Compile Data Set for Download or QSAR
Found 64 with Last Name = 'handscombe' and Initial = 'cm'
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085853(CHEMBL173251 | Sodium; [2-cyano-5-(pyridin-4-ylmet...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085845(CHEMBL174235 | [5-(Benzooxazol-6-ylmethoxy)-2-cyan...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085859((2-Chloro-phenyl)-[2-cyano-5-(pyridin-4-ylmethoxy)...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085833(CHEMBL172144 | Sodium; [5-(benzo[1,3]dioxol-5-ylme...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065518(4-[2-Cyano-5-(thiophen-3-ylmethoxy)-phenoxy]-4-o-t...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Concentration required to inhibit 50% Et-1 binding to endothelin A receptor in rat A-10 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN94SRPubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085861(CHEMBL170681 | [5-(Benzooxazol-6-ylmethoxy)-2-cyan...)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085831(CHEMBL174092 | [2-Cyano-5-(pyridin-4-ylmethoxy)-ph...)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085830(CHEMBL173792 | [5-(Benzo[1,3]dioxol-5-ylmethoxy)-2...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085838(CHEMBL352536 | [5-(Benzo[1,3]dioxol-5-ylmethoxy)-2...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085855(CHEMBL170202 | [5-(Benzo[1,3]dioxol-5-ylmethoxy)-2...)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085840((2-Chloro-phenyl)-[2-cyano-5-(thiophen-3-ylmethoxy...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085835(CHEMBL427294 | [2-Cyano-5-(thiophen-3-ylmethoxy)-p...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085854(CHEMBL171638 | [2-Cyano-5-(thiophen-3-ylmethoxy)-p...)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085832(CHEMBL171513 | [2-Cyano-5-(2-fluoro-pyridin-4-ylme...)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085839(CHEMBL170348 | [2-Cyano-5-(pyridin-3-ylmethoxy)-ph...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085864(CHEMBL354740 | [2-Cyano-5-(thiazol-5-ylmethoxy)-ph...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085856(CHEMBL355413 | [5-(Benzo[1,3]dioxol-5-ylmethoxy)-2...)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085858((2-Chloro-phenyl)-[2-cyano-5-(pyridazin-4-ylmethox...)copy SMILEScopy InChI
Affinity DataIC50: 44nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085860((5-Benzyloxy-2-cyano-phenoxy)-o-tolyl-acetic acid ...)copy SMILEScopy InChI
Affinity DataIC50: 49nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085844((2-Bromo-phenyl)-[2-cyano-5-(thiophen-3-ylmethoxy)...)copy SMILEScopy InChI
Affinity DataIC50: 51nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085837(CHEMBL170715 | [2-Cyano-5-(thiophen-3-ylmethoxy)-p...)copy SMILEScopy InChI
Affinity DataIC50: 53nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085836(CHEMBL172412 | [2-Cyano-5-(furan-3-ylmethoxy)-phen...)copy SMILEScopy InChI
Affinity DataIC50: 68nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085852(CHEMBL174229 | [2-Cyano-5-(thiophen-3-ylmethoxy)-p...)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085843(CHEMBL173444 | [5-(Benzooxazol-5-ylmethoxy)-2-cyan...)copy SMILEScopy InChI
Affinity DataIC50: 75nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065539((E)-3-[2-Cyano-5-(thiophen-3-ylmethoxy)-phenyl]-2-...)copy SMILEScopy InChI
Affinity DataIC50: 80nMAssay Description:Concentration required to inhibit 50% Et-1 binding to endothelin A receptor in rat A-10 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN94SRPubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085863((3-Chloro-phenyl)-[2-cyano-5-(thiophen-3-ylmethoxy...)copy SMILEScopy InChI
Affinity DataIC50: 98nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065533((E)-3-[2-Cyano-5-(pyridin-3-ylmethoxy)-phenyl]-2-p...)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Concentration required to inhibit 50% Et-1 binding to endothelin A receptor in rat A-10 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN94SRPubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065545((E)-2-Benzo[1,3]dioxol-5-yl-3-[2-cyano-5-(thiophen...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Concentration required to inhibit 50% Et-1 binding to endothelin A receptor in rat A-10 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN94SRPubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065548((E)-2-(2-Chloro-phenyl)-3-[2-cyano-5-(thiophen-3-y...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Concentration required to inhibit 50% Et-1 binding to endothelin A receptor in rat A-10 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN94SRPubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085862(CHEMBL366788 | [2-Cyano-5-(isothiazol-3-ylmethoxy)...)copy SMILEScopy InChI
