Compile Data Set for Download or QSAR
Found 221 with Last Name = 'gianni' and Initial = 'd'
TargetBromodomain-containing protein 4 [42-168](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM209487(US10328074, Example III-28 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:This assay is used to determine whether the compounds inhibit the interaction between the first (BRD4-BD1) or the second (BRD4-BD2) bromodomain of BR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z75M2US Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))TBA
LigandPNGBDBM209487(US10328074, Example III-28 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PV6PHQUS Patent
TargetBromodomain-containing protein 4 [44-168]/Histone H4(Homo sapiens (Human))
Boehringer Ingelheim International GmbH

US Patent
LigandPNGBDBM209487(US10328074, Example III-28 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 uM start concentration) in white OptiPlate-384 (PerkinElme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23X85G7US Patent
TargetBromodomain-containing protein 4 [44-168]/Histone H4(Homo sapiens (Human))
Boehringer Ingelheim International GmbH

US Patent
LigandPNGBDBM209481(US10328074, Example III-22 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 uM start concentration) in white OptiPlate-384 (PerkinElme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23X85G7US Patent
TargetBromodomain-containing protein 4 [44-168]/Histone H4(Homo sapiens (Human))
Boehringer Ingelheim International GmbH

US Patent
LigandPNGBDBM209482(US10328074, Example III-23 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 uM start concentration) in white OptiPlate-384 (PerkinElme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23X85G7US Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))TBA
LigandPNGBDBM242688(US9422290, I-1)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R49PPGUS Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))TBA
LigandPNGBDBM242696(US9422290, II-3)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R49PPGUS Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))TBA
LigandPNGBDBM242702(US9422290, II-9)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R49PPGUS Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))TBA
LigandPNGBDBM242713(US9422290, III-2)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R49PPGUS Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))TBA
LigandPNGBDBM242714(US9422290, III-3)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R49PPGUS Patent
TargetBromodomain-containing protein 4 [42-168](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM209474(US10328074, Example III-15 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:This assay is used to determine whether the compounds inhibit the interaction between the first (BRD4-BD1) or the second (BRD4-BD2) bromodomain of BR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z75M2US Patent
TargetBromodomain-containing protein 4 [42-168](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM209481(US10328074, Example III-22 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:This assay is used to determine whether the compounds inhibit the interaction between the first (BRD4-BD1) or the second (BRD4-BD2) bromodomain of BR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z75M2US Patent
TargetBromodomain-containing protein 4 [42-168](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM209482(US10328074, Example III-23 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:This assay is used to determine whether the compounds inhibit the interaction between the first (BRD4-BD1) or the second (BRD4-BD2) bromodomain of BR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z75M2US Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))TBA
LigandPNGBDBM209474(US10328074, Example III-15 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PV6PHQUS Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))TBA
LigandPNGBDBM209481(US10328074, Example III-22 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PV6PHQUS Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))TBA
LigandPNGBDBM209482(US10328074, Example III-23 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PV6PHQUS Patent
TargetBromodomain-containing protein 4 [44-168]/Histone H4(Homo sapiens (Human))
Boehringer Ingelheim International GmbH

US Patent
LigandPNGBDBM209474(US10328074, Example III-15 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 uM start concentration) in white OptiPlate-384 (PerkinElme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23X85G7US Patent
TargetBromodomain-containing protein 4 [44-168]/Histone H4(Homo sapiens (Human))
Boehringer Ingelheim International GmbH

US Patent
LigandPNGBDBM209457(US10328074, Example II-1 | US11077107, Example II-...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 uM start concentration) in white OptiPlate-384 (PerkinElme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23X85G7US Patent
TargetBromodomain-containing protein 4 [44-168]/Histone H4(Homo sapiens (Human))
Boehringer Ingelheim International GmbH

US Patent
LigandPNGBDBM209508(US10328074, Example III-49 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 uM start concentration) in white OptiPlate-384 (PerkinElme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23X85G7US Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))TBA
LigandPNGBDBM242701(US9422290, II-8)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R49PPGUS Patent
TargetBromodomain-containing protein 4 [42-168](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM209457(US10328074, Example II-1 | US11077107, Example II-...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:This assay is used to determine whether the compounds inhibit the interaction between the first (BRD4-BD1) or the second (BRD4-BD2) bromodomain of BR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z75M2US Patent
TargetBromodomain-containing protein 4 [42-168](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM209508(US10328074, Example III-49 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:This assay is used to determine whether the compounds inhibit the interaction between the first (BRD4-BD1) or the second (BRD4-BD2) bromodomain of BR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z75M2US Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))TBA
LigandPNGBDBM209457(US10328074, Example II-1 | US11077107, Example II-...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PV6PHQUS Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))TBA
LigandPNGBDBM209508(US10328074, Example III-49 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PV6PHQUS Patent
TargetBromodomain-containing protein 4 [44-168]/Histone H4(Homo sapiens (Human))
Boehringer Ingelheim International GmbH

US Patent
LigandPNGBDBM209475(US10328074, Example III-16 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 uM start concentration) in white OptiPlate-384 (PerkinElme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23X85G7US Patent
TargetBromodomain-containing protein 4 [44-168]/Histone H4(Homo sapiens (Human))
Boehringer Ingelheim International GmbH

US Patent
LigandPNGBDBM209485(US10328074, Example III-26 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 uM start concentration) in white OptiPlate-384 (PerkinElme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23X85G7US Patent
TargetBromodomain-containing protein 4 [42-168](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM209475(US10328074, Example III-16 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:This assay is used to determine whether the compounds inhibit the interaction between the first (BRD4-BD1) or the second (BRD4-BD2) bromodomain of BR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z75M2US Patent
TargetBromodomain-containing protein 4 [42-168](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM209485(US10328074, Example III-26 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:This assay is used to determine whether the compounds inhibit the interaction between the first (BRD4-BD1) or the second (BRD4-BD2) bromodomain of BR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z75M2US Patent
TargetBromodomain-containing protein 4 [42-168](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM209509(US10328074, Example III-50 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:This assay is used to determine whether the compounds inhibit the interaction between the first (BRD4-BD1) or the second (BRD4-BD2) bromodomain of BR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z75M2US Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))TBA
LigandPNGBDBM209475(US10328074, Example III-16 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PV6PHQUS Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))TBA
LigandPNGBDBM209485(US10328074, Example III-26 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PV6PHQUS Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))TBA
LigandPNGBDBM209509(US10328074, Example III-50 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PV6PHQUS Patent
TargetBromodomain-containing protein 4 [44-168]/Histone H4(Homo sapiens (Human))
Boehringer Ingelheim International GmbH

US Patent
LigandPNGBDBM209509(US10328074, Example III-50 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 uM start concentration) in white OptiPlate-384 (PerkinElme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23X85G7US Patent
TargetBromodomain-containing protein 4 [44-168]/Histone H4(Homo sapiens (Human))
Boehringer Ingelheim International GmbH

US Patent
LigandPNGBDBM209460(US10328074, Example III-1 | US11077107, Example II...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 uM start concentration) in white OptiPlate-384 (PerkinElme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23X85G7US Patent
TargetBromodomain-containing protein 4 [44-168]/Histone H4(Homo sapiens (Human))
Boehringer Ingelheim International GmbH

US Patent
LigandPNGBDBM209471(US10328074, Example III-12 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 uM start concentration) in white OptiPlate-384 (PerkinElme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23X85G7US Patent
TargetBromodomain-containing protein 4 [44-168]/Histone H4(Homo sapiens (Human))
Boehringer Ingelheim International GmbH

US Patent
LigandPNGBDBM209491(US10328074, Example III-32 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 uM start concentration) in white OptiPlate-384 (PerkinElme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23X85G7US Patent
TargetBromodomain-containing protein 4 [42-168](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM209460(US10328074, Example III-1 | US11077107, Example II...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:This assay is used to determine whether the compounds inhibit the interaction between the first (BRD4-BD1) or the second (BRD4-BD2) bromodomain of BR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z75M2US Patent
TargetBromodomain-containing protein 4 [42-168](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM209471(US10328074, Example III-12 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:This assay is used to determine whether the compounds inhibit the interaction between the first (BRD4-BD1) or the second (BRD4-BD2) bromodomain of BR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z75M2US Patent
TargetBromodomain-containing protein 4 [42-168](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM209491(US10328074, Example III-32 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:This assay is used to determine whether the compounds inhibit the interaction between the first (BRD4-BD1) or the second (BRD4-BD2) bromodomain of BR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z75M2US Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))TBA
LigandPNGBDBM209460(US10328074, Example III-1 | US11077107, Example II...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PV6PHQUS Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))TBA
LigandPNGBDBM209471(US10328074, Example III-12 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PV6PHQUS Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))TBA
LigandPNGBDBM209491(US10328074, Example III-32 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PV6PHQUS Patent
TargetBromodomain-containing protein 4 [44-168]/Histone H4(Homo sapiens (Human))
Boehringer Ingelheim International GmbH

US Patent
LigandPNGBDBM209453(US10328074, Example I-5 | US11077107, Example I-5 ...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 uM start concentration) in white OptiPlate-384 (PerkinElme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23X85G7US Patent
TargetBromodomain-containing protein 4 [44-168]/Histone H4(Homo sapiens (Human))
Boehringer Ingelheim International GmbH

US Patent
LigandPNGBDBM209463(US10328074, Example III-4 | US11077107, Example II...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 uM start concentration) in white OptiPlate-384 (PerkinElme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23X85G7US Patent
TargetBromodomain-containing protein 4 [44-168]/Histone H4(Homo sapiens (Human))
Boehringer Ingelheim International GmbH

US Patent
LigandPNGBDBM209507(US10328074, Example III-48 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 uM start concentration) in white OptiPlate-384 (PerkinElme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23X85G7US Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))TBA
LigandPNGBDBM242699(US9422290, II-6)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R49PPGUS Patent
TargetBromodomain-containing protein 4 [44-168](Homo sapiens (Human))TBA
LigandPNGBDBM242700(US9422290, II-7)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (Perki...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2R49PPGUS Patent
TargetBromodomain-containing protein 4 [42-168](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM209453(US10328074, Example I-5 | US11077107, Example I-5 ...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:This assay is used to determine whether the compounds inhibit the interaction between the first (BRD4-BD1) or the second (BRD4-BD2) bromodomain of BR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z75M2US Patent
TargetBromodomain-containing protein 4 [42-168](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM209463(US10328074, Example III-4 | US11077107, Example II...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:This assay is used to determine whether the compounds inhibit the interaction between the first (BRD4-BD1) or the second (BRD4-BD2) bromodomain of BR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z75M2US Patent
TargetBromodomain-containing protein 4 [42-168](Homo sapiens (Human))
Duquesne University

LigandPNGBDBM209480(US10328074, Example III-21 | US11077107, Example I...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:This assay is used to determine whether the compounds inhibit the interaction between the first (BRD4-BD1) or the second (BRD4-BD2) bromodomain of BR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z75M2US Patent
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