Compile Data Set for Download or QSAR
Found 883 with Last Name = 'mumberg' and Initial = 'd'
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM228279(US9555022, Example 02.17)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM228278(US9555022, Example 02.16)copy SMILEScopy InChI
Affinity DataIC50: 0.150nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50542581(CHEMBL4642174)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM228270(US9555022, Example 02.09)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM258444(US9512130, 2)copy SMILEScopy InChI
Affinity DataIC50: 0.25nMAssay Description:Inhibition of MPS1 in human HeLa cells assessed as reduction in spindle assembly checkpoint incubated for 4 hrs by p-histone H3/Hoechst 33342 stainin...More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50520160(CHEMBL4515413 | US10894784, Example 01.03)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged FLT3 (564 to end residues) expressed in sf21 cells using biotin labelled Ahx-GGEEEEYFELVKKKK pe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CN7795PubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50542592(CHEMBL4645348)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM259464(US9512126, 1)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Inhibition of MPS1 in human HeLa cells assessed as reduction in spindle assembly checkpoint incubated for 4 hrs by p-histone H3/Hoechst 33342 stainin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50542591(CHEMBL4640247)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Inhibition of MPS1 in human HeLa cells assessed as reduction in spindle assembly checkpoint incubated for 4 hrs by p-histone H3/Hoechst 33342 stainin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50542591(CHEMBL4640247)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM259464(US9512126, 1)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50542592(CHEMBL4645348)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50542581(CHEMBL4642174)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM329340((2R)—N-{4-[2-({4-[(3-fluoroazetidin-1-yl)carb...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50542583(CHEMBL4634949)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM259482(US9512126, 23)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50512456(CHEMBL4469414)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50520150(CHEMBL4566796)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:Inhibition of recombinant full length human N-terminal His-tagged TBK1 using biotin-labelled Ahx-GDEDFSSFAEPG peptide as substrate preincubated with ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CN7795PubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM258444(US9512130, 2)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM259482(US9512126, 23)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50520175(CHEMBL4451595 | US10894784, Example 135.02)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged FLT3 (564 to end residues) expressed in sf21 cells using biotin labelled Ahx-GGEEEEYFELVKKKK pe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CN7795PubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50542558(CHEMBL4646772)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50542559(CHEMBL4635693)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM228261(US9555022, Example 02.01)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50512459(CHEMBL4581793)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM101243(US8524722, 143)copy SMILEScopy InChI
Affinity DataIC50: 1nMpH: 7.0 T: 2°CAssay Description:EGFR inhibitory activity of compounds of the present invention is quantified employing the EGFR HTRF assay.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2B856RQUS Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM101241(US8524722, 134)copy SMILEScopy InChI
Affinity DataIC50: 1nMpH: 7.0 T: 2°CAssay Description:EGFR inhibitory activity of compounds of the present invention is quantified employing the EGFR HTRF assay.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2B856RQUS Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM101240(US8524722, 123)copy SMILEScopy InChI
Affinity DataIC50: 1nMpH: 7.0 T: 2°CAssay Description:EGFR inhibitory activity of compounds of the present invention is quantified employing the EGFR HTRF assay.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2B856RQUS Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM101239(US8524722, 119)copy SMILEScopy InChI
Affinity DataIC50: 1nMpH: 7.0 T: 2°CAssay Description:EGFR inhibitory activity of compounds of the present invention is quantified employing the EGFR HTRF assay.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2B856RQUS Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM101237(US8524722, 90)copy SMILEScopy InChI
Affinity DataIC50: 1nMpH: 7.0 T: 2°CAssay Description:EGFR inhibitory activity of compounds of the present invention is quantified employing the EGFR HTRF assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2B856RQUS Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM101232(US8524722, 70)copy SMILEScopy InChI
Affinity DataIC50: 1nMpH: 7.0 T: 2°CAssay Description:EGFR inhibitory activity of compounds of the present invention is quantified employing the EGFR HTRF assay.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2B856RQUS Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM101231(US8524722, 31)copy SMILEScopy InChI
Affinity DataIC50: 1nMpH: 7.0 T: 2°CAssay Description:EGFR inhibitory activity of compounds of the present invention is quantified employing the EGFR HTRF assay.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2B856RQUS Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM101230(US8524722, 14)copy SMILEScopy InChI
Affinity DataIC50: 1nMpH: 7.0 T: 2°CAssay Description:EGFR inhibitory activity of compounds of the present invention is quantified employing the EGFR HTRF assay.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2B856RQUS Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM228273(US9555022, Example 02.11)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM329342((2R)-2-(4-fluorophenyl)-N-[4-(2-{[2-methoxy-4-(2-o...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM258444(US9512130, 2)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50542591(CHEMBL4640247)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50520159(CHEMBL4543618)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged FLT3 (564 to end residues) expressed in sf21 cells using biotin labelled Ahx-GGEEEEYFELVKKKK pe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CN7795PubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50520142(CHEMBL4435393)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant full length human N-terminal His-tagged TBK1 using biotin-labelled Ahx-GDEDFSSFAEPG peptide as substrate preincubated with ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CN7795PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM101226(US8524722, 5)copy SMILEScopy InChI
Affinity DataIC50: 1nMpH: 7.0 T: 2°CAssay Description:EGFR inhibitory activity of compounds of the present invention is quantified employing the EGFR HTRF assay.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2B856RQUS Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM101228(US8524722, 12)copy SMILEScopy InChI
Affinity DataIC50: 1nMpH: 7.0 T: 2°CAssay Description:EGFR inhibitory activity of compounds of the present invention is quantified employing the EGFR HTRF assay.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2B856RQUS Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM101227(US8524722, 10)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMpH: 7.0 T: 2°CAssay Description:EGFR inhibitory activity of compounds of the present invention is quantified employing the EGFR HTRF assay.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2B856RQUS Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50542583(CHEMBL4634949)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM259464(US9512126, 1)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50512456(CHEMBL4469414)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50542561(CHEMBL4638962)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50542562(CHEMBL4632648)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Bayer Intellectual Property GmbH

US Patent
LigandPNGBDBM101234(US8524722, 84)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMpH: 7.0 T: 2°CAssay Description:EGFR inhibitory activity of compounds of the present invention is quantified employing the EGFR HTRF assay.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2B856RQUS Patent
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM228316(US9555022, Example 02.44)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:Inhibition of GST-tagged recombinant human MPS1 expressed in baculovirus expression system using biotin-Ahx-PWDPDDADITEILG as substrate preincubated ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP56VPPubMed
Displayed 1 to 50 (of 883 total ) | Next | Last >>
Jump to: