Compile Data Set for Download or QSAR
Found 81 with Last Name = 'pechalrieu' and Initial = 'd'
TargetHistone deacetylase 6(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50005711(CHEBI:46024 | GNF-Pf-1011 | TRICHOSTATIN | Trichos...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant human HDAC6 using RHK-K(Ac) as substrate by homogeneous fluorescence release assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50506775(CHEMBL4593437)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of recombinant human HDAC6 using RHK-K(Ac) as substrate by homogeneous fluorescence release assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50005711(CHEBI:46024 | GNF-Pf-1011 | TRICHOSTATIN | Trichos...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant human HDAC1 using RHK-K(Ac) as substrate by homogeneous fluorescence release assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50506777(CHEMBL4476057)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant human HDAC6 using RHK-K(Ac) as substrate by homogeneous fluorescence release assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50506780(CHEMBL4550522)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant human HDAC6 using RHK-K(Ac) as substrate by homogeneous fluorescence release assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50506778(CHEMBL4469596)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human HDAC6 using RHK-K(Ac) as substrate by homogeneous fluorescence release assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50506779(CHEMBL4521590)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Inhibition of recombinant human HDAC6 using RHK-K(Ac) as substrate by homogeneous fluorescence release assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50506781(CHEMBL4435005)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:Inhibition of recombinant human HDAC6 using RHK-K(Ac) as substrate by homogeneous fluorescence release assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50506775(CHEMBL4593437)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant human HDAC1 using RHK-K(Ac) as substrate by homogeneous fluorescence release assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50506780(CHEMBL4550522)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant human HDAC1 using RHK-K(Ac) as substrate by homogeneous fluorescence release assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50506781(CHEMBL4435005)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant human HDAC1 using RHK-K(Ac) as substrate by homogeneous fluorescence release assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50446481(CHEMBL3110004 | US10011611, TMP269 | US10722597, C...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys(trifluoroacetyl)-AMC as substrate by homogeneous fluorescence release assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50506779(CHEMBL4521590)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of recombinant human HDAC1 using RHK-K(Ac) as substrate by homogeneous fluorescence release assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50506778(CHEMBL4469596)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of recombinant human HDAC1 using RHK-K(Ac) as substrate by homogeneous fluorescence release assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50506777(CHEMBL4476057)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of recombinant human HDAC1 using RHK-K(Ac) as substrate by homogeneous fluorescence release assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50506780(CHEMBL4550522)copy SMILEScopy InChI
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys(trifluoroacetyl)-AMC as substrate by homogeneous fluorescence release assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50005711(CHEBI:46024 | GNF-Pf-1011 | TRICHOSTATIN | Trichos...)copy SMILEScopy InChI
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys(trifluoroacetyl)-AMC as substrate by homogeneous fluorescence release assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50506781(CHEMBL4435005)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys(trifluoroacetyl)-AMC as substrate by homogeneous fluorescence release assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50506775(CHEMBL4593437)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys(trifluoroacetyl)-AMC as substrate by homogeneous fluorescence release assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50506779(CHEMBL4521590)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys(trifluoroacetyl)-AMC as substrate by homogeneous fluorescence release assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50506778(CHEMBL4469596)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys(trifluoroacetyl)-AMC as substrate by homogeneous fluorescence release assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50506777(CHEMBL4476057)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human HDAC4 using Boc-Lys(trifluoroacetyl)-AMC as substrate by homogeneous fluorescence release assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239284(CHEMBL4096360)copy SMILEScopy InChI
Affinity DataEC50:  4.40E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239285(CHEMBL4096869)copy SMILEScopy InChI
Affinity DataEC50:  2.10E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239286(CHEMBL4084601)copy SMILEScopy InChI
Affinity DataEC50:  4.90E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239287(CHEMBL4100095)copy SMILEScopy InChI
Affinity DataEC50:  6.80E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239288(CHEMBL4097685)copy SMILEScopy InChI
Affinity DataEC50:  1.20E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239289(CHEMBL4096752)copy SMILEScopy InChI
Affinity DataEC50:  3.40E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239290(CHEMBL4099197)copy SMILEScopy InChI
Affinity DataEC50:  1.10E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239291(CHEMBL4091463)copy SMILEScopy InChI
Affinity DataEC50:  300nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239284(CHEMBL4096360)copy SMILEScopy InChI
Affinity DataEC50:  4.60E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239285(CHEMBL4096869)copy SMILEScopy InChI
Affinity DataEC50:  2.40E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239286(CHEMBL4084601)copy SMILEScopy InChI
Affinity DataEC50:  3.20E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239287(CHEMBL4100095)copy SMILEScopy InChI
Affinity DataEC50:  7.30E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239288(CHEMBL4097685)copy SMILEScopy InChI
Affinity DataEC50:  2.60E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239290(CHEMBL4099197)copy SMILEScopy InChI
Affinity DataEC50:  1.00E+5nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239292(CHEMBL4070549)copy SMILEScopy InChI
Affinity DataEC50:  1.60E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239291(CHEMBL4091463)copy SMILEScopy InChI
Affinity DataEC50:  2.00E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239293(CHEMBL4076088)copy SMILEScopy InChI
Affinity DataEC50:  1.40E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239294(CHEMBL4070517)copy SMILEScopy InChI
Affinity DataEC50:  1.00E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239292(CHEMBL4070549)copy SMILEScopy InChI
Affinity DataEC50:  1.90E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239293(CHEMBL4076088)copy SMILEScopy InChI
Affinity DataEC50:  3.00E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50239289(CHEMBL4096752)copy SMILEScopy InChI
Affinity DataEC50:  2.70E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6G1KPubMed
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50506774(CHEMBL4470149)copy SMILEScopy InChI
Affinity DataEC50:  4.80E+3nMAssay Description:Inhibition of recombinant human DNMT3a C-terminal catalytic domain (623 to 908 residues) using 5'-biotinylated/3'-FAM-oligonucleotide as substrate me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universit£ de Lille

Curated by ChEMBL
LigandPNGBDBM50506774(CHEMBL4470149)copy SMILEScopy InChI
Affinity DataEC50:  5.09E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-fused G9a (786 to 1210 residues) expressed in Escherichia coli using biotinylated H3 (1 to 21 residues...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50506776(CHEMBL4442279)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of recombinant human DNMT1 using biotinylated DNA duplex as substrate measured after 2 hrs in presence of Adomet/[methyl-3H]Adomet by topc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50506774(CHEMBL4470149)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of recombinant human DNMT1 using biotinylated DNA duplex as substrate measured after 2 hrs in presence of Adomet/[methyl-3H]Adomet by topc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50506782(CHEMBL4461581)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of recombinant human DNMT1 using biotinylated DNA duplex as substrate measured after 2 hrs in presence of Adomet/[methyl-3H]Adomet by topc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50506783(CHEMBL4582042)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of recombinant human DNMT1 using biotinylated DNA duplex as substrate measured after 2 hrs in presence of Adomet/[methyl-3H]Adomet by topc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388

Curated by ChEMBL
LigandPNGBDBM50506784(CHEMBL4527662)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of recombinant human DNMT1 using biotinylated DNA duplex as substrate measured after 2 hrs in presence of Adomet/[methyl-3H]Adomet by topc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5J76PubMed
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