Compile Data Set for Download or QSAR
Found 557 with Last Name = 'rominger' and Initial = 'cm'
TargetHexokinase-2(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50169013(CHEMBL3805703)copy SMILEScopy InChI
Affinity DataKi:  2.90E+3nMAssay Description:Competitive inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) assessed as formation of G6P by continuou...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PR7XWWPubMed
LigandPNGBDBM50420316(CHEMBL2089119)copy SMILEScopy InChI
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420311(CHEMBL2089114)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420321(CHEMBL2089112)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420309(CHEMBL2089120)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420310(CHEMBL2089116)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420317(CHEMBL2089118)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50489445(CHEMBL2322331)copy SMILEScopy InChI
Affinity DataIC50: 0.398nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7ZJTPubMed
LigandPNGBDBM50489439(CHEMBL2322340)copy SMILEScopy InChI
Affinity DataIC50: 0.398nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7ZJTPubMed
LigandPNGBDBM50381156(CHEMBL2018220 | D3RKN_94)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Inhibition of PI3Kbeta by continuous read time resolved fluorescence resonance energy transfer displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9ZBPPubMed
LigandPNGBDBM50420312(CHEMBL2089109)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420313(CHEMBL2089108)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420314(CHEMBL2089107)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420315(CHEMBL2089106)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50381161(CHEMBL2018219)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Inhibition of PI3Kbeta by continuous read time resolved fluorescence resonance energy transfer displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9ZBPPubMed
LigandPNGBDBM50489454(CHEMBL2322338)copy SMILEScopy InChI
Affinity DataIC50: 0.631nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7ZJTPubMed
LigandPNGBDBM50420315(CHEMBL2089106)copy SMILEScopy InChI
Affinity DataIC50: 0.631nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7ZJTPubMed
LigandPNGBDBM50381157(CHEMBL2018360)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of PI3Kbeta by continuous read time resolved fluorescence resonance energy transfer displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9ZBPPubMed
LigandPNGBDBM50489460(CHEMBL2322332)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7ZJTPubMed
LigandPNGBDBM50365868(CHEMBL1957857)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of PI3Kbeta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
LigandPNGBDBM50365882(CHEMBL1957870)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of PI3Kbeta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
LigandPNGBDBM50365868(CHEMBL1957857)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of PI3Kbeta by continuous read time resolved fluorescence resonance energy transfer displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9ZBPPubMed
LigandPNGBDBM50381164(CHEMBL2018214)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of PI3Kbeta by continuous read time resolved fluorescence resonance energy transfer displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9ZBPPubMed
LigandPNGBDBM50381158(CHEMBL2018222)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of PI3Kbeta by continuous read time resolved fluorescence resonance energy transfer displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9ZBPPubMed
LigandPNGBDBM50489452(CHEMBL2322344)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7ZJTPubMed
LigandPNGBDBM50381158(CHEMBL2018222)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of PI3Kbeta by continuous read time resolved fluorescence resonance energy transfer displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9ZBPPubMed
LigandPNGBDBM50381162(CHEMBL2018221)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of PI3Kbeta by continuous read time resolved fluorescence resonance energy transfer displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9ZBPPubMed
LigandPNGBDBM50381161(CHEMBL2018219)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Inhibition of PI3K beta-mediated AKT phosphorylation at serine 473 in PTEN deficient human MDA-MB-468 cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9ZBPPubMed
LigandPNGBDBM50381165(CHEMBL2018215)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of PI3Kbeta by continuous read time resolved fluorescence resonance energy transfer displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9ZBPPubMed
LigandPNGBDBM50420311(CHEMBL2089114)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of PI3K delta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420316(CHEMBL2089119)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of PI3K delta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50381159(CHEMBL2018217)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of PI3Kbeta by continuous read time resolved fluorescence resonance energy transfer displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9ZBPPubMed
LigandPNGBDBM50365869(CHEMBL1957858)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of PI3Kbeta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
LigandPNGBDBM50365867(CHEMBL1957856)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of PI3Kbeta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
LigandPNGBDBM50381163(CHEMBL2018361)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of PI3Kbeta by continuous read time resolved fluorescence resonance energy transfer displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9ZBPPubMed
LigandPNGBDBM50381159(CHEMBL2018217)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of PI3Kbeta by continuous read time resolved fluorescence resonance energy transfer displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9ZBPPubMed
LigandPNGBDBM50489444(CHEMBL2322335)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7ZJTPubMed
LigandPNGBDBM50381155(CHEMBL2018216)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Inhibition of PI3Kbeta by continuous read time resolved fluorescence resonance energy transfer displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9ZBPPubMed
LigandPNGBDBM50489455(CHEMBL2322337)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7ZJTPubMed
LigandPNGBDBM50489450(CHEMBL2322341)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Inhibition of PI3Kbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7ZJTPubMed
LigandPNGBDBM50381158(CHEMBL2018222)copy SMILEScopy InChI
Affinity DataIC50: 2.70nMAssay Description:Inhibition of PI3K beta-mediated AKT phosphorylation at serine 473 in PTEN deficient human MDA-MB-468 cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9ZBPPubMed
LigandPNGBDBM50381158(CHEMBL2018222)copy SMILEScopy InChI
Affinity DataIC50: 2.70nMAssay Description:Inhibition of PI3K beta-mediated AKT phosphorylation at serine 473 in PTEN deficient human MDA-MB-468 cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TD9ZBPPubMed
LigandPNGBDBM50420320(CHEMBL2089113)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50365882(CHEMBL1957870)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of PI3Kdelta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
LigandPNGBDBM50420325(CHEMBL2089104)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420324(CHEMBL2089105)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50420322(CHEMBL2089111)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of PI3K beta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
LigandPNGBDBM50365866(CHEMBL1957855)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of PI3Kbeta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
LigandPNGBDBM50365865(CHEMBL1957841)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of PI3Kbeta by time-resolved FRET displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9JF0PubMed
LigandPNGBDBM50420309(CHEMBL2089120)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of PI3K delta by continuous TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J967PTPubMed
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