Compile Data Set for Download or QSAR
Found 46 with Last Name = 'adpressa' and Initial = 'd'
LigandPNGBDBM50584324(CHEMBL5088471)copy SMILES
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584317(CHEMBL5082260)copy SMILES
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584331(CHEMBL5079796)copy SMILES
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584330(CHEMBL5070497)copy SMILES
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584328(CHEMBL5078277 | US20230303540, Example Ex-1.48)copy SMILES
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584325(CHEMBL5085777)copy SMILES
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584321(CHEMBL5090739)copy SMILES
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584318(CHEMBL5082563)copy SMILES
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584332(CHEMBL5076397)copy SMILES
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584316(CHEMBL5070231)copy SMILES
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584322(CHEMBL5089102)copy SMILES
Affinity DataIC50: 0.650nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584326(CHEMBL5094138)copy SMILES
Affinity DataIC50: 0.700nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584320(CHEMBL5073571)copy SMILES
Affinity DataIC50: 0.800nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584329(CHEMBL5089933)copy SMILES
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579614(CHEMBL4871970)copy SMILES
Affinity DataIC50: 1.60nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
LigandPNGBDBM50584327(CHEMBL5073735)copy SMILES
Affinity DataIC50: 1.70nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579610(CHEMBL4873520)copy SMILES
Affinity DataIC50: 2.20nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
LigandPNGBDBM50584319(CHEMBL5085536 | US20230303540, Example Ex-1.24)copy SMILES
Affinity DataIC50: 2.60nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579616(CHEMBL4845730)copy SMILES
Affinity DataIC50: 3.20nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579611(CHEMBL4871097)copy SMILES
Affinity DataIC50: 3.90nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579615(CHEMBL4865209)copy SMILES
Affinity DataIC50: 5nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
LigandPNGBDBM50584333(CHEMBL5093254)copy SMILES
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50577458(CHEMBL4858437)copy SMILES
Affinity DataIC50: 16nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579613(CHEMBL4850423)copy SMILES
Affinity DataIC50: 25nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579609(CHEMBL4872874)copy SMILES
Affinity DataIC50: 46nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579618(CHEMBL4871090)copy SMILES
Affinity DataIC50: 67nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579612(CHEMBL4847500)copy SMILES
Affinity DataIC50: 104nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579608(CHEMBL4849969)copy SMILES
Affinity DataIC50: 370nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
LigandPNGBDBM50584335(CHEMBL5076674)copy SMILES
Affinity DataIC50: 570nMAssay Description:Inhibition of human ERG by voltage clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
TargetMitogen-activated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50584332(CHEMBL5076397)copy SMILES
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of ERK1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584321(CHEMBL5090739)copy SMILES
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of human ERG by voltage clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
TargetSubstance-P receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50584332(CHEMBL5076397)copy SMILES
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of tachykinin NK1 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
TargetMAP/microtubule affinity-regulating kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50584334(CHEMBL5075047)copy SMILES
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of MARK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579617(CHEMBL4863411)copy SMILES
Affinity DataIC50: 5.74E+3nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
LigandPNGBDBM50584334(CHEMBL5075047)copy SMILES
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of human ERG by voltage clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584323(CHEMBL5074799)copy SMILES
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of recombinant N-terminal GST-fused LRRK2 G2109S mutant (970 to 2527 residues) (unknown origin) preincubated with enzyme for 15 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584331(CHEMBL5079796)copy SMILES
Affinity DataIC50: 8.60E+3nMAssay Description:Inhibition of human ERG by voltage clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579607(CHEMBL4865167)copy SMILES
Affinity DataIC50: 8.78E+3nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
LigandPNGBDBM50584332(CHEMBL5076397)copy SMILES
Affinity DataIC50: 9.70E+3nMAssay Description:Inhibition of human ERG by voltage clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50579606(CHEMBL4851004)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8XQ7PubMed
LigandPNGBDBM50584318(CHEMBL5082563)copy SMILES
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of human ERG by voltage clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584322(CHEMBL5089102)copy SMILES
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of human ERG by voltage clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584316(CHEMBL5070231)copy SMILES
Affinity DataIC50: 1.83E+4nMAssay Description:Inhibition of human ERG by voltage clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584320(CHEMBL5073571)copy SMILES
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of human ERG by voltage clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584319(CHEMBL5085536 | US20230303540, Example Ex-1.24)copy SMILES
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of human ERG by voltage clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed
LigandPNGBDBM50584330(CHEMBL5070497)copy SMILES
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of human ERG by voltage clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GZHPubMed