Affinity DataIC50: 220nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065543(2-((E)-3-Hydroxy-2-o-tolyl-propenyl)-4-(thiophen-3...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Concentration required to inhibit 50% Et-1 binding to endothelin A receptor in rat A-10 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN94SRPubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065544((E)-3-[2-Cyano-5-(thiophen-3-ylmethoxy)-phenyl]-2-...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Concentration required to inhibit 50% Et-1 binding to endothelin A receptor in rat A-10 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN94SRPubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065537((E)-2-(2-Chloro-phenyl)-3-[2-nitro-5-(thiophen-3-y...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Concentration required to inhibit 50% Et-1 binding to endothelin A receptor in rat A-10 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN94SRPubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065528((E)-3-[2-Nitro-5-(thiophen-3-ylmethoxy)-phenyl]-2-...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Concentration required to inhibit 50% Et-1 binding to endothelin A receptor in rat A-10 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN94SRPubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085841((4-Chloro-phenyl)-[2-cyano-5-(thiophen-3-ylmethoxy...)copy SMILEScopy InChI
Affinity DataIC50: 504nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085848(CHEMBL172164 | [2-Cyano-5-(thiophen-3-ylmethoxy)-p...)copy SMILEScopy InChI
Affinity DataIC50: 529nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065540((E)-3-(5-Benzyloxy-2-nitro-phenyl)-2-phenyl-acryli...)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Concentration required to inhibit 50% Et-1 binding to endothelin A receptor in rat A-10 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN94SRPubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065531((E)-3-[2-Bromo-5-(thiophen-3-ylmethoxy)-phenyl]-2-...)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Concentration required to inhibit 50% Et-1 binding to endothelin A receptor in rat A-10 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN94SRPubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065550((E)-2-(2-Fluoro-phenyl)-3-[2-nitro-5-(thiophen-3-y...)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Concentration required to inhibit 50% Et-1 binding to endothelin A receptor in rat A-10 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN94SRPubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085850(CHEMBL172879 | [2-Cyano-5-(thiophen-3-ylmethoxy)-p...)copy SMILEScopy InChI
Affinity DataIC50: 630nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065549((Z)-5-[2-Cyano-5-(thiophen-3-ylmethoxy)-phenyl]-4-...)copy SMILEScopy InChI
Affinity DataIC50: 700nMAssay Description:Concentration required to inhibit 50% Et-1 binding to endothelin A receptor in rat A-10 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN94SRPubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065529((E)-3-[2-Bromo-5-(thiophen-3-ylmethoxy)-phenyl]-2-...)copy SMILEScopy InChI
Affinity DataIC50: 700nMAssay Description:Concentration required to inhibit 50% Et-1 binding to endothelin A receptor in rat A-10 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN94SRPubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065538(2-((E)-3-Hydroxy-2-phenyl-propenyl)-4-(thiophen-3-...)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Concentration required to inhibit 50% Et-1 binding to endothelin A receptor in rat A-10 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN94SRPubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50085846(CHEMBL173054 | [2-Cyano-5-(2,6-dimethyl-benzyloxy)...)copy SMILEScopy InChI
Affinity DataIC50: 857nMAssay Description:In vitro ability to antagonise the binding of [125I]-ET-1 to the rat aortic A10 cell membrane endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2154G73PubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065536((E)-3-(5-Benzyloxy-2-nitro-phenyl)-2-(2-fluoro-phe...)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Concentration required to inhibit 50% Et-1 binding to endothelin A receptor in rat A-10 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN94SRPubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065541(5-(3-Benzyloxy-phenyl)-5-oxo-4-phenyl-pentanoic ac...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Concentration required to inhibit 50% Et-1 binding to endothelin A receptor in rat A-10 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN94SRPubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065535((E)-3-[2-Cyano-5-(thiophen-3-ylmethoxy)-phenyl]-2-...)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Concentration required to inhibit 50% Et-1 binding to endothelin A receptor in rat A-10 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN94SRPubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065547((E)-2-(2-Chloro-phenyl)-3-[2-nitro-5-(thiophen-3-y...)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Concentration required to inhibit 50% Et-1 binding to endothelin A receptor in rat A-10 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN94SRPubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065532((E)-3-[5-(Benzo[1,3]dioxol-5-ylmethoxy)-2-cyano-ph...)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Concentration required to inhibit 50% Et-1 binding to endothelin A receptor in rat A-10 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN94SRPubMed
TargetEndothelin-1 receptor(RAT)
Rhône-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065542((E)-3-[2-Nitro-5-(thiophen-3-ylmethoxy)-phenyl]-2-...)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Concentration required to inhibit 50% Et-1 binding to endothelin A receptor in rat A-10 cells.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN94SRPubMed
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