TargetSolute carrier family 22 member 12(Homo sapiens (Human))
The Chinese University of Hong Kong
Curated by ChEMBL
The Chinese University of Hong Kong
Curated by ChEMBL
Affinity DataKi: 5.74E+3nMAssay Description:Inhibition of human URAT1-mediated urate uptake in HEK293 cells by competitive inhibition assayMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
The Chinese University of Hong Kong
Curated by ChEMBL
The Chinese University of Hong Kong
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of human URAT1-mediated urate uptake in HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
The Chinese University of Hong Kong
Curated by ChEMBL
The Chinese University of Hong Kong
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human URAT1-mediated urate uptake in HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Rattus norvegicus)
The Chinese University of Hong Kong
Curated by ChEMBL
The Chinese University of Hong Kong
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of human URAT1-mediated urate uptake in rat renal brush border membrane vesiclesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.42E+4nMAssay Description:Inhibition of xanthine oxidase (unknown origin) by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60E+4nMAssay Description:Inhibition of xanthine oxidase (unknown origin) by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 3.65E+4nMAssay Description:Inhibition of xanthine oxidase (unknown origin) by spectrophotometryMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
The Chinese University of Hong Kong
Curated by ChEMBL
The Chinese University of Hong Kong
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human URAT1-mediated urate uptake in HEK293 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
The Chinese University of Hong Kong
Curated by ChEMBL
The Chinese University of Hong Kong
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human URAT1-mediated urate uptake in HEK293 cellsMore data for this Ligand-Target Pair
![](/img/powered_by_small.gif)