Compile Data Set for Download or QSAR
Found 197 with Last Name = 'khadka' and Initial = 'db'
TargetAndrogen receptor(Mus musculus)
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM18161((1S,2S,7S,10R,11S,14S,15S)-14-hydroxy-2,15-dimethy...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Displacement of [3H] ]5alpha-DHT from mouse androgen receptor expressed in monkey COS7 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50500613(CHEMBL3752642)copy SMILEScopy InChI
Affinity DataIC50: 5.5nMAssay Description:Inhibition of Cyclophilin A peptidyl-prolyl cis-trans isomerase activity (unknown origin) using Succ-Ala-Leu-Pro-Phe-p-nitroaniline as substrate by I...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5Z1VPubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50022815((3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33...)copy SMILEScopy InChI
Affinity DataIC50: 7.20nMAssay Description:Inhibition of Cyclophilin A peptidyl-prolyl cis-trans isomerase activity (unknown origin) using Succ-Ala-Leu-Pro-Phe-p-nitroaniline as substrate by I...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5Z1VPubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50500614(CHEMBL3754544)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of Cyclophilin A peptidyl-prolyl cis-trans isomerase activity (unknown origin) using Succ-Ala-Leu-Pro-Phe-p-nitroaniline as substrate by I...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RF5Z1VPubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM22165(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-(3-pheny...)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of re-uptake of [3H]-DA at human DAT expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9ZPVPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50117973(CHEMBL3612829)copy SMILEScopy InChI
Affinity DataIC50: 56nMAssay Description:Inhibition of re-uptake of [3H]-5-HT at human SERT expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9ZPVPubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50469312(CHEMBL4277585)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibition of [3H]dopamine uptake at DAT (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89G42PubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50117974(CHEMBL3612833)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of [3H]serotonin uptake at SERT (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89G42PubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM22165(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-(3-pheny...)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibition of re-uptake of [3H]-NE at human NET expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9ZPVPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50235734(CHEMBL4083724)copy SMILEScopy InChI
Affinity DataIC50: 159nMAssay Description:Inhibition of re-uptake of [3H]-5-HT at human SERT expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9ZPVPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM82071(CAS_93413-69-5 | CAS_99300-78-4 | NSC_62923 | VENL...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of [3H]serotonin uptake at human SERT expressed in HEK293 cells after 15 to 20 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89G42PubMedDrugBank
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM82071(CAS_93413-69-5 | CAS_99300-78-4 | NSC_62923 | VENL...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of human SERT expressed in HEK293 cells assessed as reduction in [3H]5-HT uptake by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474DHGPubMedDrugBank
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM82071(CAS_93413-69-5 | CAS_99300-78-4 | NSC_62923 | VENL...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of re-uptake of [3H]-5-HT at human SERT expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9ZPVPubMedDrugBank
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50462927(CHEMBL4250965)copy SMILEScopy InChI
Affinity DataIC50: 230nMAssay Description:Inhibition of human SERT expressed in HEK293 cells assessed as reduction in [3H]5-HT uptake by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474DHGPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50462933(CHEMBL4240379)copy SMILEScopy InChI
Affinity DataIC50: 230nMAssay Description:Inhibition of human SERT expressed in HEK293 cells assessed as reduction in [3H]5-HT uptake by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474DHGPubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50462918(CHEMBL4245867)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Inhibition of [3H]norepinephrine uptake at human NET expressed in HEK293 cells after 15 to 20 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89G42PubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50462918(CHEMBL4245867)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Inhibition of human NET expressed in HEK293 cells assessed as reduction in [3H]-NE uptake by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474DHGPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50462919(CHEMBL4244291)copy SMILEScopy InChI
Affinity DataIC50: 273nMAssay Description:Inhibition of human SERT expressed in HEK293 cells assessed as reduction in [3H]5-HT uptake by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474DHGPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50462916(CHEMBL4243340)copy SMILEScopy InChI
Affinity DataIC50: 280nMAssay Description:Inhibition of human SERT expressed in HEK293 cells assessed as reduction in [3H]5-HT uptake by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474DHGPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50261046(CHEMBL4071385)copy SMILEScopy InChI
Affinity DataIC50: 310nMAssay Description:Inhibition of re-uptake of [3H]-5-HT at human SERT expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9ZPVPubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50117974(CHEMBL3612833)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:Inhibition of [3H]norepinephrine uptake at NET (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89G42PubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50462911(CHEMBL4237635)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibition of human SERT expressed in HEK293 cells assessed as reduction in [3H]5-HT uptake by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474DHGPubMed
TargetAndrogen receptor(Mus musculus)
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50430945(CHEMBL2336987)copy SMILEScopy InChI
Affinity DataIC50: 460nMAssay Description:Agonist activity at mouse androgen receptor assessed as inhibition of transactivation after 24 hrs by cell-based luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0HHMPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50462934(CHEMBL4239115)copy SMILEScopy InChI
Affinity DataIC50: 460nMAssay Description:Inhibition of human SERT expressed in HEK293 cells assessed as reduction in [3H]5-HT uptake by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474DHGPubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50469310(CHEMBL4288240)copy SMILEScopy InChI
Affinity DataIC50: 510nMAssay Description:Inhibition of [3H]norepinephrine uptake at human NET expressed in HEK293 cells after 15 to 20 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89G42PubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50469312(CHEMBL4277585)copy SMILEScopy InChI
Affinity DataIC50: 510nMAssay Description:Inhibition of [3H]norepinephrine uptake at NET (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89G42PubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50261040(CHEMBL4099475)copy SMILEScopy InChI
Affinity DataIC50: 540nMAssay Description:Inhibition of re-uptake of [3H]-5-HT at human SERT expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9ZPVPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50462926(CHEMBL4243862)copy SMILEScopy InChI
Affinity DataIC50: 550nMAssay Description:Inhibition of human SERT expressed in HEK293 cells assessed as reduction in [3H]5-HT uptake by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474DHGPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50235723(CHEMBL4082902)copy SMILEScopy InChI
Affinity DataIC50: 570nMAssay Description:Inhibition of [3H]serotonin uptake at human SERT expressed in HEK293 cells after 15 to 20 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89G42PubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50235723(CHEMBL4082902)copy SMILEScopy InChI
Affinity DataIC50: 579nMAssay Description:Inhibition of re-uptake of [3H]-5-HT at human SERT expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9ZPVPubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50235723(CHEMBL4082902)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition of [3H]norepinephrine uptake at human NET expressed in HEK293 cells after 15 to 20 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89G42PubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50469318(CHEMBL4278945)copy SMILEScopy InChI
Affinity DataIC50: 680nMAssay Description:Inhibition of [3H]serotonin uptake at human SERT expressed in HEK293 cells after 15 to 20 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89G42PubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50462918(CHEMBL4245867)copy SMILEScopy InChI
Affinity DataIC50: 740nMAssay Description:Inhibition of [3H]serotonin uptake at human SERT expressed in HEK293 cells after 15 to 20 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89G42PubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50462918(CHEMBL4245867)copy SMILEScopy InChI
Affinity DataIC50: 740nMAssay Description:Inhibition of human SERT expressed in HEK293 cells assessed as reduction in [3H]5-HT uptake by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474DHGPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50462930(CHEMBL4240083)copy SMILEScopy InChI
Affinity DataIC50: 741nMAssay Description:Inhibition of human SERT expressed in HEK293 cells assessed as reduction in [3H]5-HT uptake by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474DHGPubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50469310(CHEMBL4288240)copy SMILEScopy InChI
Affinity DataIC50: 820nMAssay Description:Inhibition of [3H]dopamine uptake at human DAT expressed in HEK293 cells after 15 to 20 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89G42PubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50469308(CHEMBL4283496)copy SMILEScopy InChI
Affinity DataIC50: 830nMAssay Description:Inhibition of [3H]serotonin uptake at human SERT expressed in HEK293 cells after 15 to 20 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89G42PubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50261032(CHEMBL4061167)copy SMILEScopy InChI
Affinity DataIC50: 880nMAssay Description:Inhibition of re-uptake of [3H]-5-HT at human SERT expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9ZPVPubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50235723(CHEMBL4082902)copy SMILEScopy InChI
Affinity DataIC50: 980nMAssay Description:Inhibition of [3H]dopamine uptake at human DAT expressed in HEK293 cells after 15 to 20 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89G42PubMed
TargetAndrogen receptor(Mus musculus)
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50430946(CHEMBL2336980)copy SMILEScopy InChI
Affinity DataIC50: 990nMAssay Description:Agonist activity at mouse androgen receptor assessed as inhibition of transactivation after 24 hrs by cell-based luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PK0HHMPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50469307(CHEMBL4283917)copy SMILEScopy InChI
Affinity DataIC50: 990nMAssay Description:Inhibition of [3H]serotonin uptake at human SERT expressed in HEK293 cells after 15 to 20 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89G42PubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50462936(CHEMBL4248022)copy SMILEScopy InChI
Affinity DataIC50: 1.01E+3nMAssay Description:Inhibition of human SERT expressed in HEK293 cells assessed as reduction in [3H]5-HT uptake by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474DHGPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50469311(CHEMBL4295202)copy SMILEScopy InChI
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibition of [3H]serotonin uptake at human SERT expressed in HEK293 cells after 15 to 20 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89G42PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50051985(CHEMBL288826 | N-[3-(4-Benzyl-piperidin-1-yl)-prop...)copy SMILEScopy InChI
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of [3H]dopamine uptake at DAT (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89G42PubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50469316(CHEMBL4277619)copy SMILEScopy InChI
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of [3H]serotonin uptake at human SERT expressed in HEK293 cells after 15 to 20 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89G42PubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50462924(CHEMBL4251399)copy SMILEScopy InChI
Affinity DataIC50: 1.17E+3nMAssay Description:Inhibition of human SERT expressed in HEK293 cells assessed as reduction in [3H]5-HT uptake by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474DHGPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50155558(CHEMBL3774957)copy SMILEScopy InChI
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of re-uptake of [3H]-5-HT at human SERT expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9ZPVPubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50048392(2-(tert-butylamino)-1-(3-chlorophenyl)propan-1-one...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human DAT expressed in HEK293 cells assessed as reduction in [3H]-DA uptake by micro beta scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474DHGPubMedDrugBank
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50048392(2-(tert-butylamino)-1-(3-chlorophenyl)propan-1-one...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of re-uptake of [3H]-DA at human DAT expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9ZPVPubMedDrugBank
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
College of Pharmacy and Research Institute of Drug Development, Chonnam National University, Gwangju 61186, Republic of Korea.

Curated by ChEMBL
LigandPNGBDBM50469311(CHEMBL4295202)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of [3H]norepinephrine uptake at human NET expressed in HEK293 cells after 15 to 20 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89G42PubMed
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