Compile Data Set for Download or QSAR
Found 292 with Last Name = 'feldman' and Initial = 'd'
TargetSigma non-opioid intracellular receptor 1(RAT)
Hoechst Marion Roussel, Inc.

Curated by PDSP Ki Database
LigandPNGBDBM50095027((2,3-Dimethoxy-phenyl)-{1-[2-(4-fluoro-phenyl)-eth...)copy SMILEScopy InChI
Affinity DataKi:  87nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FN14R3PubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Hoechst Marion Roussel, Inc.

Curated by PDSP Ki Database
LigandPNGBDBM50095027((2,3-Dimethoxy-phenyl)-{1-[2-(4-fluoro-phenyl)-eth...)copy SMILEScopy InChI
Affinity DataKi:  88nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FN14R3PubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Hoechst Marion Roussel, Inc.

Curated by PDSP Ki Database
LigandPNGBDBM50095027((2,3-Dimethoxy-phenyl)-{1-[2-(4-fluoro-phenyl)-eth...)copy SMILEScopy InChI
Affinity DataKi:  128nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FN14R3PubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Hoechst Marion Roussel, Inc.

Curated by PDSP Ki Database
LigandPNGBDBM50095027((2,3-Dimethoxy-phenyl)-{1-[2-(4-fluoro-phenyl)-eth...)copy SMILEScopy InChI
Affinity DataKi:  540nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FN14R3PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Hoechst Marion Roussel, Inc.

Curated by PDSP Ki Database
LigandPNGBDBM50095027((2,3-Dimethoxy-phenyl)-{1-[2-(4-fluoro-phenyl)-eth...)copy SMILEScopy InChI
Affinity DataKi:  2.25E+3nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FN14R3PubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Hoechst Marion Roussel, Inc.

Curated by PDSP Ki Database
LigandPNGBDBM50095027((2,3-Dimethoxy-phenyl)-{1-[2-(4-fluoro-phenyl)-eth...)copy SMILEScopy InChI
Affinity DataKi:  5.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FN14R3PubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Hoechst Marion Roussel, Inc.

Curated by PDSP Ki Database
LigandPNGBDBM50095027((2,3-Dimethoxy-phenyl)-{1-[2-(4-fluoro-phenyl)-eth...)copy SMILEScopy InChI
Affinity DataKi:  6.70E+3nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FN14R3PubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Hoechst Marion Roussel, Inc.

