMBL4758800)copy SMILES
Affinity DataIC50: 610nMAssay Description:Inhibition of recombinant human C-terminal His-tagged N-terminal GST-tagged PDE4B2 expressed in baculovirus infected Sf9 cells by radioligand binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J4PPubMed
LigandPNGBDBM355750(N-Cyclopropyl-3-(3,4-dichlorophenyl)-3H-imidazo[4,...)copy SMILEScopy InChI
Affinity DataIC50: 630nMAssay Description:Inhibition of recombinant human C-terminal His-tagged N-terminal GST-tagged PDE4B2 expressed in baculovirus infected Sf9 cells by radioligand binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J4PPubMed
LigandPNGBDBM355756(3-(3-Chloro-4-methylphenyl)-N-cyclopropyl-3H-imida...)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibition of recombinant human C-terminal His-tagged N-terminal GST-tagged PDE4B2 expressed in baculovirus infected Sf9 cells by radioligand binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J4PPubMed
LigandPNGBDBM50561537(CHEMBL4783529)copy SMILES
Affinity DataIC50: 880nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged PDE4D3 expressed in baculovirus infected Sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J4PPubMed
LigandPNGBDBM50561542(CHEMBL4797566)copy SMILES
Affinity DataIC50: 910nMAssay Description:Inhibition of recombinant human C-terminal His-tagged N-terminal GST-tagged PDE4B2 expressed in baculovirus infected Sf9 cells by radioligand binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J4PPubMed
LigandPNGBDBM50561551(CHEMBL4795799)copy SMILES
Affinity DataIC50: 970nMAssay Description:Inhibition of recombinant human C-terminal His-tagged N-terminal GST-tagged PDE4B2 expressed in baculovirus infected Sf9 cells by radioligand binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J4PPubMed
LigandPNGBDBM50561555(CHEMBL4758348)copy SMILES
Affinity DataIC50: 980nMAssay Description:Inhibition of recombinant human C-terminal His-tagged N-terminal GST-tagged PDE4B2 expressed in baculovirus infected Sf9 cells by radioligand binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J4PPubMed
LigandPNGBDBM50561539(CHEMBL4786718)copy SMILES
Affinity DataIC50: 980nMAssay Description:Inhibition of recombinant human C-terminal His-tagged N-terminal GST-tagged PDE4B2 expressed in baculovirus infected Sf9 cells by radioligand binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J4PPubMed
LigandPNGBDBM50561538(CHEMBL4759907)copy SMILES
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged PDE4D3 expressed in baculovirus infected Sf9 cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J4PPubMed
LigandPNGBDBM50561533(CHEMBL4763816)copy SMILES
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of recombinant human C-terminal His-tagged N-terminal GST-tagged PDE4B2 expressed in baculovirus infected Sf9 cells by radioligand binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J4PPubMed
LigandPNGBDBM50561544(CHEMBL4798020)copy SMILES
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of recombinant human C-terminal His-tagged N-terminal GST-tagged PDE4B2 expressed in baculovirus infected Sf9 cells by radioligand binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J4PPubMed
LigandPNGBDBM50561552(CHEMBL4763514)copy SMILES
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of recombinant human C-terminal His-tagged N-terminal GST-tagged PDE4B2 expressed in baculovirus infected Sf9 cells by radioligand binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J4PPubMed
LigandPNGBDBM50561543(CHEMBL4751002)copy SMILES
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of recombinant human C-terminal His-tagged N-terminal GST-tagged PDE4B2 expressed in baculovirus infected Sf9 cells by radioligand binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WM1J4PPubMed
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