Compile Data Set for Download or QSAR
Found 345 with Last Name = 'madge' and Initial = 'd'
TargetTryptophan 2,3-dioxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50289136(6-Fluoro-3-((E)-2-pyridin-4-yl-vinyl)-1H-indole | ...)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Compound was tested for inhibition of Tryptophan dioxygenase (TDO) from rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833S17
TargetTryptophan 2,3-dioxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50289137(6-Fluoro-3-((E)-2-pyridin-3-yl-vinyl)-1H-indole | ...)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Compound was tested for inhibition of Tryptophan dioxygenase (TDO) from rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833S17
TargetTryptophan 2,3-dioxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50289142(3-((E)-2-Pyridin-4-yl-vinyl)-1H-indole | CHEMBL166...)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Compound was tested for inhibition of Tryptophan dioxygenase (TDO) from rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833S17
TargetTryptophan 2,3-dioxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50289138(3-((E)-2-Pyridin-3-yl-vinyl)-1H-indole | CHEMBL441...)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Compound was tested for inhibition of Tryptophan dioxygenase (TDO) from rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833S17
TargetTryptophan 2,3-dioxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50289141(5-Fluoro-3-((E)-2-pyridin-4-yl-vinyl)-1H-indole | ...)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Compound was tested for inhibition of Tryptophan dioxygenase (TDO) from rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833S17
TargetTryptophan 2,3-dioxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50289140(5-Fluoro-3-((E)-2-pyridin-3-yl-vinyl)-1H-indole | ...)copy SMILEScopy InChI
Affinity DataKi:  50nMAssay Description:Compound was tested for inhibition of Tryptophan dioxygenase (TDO) from rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833S17
TargetTryptophan 2,3-dioxygenase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50289139(3-((E)-2-Pyridin-2-yl-vinyl)-1H-indole | CHEMBL171...)copy SMILEScopy InChI
Affinity DataKi:  100nMAssay Description:Compound was tested for inhibition of Tryptophan dioxygenase (TDO) from rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833S17
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344356(CHEMBL1779676 | ethyl 3-(3-(7-hydroxynaphthalen-1-...)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin-i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344356(CHEMBL1779676 | ethyl 3-(3-(7-hydroxynaphthalen-1-...)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344367(1-(4-chloro-3-(trifluoromethyl)phenyl)-3-(7-hydrox...)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin-i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344378(1-(4-chloro-3-(trifluoromethyl)phenyl)-3-(2,3-dich...)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin-i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344367(1-(4-chloro-3-(trifluoromethyl)phenyl)-3-(7-hydrox...)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344367(1-(4-chloro-3-(trifluoromethyl)phenyl)-3-(7-hydrox...)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Antagonist activity at human TRPV1 expressed in CHOluc9aeq cells assessed as inhibition of capsaicin-stimulated response by aequorin and CRE-lucifear...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C24XF7PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344348(1-(3-chlorophenyl)-3-(7-hydroxynaphthalen-1-yl)ure...)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin-i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50382237(CHEMBL2024668)copy SMILEScopy InChI
Affinity DataIC50: 3.30nMAssay Description:Antagonist activity at human TRPV1 expressed in CHOluc9aeq cells assessed as inhibition of capsaicin-stimulated response by aequorin and CRE-lucifear...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C24XF7PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50382237(CHEMBL2024668)copy SMILEScopy InChI
Affinity DataIC50: 3.30nMAssay Description:Antagonist activity at human TRPV1 expressed in CHOluc9aeq cells assessed as inhibition of capsaicin-stimulated response by aequorin and CRE-lucifear...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C24XF7PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344377(1-(4-chloro-3-(trifluoromethyl)phenyl)-3-(2-chloro...)copy SMILEScopy InChI
Affinity DataIC50: 3.40nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344345(1-(7-hydroxynaphthalen-1-yl)-3-(3-(trifluoromethyl...)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM20412(3-(7-hydroxynaphthalen-1-yl)-1-[3-(methylsulfanyl)...)copy SMILEScopy InChI
Affinity DataIC50: 3.90nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344377(1-(4-chloro-3-(trifluoromethyl)phenyl)-3-(2-chloro...)copy SMILEScopy InChI
Affinity DataIC50: 4.5nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin-i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344363(1-(3,4-dichlorophenyl)-3-(7-hydroxynaphthalen-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 4.5nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin-i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344345(1-(7-hydroxynaphthalen-1-yl)-3-(3-(trifluoromethyl...)copy SMILEScopy InChI
Affinity DataIC50: 4.5nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin-i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344346(1-(7-hydroxynaphthalen-1-yl)-3-(4-(trifluoromethyl...)copy SMILEScopy InChI
Affinity DataIC50: 4.90nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin-i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344363(1-(3,4-dichlorophenyl)-3-(7-hydroxynaphthalen-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 4.90nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344372(1-(3-bromo-2-chloro-7-hydroxynaphthalen-1-yl)-3-(4...)copy SMILEScopy InChI
Affinity DataIC50: 4.90nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin-i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344346(1-(7-hydroxynaphthalen-1-yl)-3-(4-(trifluoromethyl...)copy SMILEScopy InChI
Affinity DataIC50: 5.40nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344355(1-(3-bromophenyl)-3-(7-hydroxynaphthalen-1-yl)urea...)copy SMILEScopy InChI
Affinity DataIC50: 5.70nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344378(1-(4-chloro-3-(trifluoromethyl)phenyl)-3-(2,3-dich...)copy SMILEScopy InChI
Affinity DataIC50: 5.90nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344348(1-(3-chlorophenyl)-3-(7-hydroxynaphthalen-1-yl)ure...)copy SMILEScopy InChI
Affinity DataIC50: 6.10nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344372(1-(3-bromo-2-chloro-7-hydroxynaphthalen-1-yl)-3-(4...)copy SMILEScopy InChI
Affinity DataIC50: 6.80nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM20412(3-(7-hydroxynaphthalen-1-yl)-1-[3-(methylsulfanyl)...)copy SMILEScopy InChI
Affinity DataIC50: 7.10nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin-i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344353(1-(7-hydroxynaphthalen-1-yl)-3-(3-nitrophenyl)urea...)copy SMILEScopy InChI
Affinity DataIC50: 7.5nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344373(1-(4-chloro-3-(trifluoromethyl)phenyl)-3-(2,3-dibr...)copy SMILEScopy InChI
Affinity DataIC50: 7.5nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344352(1-(7-hydroxynaphthalen-1-yl)-3-(3-methoxyphenyl)ur...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344355(1-(3-bromophenyl)-3-(7-hydroxynaphthalen-1-yl)urea...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin-i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344352(1-(7-hydroxynaphthalen-1-yl)-3-(3-methoxyphenyl)ur...)copy SMILEScopy InChI
Affinity DataIC50: 8.60nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin-i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50382245(CHEMBL2024494)copy SMILEScopy InChI
Affinity DataIC50: 9.10nMAssay Description:Antagonist activity at human TRPV1 expressed in CHOluc9aeq cells assessed as inhibition of capsaicin-stimulated response by aequorin and CRE-lucifear...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C24XF7PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344349(1-(4-chlorophenyl)-3-(7-hydroxynaphthalen-1-yl)ure...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin-i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344350(1-(7-hydroxynaphthalen-1-yl)-3-m-tolylurea | CHEMB...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344349(1-(4-chlorophenyl)-3-(7-hydroxynaphthalen-1-yl)ure...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344362(1-(2,4-dichlorophenyl)-3-(7-hydroxynaphthalen-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344364(1-(3,5-dichlorophenyl)-3-(7-hydroxynaphthalen-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344366(1-(2-chloro-5-(trifluoromethyl)phenyl)-3-(7-hydrox...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin-i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344364(1-(3,5-dichlorophenyl)-3-(7-hydroxynaphthalen-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin-i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344366(1-(2-chloro-5-(trifluoromethyl)phenyl)-3-(7-hydrox...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344351(1-(3-fluorophenyl)-3-(7-hydroxynaphthalen-1-yl)ure...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Antagonist activity at human TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344353(1-(7-hydroxynaphthalen-1-yl)-3-(3-nitrophenyl)urea...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin-i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344373(1-(4-chloro-3-(trifluoromethyl)phenyl)-3-(2,3-dibr...)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin-i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50382240(CHEMBL2024667)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human TRPV1 expressed in CHOluc9aeq cells assessed as inhibition of capsaicin-stimulated response by aequorin and CRE-lucifear...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C24XF7PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Bayer Yakuhin, Ltd

Curated by ChEMBL
LigandPNGBDBM50344362(1-(2,4-dichlorophenyl)-3-(7-hydroxynaphthalen-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Antagonist activity at rat TRPV1 expressed in CHO cells co-expressing aequorin and CRE-luciferase reporter gene assessed as inhibition of capsaicin-i...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NG4QXNPubMed
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