Compile Data Set for Download or QSAR
Found 51 with Last Name = 'colby' and Initial = 'da'
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM24182(4-amino-3-(4-chlorophenyl)butanoic acid | Baclofen...)copy SMILEScopy InChI
Affinity DataKi:  6.00E+3nMAssay Description:Displacement of [3H]CGP54626 from GABA-B receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50007119(4-Amino-3-phenyl-butyric acid | CHEMBL53073)copy SMILEScopy InChI
Affinity DataKi:  9.20E+4nMAssay Description:Displacement of [3H]CGP54626 from GABA-B receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T155F6PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50007119(4-Amino-3-phenyl-butyric acid | CHEMBL53073)copy SMILEScopy InChI
Affinity DataKi:  1.77E+5nMAssay Description:Displacement of [3H]CGP54626 from GABA-B receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T155F6PubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
University of California at Irvine

Curated by ChEMBL
LigandPNGBDBM50127377(10-[3,9-dimethyl-8-(3-methyl-4-oxopentyl)-(9R)-1,7...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of protein phosphatase 2A (PP2A) was determined by standard phosphorylase a inhibition assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DB82CKPubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50007118(4-Amino-3-(5-chloro-thiophen-2-yl)-butyric acid | ...)copy SMILEScopy InChI
Affinity DataIC50: 610nMAssay Description:Binding affinity to GABA-B receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T155F6PubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
University of California at Irvine

Curated by ChEMBL
LigandPNGBDBM50127375((E)-(R)-4-Hydroxy-2-methyl-hex-2-enedioic acid 6-{...)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of protein phosphatase 2A (PP2A) was determined by standard phosphorylase a inhibition assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DB82CKPubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
University of California at Irvine

Curated by ChEMBL
LigandPNGBDBM50366883(TAUTOMYCIN)copy SMILEScopy InChI
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibition of protein phosphatase 2A (PP2A) was determined by standard phosphorylase a inhibition assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DB82CKPubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
University of California at Irvine

Curated by ChEMBL
LigandPNGBDBM50127378((S)-2-Hydroxy-2-methyl-succinic acid 4-{(1R,2S,3R,...)copy SMILEScopy InChI
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of protein phosphatase 2A (PP2A) was determined by standard phosphorylase a inhibition assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DB82CKPubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
University of California at Irvine

Curated by ChEMBL
LigandPNGBDBM50127376((R)-2-Hydroxy-2-methyl-succinic acid 4-{(1R,2S,3R,...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of protein phosphatase 2A (PP2A) was determined by standard phosphorylase a inhibition assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DB82CKPubMed
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
University of California at Irvine

Curated by ChEMBL
LigandPNGBDBM50127379(4-Phosphono-butyric acid (1R,2S,3R,6S,7S,10R)-10-[...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of protein phosphatase 2A (PP2A) was determined by standard phosphorylase a inhibition assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DB82CKPubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50427606(CHEMBL2322945)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GABA-B B1/B2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 3 hr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3MTSPubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50427607(CHEMBL2322944)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GABA-B B1/B2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 3 hr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3MTSPubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50427608(CHEMBL2322943)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GABA-B B1/B2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 3 hr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3MTSPubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50427609(CHEMBL2322941)copy SMILEScopy InChI
Affinity DataEC50:  9.93E+4nMAssay Description:Agonist activity at human GABA-B B1/B2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 3 hr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3MTSPubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50427610(CHEMBL2322940)copy SMILEScopy InChI
Affinity DataEC50:  6.69E+4nMAssay Description:Agonist activity at human GABA-B B1/B2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 3 hr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3MTSPubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50427611(CHEMBL2322939)copy SMILEScopy InChI
Affinity DataEC50:  6.18E+4nMAssay Description:Agonist activity at human GABA-B B1/B2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 3 hr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3MTSPubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50427612(CHEMBL2322942)copy SMILEScopy InChI
Affinity DataEC50:  5.35E+4nMAssay Description:Agonist activity at human GABA-B B1/B2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 3 hr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3MTSPubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50427613(CHEMBL2322935)copy SMILEScopy InChI
Affinity DataEC50:  4.00E+4nMAssay Description:Agonist activity at human GABA-B B1/B2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 3 hr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3MTSPubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50427603(CHEMBL2322934)copy SMILEScopy InChI
Affinity DataEC50:  1.59E+4nMAssay Description:Agonist activity at human GABA-B B1/B2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 3 hr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3MTSPubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50427614(CHEMBL2322946)copy SMILEScopy InChI
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at human GABA-B B1/B2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 3 hr...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM24182(4-amino-3-(4-chlorophenyl)butanoic acid | Baclofen...)copy SMILEScopy InChI
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at human GABA-B B1/B2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 3 hr...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50462450(CHEMBL4238712)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at rat GFP-fused GABA-A alpha1/beta2/gamma2 receptor expressed in human tsA201 cells at -60 mV holding potential by whole-cell volta...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P12N7PubMed
TargetGamma-aminobutyric acid receptor subunit beta-1/beta-2(Homo sapiens (Human))
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50462442(CHEMBL4245403)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P12N7PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50427613(CHEMBL2322935)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at rat GFP-fused GABA-A alpha1/beta2/gamma2 receptor expressed in human tsA201 cells at -60 mV holding potential by whole-cell volta...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P12N7PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50462443(CHEMBL4238315)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at rat GFP-fused GABA-A alpha1/beta2/gamma2 receptor expressed in human tsA201 cells at -60 mV holding potential by whole-cell volta...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P12N7PubMed
TargetGamma-aminobutyric acid receptor subunit beta-1/beta-2(Homo sapiens (Human))
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50462444(CHEMBL4244129)copy SMILEScopy InChI
Affinity DataEC50:  9.10E+4nMAssay Description:Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P12N7PubMed
TargetGamma-aminobutyric acid receptor subunit beta-1/beta-2(Homo sapiens (Human))
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50427613(CHEMBL2322935)copy SMILEScopy InChI
Affinity DataEC50:  4.00E+4nMAssay Description:Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P12N7PubMed
TargetGamma-aminobutyric acid receptor subunit beta-1/beta-2(Homo sapiens (Human))
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50462445(CHEMBL4246158)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P12N7PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50462444(CHEMBL4244129)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at rat GFP-fused GABA-A alpha1/beta2/gamma2 receptor expressed in human tsA201 cells at -60 mV holding potential by whole-cell volta...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P12N7PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50462446(CHEMBL4238634)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at rat GFP-fused GABA-A alpha1/beta2/gamma2 receptor expressed in human tsA201 cells at -60 mV holding potential by whole-cell volta...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P12N7PubMed
TargetGamma-aminobutyric acid receptor subunit beta-1/beta-2(Homo sapiens (Human))
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50462447(CHEMBL4248377)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P12N7PubMed
TargetGamma-aminobutyric acid receptor subunit beta-1/beta-2(Homo sapiens (Human))
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50462448(CHEMBL4241188)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P12N7PubMed
TargetGamma-aminobutyric acid receptor subunit beta-1/beta-2(Homo sapiens (Human))
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50462449(CHEMBL4247210)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P12N7PubMed
TargetGamma-aminobutyric acid receptor subunit beta-1/beta-2(Homo sapiens (Human))
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50462450(CHEMBL4238712)copy SMILEScopy InChI
Affinity DataEC50:  3.27E+4nMAssay Description:Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P12N7PubMed
TargetGamma-aminobutyric acid receptor subunit beta-1/beta-2(Homo sapiens (Human))
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50462451(CHEMBL4249205)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P12N7PubMed
TargetGamma-aminobutyric acid receptor subunit beta-1/beta-2(Homo sapiens (Human))
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50462452(CHEMBL4244940)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P12N7PubMed
TargetGamma-aminobutyric acid receptor subunit beta-1/beta-2(Homo sapiens (Human))
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50462453(CHEMBL4244933)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P12N7PubMed
TargetGamma-aminobutyric acid receptor subunit beta-1/beta-2(Homo sapiens (Human))
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50462446(CHEMBL4238634)copy SMILEScopy InChI
Affinity DataEC50:  1.94E+4nMAssay Description:Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P12N7PubMed
TargetGamma-aminobutyric acid receptor subunit beta-1/beta-2(Homo sapiens (Human))
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50462454(CHEMBL4250786)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P12N7PubMed
TargetGamma-aminobutyric acid receptor subunit beta-1/beta-2(Homo sapiens (Human))
University of Mississippi

Curated by ChEMBL
LigandPNGBDBM50462443(CHEMBL4238315)copy SMILEScopy InChI
Affinity DataEC50:  5.74E+4nMAssay Description:Agonist activity at human GABA-B1/B2 receptor expressed in HEK293/Cre-luc cells assessed as inhibition of forskolin-stimulated cAMP accumulation afte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20P12N7PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50427605(CHEMBL2322932)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GABA-B B1/B2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 3 hr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3MTSPubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50427604(CHEMBL2322936)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GABA-B B1/B2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 3 hr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3MTSPubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50032964((R)-4-Amino-3-(4-chloro-phenyl)-butyric acid | 4-A...)copy SMILEScopy InChI
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human GABA-B B1/B2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 3 hr...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50427603(CHEMBL2322934)copy SMILEScopy InChI
Affinity DataEC50:  3.78E+4nMAssay Description:Agonist activity at human GABA-B B1/B2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 3 hr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3MTSPubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50427603(CHEMBL2322934)copy SMILEScopy InChI
Affinity DataEC50:  3.78E+4nMAssay Description:Agonist activity at human GABA-B B1/B2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 3 hr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3MTSPubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50427602(CHEMBL2322937)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GABA-B B1/B2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 3 hr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3MTSPubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50427601(CHEMBL2322938)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GABA-B B1/B2 receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 3 hr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3MTSPubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50108998(CHEMBL3600560)copy SMILEScopy InChI
Affinity DataEC50:  8.60nMAssay Description:Agonist activity at human recombinant GABA-B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T155F6PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50108997(CGP-71872 | CHEMBL1628548)copy SMILEScopy InChI
Affinity DataKd:  1nMAssay Description:Binding affinity to GABA-B receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T155F6PubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50108996(CGP-7930 | CHEMBL1256697)copy SMILEScopy InChI
Affinity DataEC50:  5.37E+3nMAssay Description:Positive allosteric modulator activity at GABA-B receptor (unknown origin) assessed as potentiation of 1 uM GABA-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T155F6PubMed
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