Affinity DataKi: 0.200nM ΔG°: -54.8kJ/molepH: 7.2 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 0.200nM ΔG°: -54.8kJ/molepH: 7.2 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.320nM ΔG°: -53.6kJ/molepH: 7.2 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Lundbeck Research USA, Inc.
Curated by ChEMBL
Lundbeck Research USA, Inc.
Curated by ChEMBL
Affinity DataKi: 0.460nMAssay Description:Binding affinity for human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.620nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.790nM ΔG°: -51.4kJ/molepH: 7.2 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Lundbeck Research USA, Inc.
Curated by ChEMBL
Lundbeck Research USA, Inc.
Curated by ChEMBL
Affinity DataKi: 0.830nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Lundbeck Research USA, Inc.
Curated by ChEMBL
Lundbeck Research USA, Inc.
Curated by ChEMBL
Affinity DataKi: 0.950nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nM ΔG°: -50.4kJ/molepH: 7.2 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Lundbeck Research USA, Inc.
Curated by ChEMBL
Lundbeck Research USA, Inc.
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Lundbeck Research USA, Inc.
Curated by ChEMBL
Lundbeck Research USA, Inc.
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nM ΔG°: -49.7kJ/molepH: 7.2 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Lundbeck Research USA, Inc.
Curated by ChEMBL
Lundbeck Research USA, Inc.
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nM ΔG°: -49.2kJ/molepH: 7.2 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3nM ΔG°: -48.2kJ/molepH: 7.2 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 3nM ΔG°: -48.2kJ/molepH: 7.2 T: 2°CAssay Description:IC50 values for test compounds were determined from nonlinear regression analysis of data collected from ligand displacement experiments. The inhibit...More data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Binding affinity for rat Dopamine receptor D3More data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Binding affinity for rat Dopamine receptor D3More data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Lundbeck Research USA, Inc.
Curated by ChEMBL
Lundbeck Research USA, Inc.
Curated by ChEMBL
Affinity DataKi: 5.60nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.5nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Lundbeck Research USA, Inc.
Curated by ChEMBL
Lundbeck Research USA, Inc.
Curated by ChEMBL
Affinity DataKi: 7.5nMAssay Description:Binding affinity for human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Lundbeck Research USA, Inc.
Curated by ChEMBL
Lundbeck Research USA, Inc.
Curated by ChEMBL
Affinity DataKi: 7.90nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8.10nMAssay Description:Binding affinity for rat Dopamine receptor D3More data for this Ligand-Target Pair
Affinity DataKi: 8.20nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8.5nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Lundbeck Research USA, Inc.
Curated by ChEMBL
Lundbeck Research USA, Inc.
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity for human Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding affinity for rat Dopamine receptor D3More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Lundbeck Research USA, Inc.
Curated by ChEMBL
Lundbeck Research USA, Inc.
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Binding affinity for human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
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