Compile Data Set for Download or QSAR
Found 310 with Last Name = 'cashion' and Initial = 'd'
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50512318(CHEMBL4546504)copy SMILEScopy InChI
Affinity DataIC50: 0.00100nMAssay Description:Inhibition of recombinant human GST-tagged LRRK2 G2019S mutant catalytic domain (970 to 2527 residues) expressed in baculovirus expression system usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6VVNPubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50512318(CHEMBL4546504)copy SMILEScopy InChI
Affinity DataIC50: 0.00100nMAssay Description:Inhibition of recombinant human GST-tagged LRRK2 catalytic domain (970 to 2527 residues) expressed in baculovirus expression system using LRRKtide as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6VVNPubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50512318(CHEMBL4546504)copy SMILEScopy InChI
Affinity DataIC50: 0.0320nMAssay Description:Inhibition of recombinant human full length His-tagged JNK1 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6VVNPubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50512318(CHEMBL4546504)copy SMILEScopy InChI
Affinity DataIC50: 0.0590nMAssay Description:Inhibition of recombinant human full length His-tagged JNK2 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6VVNPubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 3(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50512318(CHEMBL4546504)copy SMILEScopy InChI
Affinity DataIC50: 0.104nMAssay Description:Inhibition of recombinant human full length GST-tagged DYRK3 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6VVNPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50512318(CHEMBL4546504)copy SMILEScopy InChI
Affinity DataIC50: 0.107nMAssay Description:Inhibition of recombinant human full length N-terminal GST-tagged JNK3 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6VVNPubMed
TargetTestis-specific serine/threonine-protein kinase 1(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50512318(CHEMBL4546504)copy SMILEScopy InChI
Affinity DataIC50: 0.217nMAssay Description:Inhibition of recombinant human full length His-tagged TSSK1 expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6VVNPubMed
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50512318(CHEMBL4546504)copy SMILEScopy InChI
Affinity DataIC50: 0.261nMAssay Description:Inhibition of recombinant human GST-tagged CLK2 catalytic domain (137 to 498 residues) expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6VVNPubMed
TargetProtein kinase C theta type(Homo sapiens (Human))TBA
LigandPNGBDBM251460(US9452998, 9)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Inhibition of PKA-theta (unknown origin) using Fam-labelled S6-derived peptide incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6GPSPubMed
TargetLeukocyte tyrosine kinase receptor(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50512318(CHEMBL4546504)copy SMILEScopy InChI
Affinity DataIC50: 0.567nMAssay Description:Inhibition of recombinant human GST-tagged LTK cytoplasmic domain (450 to 864 residues) expressed in baculovirus expression system by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6VVNPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50512326(CHEMBL4476012)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Inhibition of Kinase Tracer 236 binding to recombinant human full-length GST-tagged TTk expressed in baculovirus expression system measured after 1 h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6VVNPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50512318(CHEMBL4546504)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:Inhibition of Kinase Tracer 236 binding to recombinant human full-length GST-tagged TTk expressed in baculovirus expression system measured after 1 h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50512322(CHEMBL4450891)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:Inhibition of Kinase Tracer 236 binding to recombinant human full-length GST-tagged TTk expressed in baculovirus expression system measured after 1 h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6VVNPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM532292(JGS79C | N-(2,6-diethylphenyl)-2-[2-methoxy-4-(4-m...)copy SMILES
Affinity DataIC50: 0.900nMAssay Description:Inhibition of full length TTK (unknown origin) using MBP-derived peptide as substrate preincubated for 1 hr in dark followed by substrate addition an...More data for this Ligand-Target Pair
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50582063(CHEMBL5092826)copy SMILES
Affinity DataIC50: 1nMAssay Description:Displacement of kinase tracer 236 from TTK (unknown origin) by LanthaScreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3QC6PubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50512321(CHEMBL4472951)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of Kinase Tracer 236 binding to recombinant human full-length GST-tagged TTk expressed in baculovirus expression system measured after 1 h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6VVNPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50582067(CHEMBL5093015)copy SMILES
Affinity DataIC50: 1nMAssay Description:Displacement of kinase tracer 236 from TTK (unknown origin) by LanthaScreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3QC6PubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50512323(CHEMBL4558047)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of Kinase Tracer 236 binding to recombinant human full-length GST-tagged TTk expressed in baculovirus expression system measured after 1 h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6VVNPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50512325(CHEMBL4585148)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of Kinase Tracer 236 binding to recombinant human full-length GST-tagged TTk expressed in baculovirus expression system measured after 1 h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6VVNPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50512316(CHEMBL4530475)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of Kinase Tracer 236 binding to recombinant human full-length GST-tagged TTk expressed in baculovirus expression system measured after 1 h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6VVNPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50512324(CHEMBL4521278)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of Kinase Tracer 236 binding to recombinant human full-length GST-tagged TTk expressed in baculovirus expression system measured after 1 h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6VVNPubMed
TargetProtein kinase C theta type(Homo sapiens (Human))TBA
LigandPNGBDBM50573043(CHEMBL4849510)copy SMILES
Affinity DataIC50: 1.30nMAssay Description:Inhibition of PKA-theta (unknown origin) using Fam-labelled S6-derived peptide incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6GPSPubMed
TargetProtein kinase C theta type(Homo sapiens (Human))TBA
LigandPNGBDBM50573038(CHEMBL4853353)copy SMILES
Affinity DataIC50: 1.40nMAssay Description:Inhibition of PKA-theta (unknown origin) using Fam-labelled S6-derived peptide incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6GPSPubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))TBA
LigandPNGBDBM251460(US9452998, 9)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Inhibition of PKC-alpha (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50582061(CHEMBL5081270)copy SMILES
Affinity DataIC50: 2nMAssay Description:Displacement of kinase tracer 236 from TTK (unknown origin) by LanthaScreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3QC6PubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50582069(CHEMBL5073101)copy SMILES
Affinity DataIC50: 2nMAssay Description:Displacement of kinase tracer 236 from TTK (unknown origin) by LanthaScreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3QC6PubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50582068(CHEMBL5077668)copy SMILES
Affinity DataIC50: 2nMAssay Description:Displacement of kinase tracer 236 from TTK (unknown origin) by LanthaScreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3QC6PubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50582065(CHEMBL5075313)copy SMILES
Affinity DataIC50: 2nMAssay Description:Displacement of kinase tracer 236 from TTK (unknown origin) by LanthaScreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3QC6PubMed
TargetProtein kinase C theta type(Homo sapiens (Human))TBA
LigandPNGBDBM50573042(CHEMBL4854104)copy SMILES
Affinity DataIC50: 2.20nMAssay Description:Inhibition of PKA-theta (unknown origin) using Fam-labelled S6-derived peptide incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6GPSPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50512317(CHEMBL4569626)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Inhibition of Kinase Tracer 236 binding to recombinant human full-length GST-tagged TTk expressed in baculovirus expression system measured after 1 h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6VVNPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50582074(CHEMBL5081668)copy SMILES
Affinity DataIC50: 2.80nMAssay Description:Displacement of kinase tracer 236 from TTK (unknown origin) by LanthaScreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3QC6PubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50582066(CHEMBL5084062)copy SMILES
Affinity DataIC50: 3nMAssay Description:Displacement of kinase tracer 236 from TTK (unknown origin) by LanthaScreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3QC6PubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50582077(CHEMBL5085753)copy SMILES
Affinity DataIC50: 3nMAssay Description:Displacement of kinase tracer 236 from TTK (unknown origin) by LanthaScreen Eu kinase binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3QC6PubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50582064(CHEMBL5091689)copy SMILES
Affinity DataIC50: 3nMAssay Description:Displacement of kinase tracer 236 from TTK (unknown origin) by LanthaScreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3QC6PubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50512320(CHEMBL4467041)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Inhibition of Kinase Tracer 236 binding to recombinant human full-length GST-tagged TTk expressed in baculovirus expression system measured after 1 h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6VVNPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50582071(CHEMBL5086022)copy SMILES
Affinity DataIC50: 4nMAssay Description:Displacement of kinase tracer 236 from TTK (unknown origin) by LanthaScreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3QC6PubMed
TargetProtein kinase C theta type(Homo sapiens (Human))TBA
LigandPNGBDBM50573034(CHEMBL4859091)copy SMILES
Affinity DataIC50: 4nMAssay Description:Inhibition of PKA-theta (unknown origin) using Fam-labelled S6-derived peptide incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6GPSPubMed
TargetProtein kinase C theta type(Homo sapiens (Human))TBA
LigandPNGBDBM50572994(CHEMBL4854326)copy SMILES
Affinity DataIC50: 4nMAssay Description:Inhibition of PKA-theta (unknown origin) using Fam-labelled S6-derived peptide incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6GPSPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50582070(CHEMBL5085278)copy SMILES
Affinity DataIC50: 4nMAssay Description:Displacement of kinase tracer 236 from TTK (unknown origin) by LanthaScreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3QC6PubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM317462(4-(4-(cyclopentyloxy)-5-(2- methylbenzo[d]oxazol-6...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of human full length recombinant GST-tagged TTK expressed in baculovirus by LanthaScreen Eu kinase binding assayMore data for this Ligand-Target Pair
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50582076(CHEMBL5079606)copy SMILES
Affinity DataIC50: 5.30nMAssay Description:Displacement of kinase tracer 236 from TTK (unknown origin) by LanthaScreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3QC6PubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50582075(CHEMBL5085182)copy SMILES
Affinity DataIC50: 5.60nMAssay Description:Displacement of kinase tracer 236 from TTK (unknown origin) by LanthaScreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3QC6PubMed
TargetProtein kinase C theta type(Homo sapiens (Human))TBA
LigandPNGBDBM50573033(CHEMBL4851695)copy SMILES
Affinity DataIC50: 6nMAssay Description:Inhibition of PKA-theta (unknown origin) using Fam-labelled S6-derived peptide incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6GPSPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50582062(CHEMBL5086435)copy SMILES
Affinity DataIC50: 6nMAssay Description:Displacement of kinase tracer 236 from TTK (unknown origin) by LanthaScreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3QC6PubMed
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM317462(4-(4-(cyclopentyloxy)-5-(2- methylbenzo[d]oxazol-6...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of human GST-tagged CLK2 expressed in baculovirus by Z'-LYTE assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0WX9PubMed
TargetProtein kinase C theta type(Homo sapiens (Human))TBA
LigandPNGBDBM50573015(CHEMBL4870774)copy SMILES
Affinity DataIC50: 7nMAssay Description:Inhibition of PKA-theta (unknown origin) using Fam-labelled S6-derived peptide incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6GPSPubMed
TargetProtein kinase C theta type(Homo sapiens (Human))TBA
LigandPNGBDBM50573029(CHEMBL4861883)copy SMILES
Affinity DataIC50: 7nMAssay Description:Inhibition of PKA-theta (unknown origin) using Fam-labelled S6-derived peptide incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6GPSPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50512319(CHEMBL4547530)copy SMILEScopy InChI
Affinity DataIC50: 7.20nMAssay Description:Inhibition of Kinase Tracer 236 binding to recombinant human full-length GST-tagged TTk expressed in baculovirus expression system measured after 1 h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6VVNPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Celgene Corporation

Curated by ChEMBL
LigandPNGBDBM50582073(CHEMBL5077627)copy SMILES
Affinity DataIC50: 7.5nMAssay Description:Displacement of kinase tracer 236 from TTK (unknown origin) by LanthaScreen Eu kinase binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3QC6PubMed
TargetProtein kinase C theta type(Homo sapiens (Human))TBA
LigandPNGBDBM50573044(CHEMBL4873647)copy SMILES
Affinity DataIC50: 8nMAssay Description:Inhibition of PKA-theta (unknown origin) using Fam-labelled S6-derived peptide incubated for 2 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6GPSPubMed
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