Curated by PDSP Ki Database
LigandPNGBDBM50095027((2,3-Dimethoxy-phenyl)-{1-[2-(4-fluoro-phenyl)-eth...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FN14R3PubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50542738(CHEMBL4637027)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human F11a using D-Leu-Pro-Arg*Rh110-D-Pro as substrate preincubated for 60 mins followed by substrate addition and measured after 60 m...More data for this Ligand-Target Pair
TargetCoagulation factor XI(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50542741(CHEMBL4647950)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:Inhibition of human F11a using D-Leu-Pro-Arg*Rh110-D-Pro as substrate preincubated for 60 mins followed by substrate addition and measured after 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6W36PubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50542731(CHEMBL4642845)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:Inhibition of human F11a using D-Leu-Pro-Arg*Rh110-D-Pro as substrate preincubated for 60 mins followed by substrate addition and measured after 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6W36PubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107813((S)-methyl 5-(6-methyl-4'-(trifluoromethyl)bipheny...)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107808(6-Methyl-4'-trifluoromethyl-biphenyl-2-carboxylic ...)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107774(4,6-Dimethyl-4'-trifluoromethyl-biphenyl-2-carboxy...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetPlasma kallikrein(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50542738(CHEMBL4637027)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of PKL (unknown origin) using D-Leu-Pro-Arg*Rh110-D-Pro as substrate preincubated for 60 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6W36PubMed
TargetPlasma kallikrein(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50542731(CHEMBL4642845)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of PKL (unknown origin) using D-Leu-Pro-Arg*Rh110-D-Pro as substrate preincubated for 60 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6W36PubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107809(CHEMBL143284 | {5-[(4,6-Dimethyl-4'-trifluoromethy...)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107797(4'-Fluoro-6-methyl-biphenyl-2-carboxylic acid (2-b...)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107790(4'-Trifluoromethyl-biphenyl-2-carboxylic acid (2-b...)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107772(4'-Fluoro-6-methyl-biphenyl-2-carboxylic acid [2-(...)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107804(CHEMBL142975 | {2-[(6-Methyl-4'-trifluoromethyl-bi...)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107803(6-Methyl-4'-trifluoromethyl-biphenyl-2-carboxylic ...)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107787((S)-6-methyl-N-(2-(pyridin-2-ylmethylamino)-2,3-di...)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107810(6-Methyl-4'-trifluoromethyl-biphenyl-2-carboxylic ...)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107775(4-{5-[(6-Methyl-4'-trifluoromethyl-biphenyl-2-carb...)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107812(CHEMBL142928 | {5-[(6,4'-Bis-trifluoromethyl-biphe...)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107815(6-Methyl-4'-trifluoromethyl-biphenyl-2-carboxylic ...)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107798(CHEMBL139992 | {5-[(4'-Trifluoromethyl-biphenyl-2-...)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107800(CHEMBL356126 | {2-[(4'-Chloro-6-methyl-biphenyl-2-...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107802(4'-Chloro-6-methoxy-biphenyl-2-carboxylic acid (2-...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetPlasma kallikrein(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50542740(CHEMBL4646398)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of PKL (unknown origin) using D-Leu-Pro-Arg*Rh110-D-Pro as substrate preincubated for 60 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6W36PubMed
TargetPlasma kallikrein(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50542724(CHEMBL4636415)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of PKL (unknown origin) using D-Leu-Pro-Arg*Rh110-D-Pro as substrate preincubated for 60 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6W36PubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50542740(CHEMBL4646398)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of human F11a using D-Leu-Pro-Arg*Rh110-D-Pro as substrate preincubated for 60 mins followed by substrate addition and measured after 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6W36PubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107788(CHEMBL143514 | {5-[(4-Methyl-4'-trifluoromethyl-bi...)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107811(CHEMBL142733 | {5-[(4,6-Dimethyl-4'-trifluoromethy...)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107805(6-Methyl-4'-trifluoromethyl-biphenyl-2-carboxylic ...)copy SMILEScopy InChI
Affinity DataIC50: 2.30nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107792(4'-Chloro-6-methyl-biphenyl-2-carboxylic acid (2-b...)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107785(CHEMBL341974 | {2-[(4,6-Dimethyl-4'-trifluoromethy...)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107793(CHEMBL358141 | {5-[(4,6-Dimethyl-4'-trifluoromethy...)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107781(6,4'-Dimethyl-biphenyl-2-carboxylic acid (2-benzen...)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107777(4,6-Dimethyl-4'-trifluoromethyl-biphenyl-2-carboxy...)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50542723(CHEMBL4643449)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of human F11a using D-Leu-Pro-Arg*Rh110-D-Pro as substrate preincubated for 60 mins followed by substrate addition and measured after 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6W36PubMed
TargetPlasma kallikrein(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50542723(CHEMBL4643449)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of PKL (unknown origin) using D-Leu-Pro-Arg*Rh110-D-Pro as substrate preincubated for 60 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6W36PubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50542733(CHEMBL4646141)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of human F11a using D-Leu-Pro-Arg*Rh110-D-Pro as substrate preincubated for 60 mins followed by substrate addition and measured after 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107770(4'-Chloro-6-methyl-biphenyl-2-carboxylic acid [2-(...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50542728(CHEMBL4635912)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of human F11a using D-Leu-Pro-Arg*Rh110-D-Pro as substrate preincubated for 60 mins followed by substrate addition and measured after 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6W36PubMed
TargetApolipoprotein B-100(Homo sapiens (Human))
Novartis Institute for Biomedical Reasearch

Curated by ChEMBL
LigandPNGBDBM50107783(CHEMBL343837 | {5-[(4'-Chloro-4,6-dimethyl-bipheny...)copy SMILEScopy InChI
Affinity DataIC50: 3.40nMAssay Description:Inhibition of apolipoprotein B (apoB) secreted by human hepatoma cells (Hep G2) at 100 nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23F4NXHPubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50542724(CHEMBL4636415)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of human F11a using D-Leu-Pro-Arg*Rh110-D-Pro as substrate preincubated for 60 mins followed by substrate addition and measured after 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPlasma kallikrein(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50542730(CHEMBL4647909)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of PKL (unknown origin) using D-Leu-Pro-Arg*Rh110-D-Pro as substrate preincubated for 60 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6W36PubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50542725(CHEMBL4637683)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of human F11a using D-Leu-Pro-Arg*Rh110-D-Pro as substrate preincubated for 60 mins followed by substrate addition and measured after 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KS6W36PubMed
Displayed 1 to 50 (of 292 total ) | Next | Last >>
Jump to: