Compile Data Set for Download or QSAR
Found 74 with Last Name = 'perez fernandez' and Initial = 'di'
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350906(3-Phenyl-2-(2-naphthylmethylthio)-4-oxo-3,4-dihydr...)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350888(3-Phenyl-2-neopentylthio-4-oxo-3,4-dihydroquinazol...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350903(3-(2-Methylphenyl)-2-(3-pyridylmethylthio)-4-oxo-3...)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350886(2-Cyclohexylmethylthio-3-phenyl-4-oxo-3,4-dihydroq...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350902(8-Chloro-2-(3-pyridylmethylthio)-4-oxo-3,4-dihydro...)copy SMILEScopy InChI
Affinity DataIC50: 540nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350899(2-Benzylthio-3-phenyl-4-oxo-3,4-dihydroquinazoline...)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350901(3-Phenyl-2-(3-pyridylmethylthio)-4-oxo-3,4-dihydro...)copy SMILEScopy InChI
Affinity DataIC50: 700nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350900(3-Phenyl-2-(2-pyridylmethylthio)-4-oxo-3,4-dihydro...)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350890(8-Chloro-3-phenyl-2-neopentylthio-4-oxo-3,4-dihydr...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350891(3-(2-Methylphenyl)-2-neopentylthio-4-oxo-3,4-dihyd...)copy SMILEScopy InChI
Affinity DataIC50: 1.85E+3nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294083(6-Bromo-N′-dodecanoyl-1-ethyl-4-hydroxy-2-ox...)copy SMILEScopy InChI
Affinity DataIC50: 2.01E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294083(6-Bromo-N′-dodecanoyl-1-ethyl-4-hydroxy-2-ox...)copy SMILEScopy InChI
Affinity DataIC50: 2.01E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350887(3-(2-Bromophenyl)-2-cyclohexylmethylthio-4-oxo-3,4...)copy SMILEScopy InChI
Affinity DataIC50: 2.11E+3nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350898(8-Chloro-2-ethylthio-3-(2,6-difluorophenyl)-4-oxo-...)copy SMILEScopy InChI
Affinity DataIC50: 2.44E+3nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294091(7-Chloro-N′-dodecanoyl-1-ethyl-4-hydroxy-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 2.48E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294091(7-Chloro-N′-dodecanoyl-1-ethyl-4-hydroxy-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 2.48E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350904(3-Phenyl-2-(4-pyridylmethylthio)-4-oxo-3,4-dihydro...)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM50384798(CHEMBL2037482 | US9585879, 6 | US9757369, 6)copy SMILEScopy InChI
Affinity DataIC50: 2.85E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM50384798(CHEMBL2037482 | US9585879, 6 | US9757369, 6)copy SMILEScopy InChI
Affinity DataIC50: 2.85E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294072(7-Chloro-N′-dodecanoyl-4-hydroxy-2-oxo-2-hyd...)copy SMILEScopy InChI
Affinity DataIC50: 3.12E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM339879(7-Chloro-N′-dodecanoyl-4-hydroxy-2-oxo-2-hyd...)copy SMILEScopy InChI
Affinity DataIC50: 3.12E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294087(6-Chloro-N′-dodecanoyl-1-ethyl-4-hydroxy-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 3.18E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294087(6-Chloro-N′-dodecanoyl-1-ethyl-4-hydroxy-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 3.18E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM339885(6-Bromo-N′-dodecanoyl-4-hydroxy-2-oxo-2-hydr...)copy SMILEScopy InChI
Affinity DataIC50: 3.54E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294078(6-Bromo-N′-dodecanoyl-4-hydroxy-2-oxo-2-hydr...)copy SMILES
Affinity DataIC50: 3.54E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294079(6-Chloro-N′-dodecanoyl-4-hydroxy-2-oxo-2-hyd...)copy SMILES
Affinity DataIC50: 3.81E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM339886(6-Chloro-N′-dodecanoyl-4-hydroxy-2-oxo-2-hyd...)copy SMILEScopy InChI
Affinity DataIC50: 3.81E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294089(7-Chloro-N′-dodecanoyl-4-hydroxy-1-methyl-2-...)copy SMILEScopy InChI
Affinity DataIC50: 4.03E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294089(7-Chloro-N′-dodecanoyl-4-hydroxy-1-methyl-2-...)copy SMILEScopy InChI
Affinity DataIC50: 4.03E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294081(6-Bromo-N′-dodecanoyl-4-hydroxy-1-methyl-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 4.28E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294081(6-Bromo-N′-dodecanoyl-4-hydroxy-1-methyl-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 4.28E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM339875(N′-Dodecanoyl-4-hydroxy-1-methyl-2-oxo-1,2-d...)copy SMILEScopy InChI
Affinity DataIC50: 4.47E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294070(N′-Dodecanoyl-4-hydroxy-2-oxo-2-hydroquinoli...)copy SMILEScopy InChI
Affinity DataIC50: 4.47E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350893(2-Cyclopropylmethylthio-3-(2,6-difluorophenyl)-8-m...)copy SMILEScopy InChI
Affinity DataIC50: 4.56E+3nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294090(7-Chloro-1-ethyl-4-hydroxy-N′-octanoyl-2-oxo...)copy SMILEScopy InChI
Affinity DataIC50: 4.83E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294090(7-Chloro-1-ethyl-4-hydroxy-N′-octanoyl-2-oxo...)copy SMILEScopy InChI
Affinity DataIC50: 4.83E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294076(1-(cyclopropylmethyl)-N′-dodecanoyl-4-hydrox...)copy SMILEScopy InChI
Affinity DataIC50: 5.25E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294076(1-(cyclopropylmethyl)-N′-dodecanoyl-4-hydrox...)copy SMILEScopy InChI
Affinity DataIC50: 5.25E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294077(1-Benzyl-N′-dodecanoyl-4-hydroxy-2-oxo-1,2-d...)copy SMILEScopy InChI
Affinity DataIC50: 5.51E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294077(1-Benzyl-N′-dodecanoyl-4-hydroxy-2-oxo-1,2-d...)copy SMILEScopy InChI
Affinity DataIC50: 5.51E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM339880(6-Fluoro-N′-dodecanoyl-4-hydroxy-2-oxo-2-hyd...)copy SMILEScopy InChI
Affinity DataIC50: 5.81E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294073(6-Fluoro-N′-dodecanoyl-4-hydroxy-2-oxo-2-hyd...)copy SMILEScopy InChI
Affinity DataIC50: 5.81E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294085(6-Chloro-N′-dodecanoyl-4-hydroxy-1-methyl-2-...)copy SMILEScopy InChI
Affinity DataIC50: 5.95E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294085(6-Chloro-N′-dodecanoyl-4-hydroxy-1-methyl-2-...)copy SMILEScopy InChI
Affinity DataIC50: 5.95E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294092(1-Benzyl-7-chloro-4-hydroxy-N′-octanoyl-2-ox...)copy SMILEScopy InChI
Affinity DataIC50: 5.96E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294092(1-Benzyl-7-chloro-4-hydroxy-N′-octanoyl-2-ox...)copy SMILEScopy InChI
Affinity DataIC50: 5.96E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294093(1-Benzyl-7-chloro-N′dodecanoyl-4-hydroxy-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 5.99E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294093(1-Benzyl-7-chloro-N′dodecanoyl-4-hydroxy-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 5.99E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294080(6-Bromo-4-hydroxy-1-methyl-N′-octanoyl-2-oxo...)copy SMILEScopy InChI
Affinity DataIC50: 6.28E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294080(6-Bromo-4-hydroxy-1-methyl-N′-octanoyl-2-oxo...)copy SMILEScopy InChI
Affinity DataIC50: 6.28E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
Displayed 1 to 50 (of 74 total ) | Next | Last >>
Jump to: