TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 630nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 760nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 820nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 860nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 1.31E+3nMAssay Description:Blockade of synaptosomal sodium channels, inhibition of [14C]-guanidinium ion flux into CHO cells expressing Type II sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 1.39E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 1.48E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 1.51E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 1.75E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 1.76E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 1.76E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 1.92E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 1.95E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 1.97E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 2.02E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 2.03E+3nMAssay Description:Blockade of synaptosomal sodium channels, inhibition of [14C]-guanidinium ion flux into CHO cells expressing Type II sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 2.11E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Blockade of synaptosomal sodium channels, inhibition of [14C]-guanidinium ion flux into CHO cells expressing Type II sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 2.35E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 2.38E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 2.55E+3nMAssay Description:Blockade of synaptosomal sodium channels, inhibition of [14C]-guanidinium ion flux into CHO cells expressing Type II sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 2.66E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 2.67E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 2.71E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 2.85E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 3.23E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 3.25E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 3.29E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 3.35E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 3.87E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 3.92E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 4.16E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 4.31E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 4.36E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 4.95E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 5.03E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 5.25E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing human cardiac (hHI) sodium channelMore data for this Ligand-Target Pair
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
CeNeS Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 5.44E+3nMAssay Description:Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channelMore data for this Ligand-Target Pair
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