Compile Data Set for Download or QSAR
Found 67 with Last Name = 'bull' and Initial = 'dj'
TargetCarboxypeptidase B2(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50305346((S)-2-(2-aminoethoxy)-3-(1-phenyl-1H-imidazol-4-yl...)copy SMILEScopy InChI
Affinity DataKi:  3.5nMAssay Description:Inhibition of active form of human recombinant TAFI assessed as substrate turnover every 15 seconds for 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1038RPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50305347((S)-2-(2-aminoethoxy)-3-(1-(4-tert-butylphenyl)-1H...)copy SMILEScopy InChI
Affinity DataKi:  5.70nMAssay Description:Inhibition of active form of human recombinant TAFI assessed as substrate turnover every 15 seconds for 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1038RPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50305351((S)-2-((R)-1-aminopropan-2-yloxy)-3-(1-(pyridin-2-...)copy SMILEScopy InChI
Affinity DataKi:  5.80nMAssay Description:Inhibition of active form of human recombinant TAFI assessed as substrate turnover every 15 seconds for 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1038RPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50305345((S)-2-(2-aminoethoxy)-3-(1-propyl-1H-imidazol-4-yl...)copy SMILEScopy InChI
Affinity DataKi:  6.70nMAssay Description:Inhibition of active form of human recombinant TAFI assessed as substrate turnover every 15 seconds for 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1038RPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50305352((S)-2-((R)-1-aminopropan-2-yloxy)-3-(1-phenyl-1H-i...)copy SMILEScopy InChI
Affinity DataKi:  7.5nMAssay Description:Inhibition of active form of human recombinant TAFI assessed as substrate turnover every 15 seconds for 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1038RPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50305348((S)-2-(2-aminoethoxy)-3-(1-(2-cyclohexylethyl)-1H-...)copy SMILEScopy InChI
Affinity DataKi:  8.20nMAssay Description:Inhibition of active form of human recombinant TAFI assessed as substrate turnover every 15 seconds for 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1038RPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50305349((+/-)-2-(2-aminoethoxy)-3-(1-butyl-1H-imidazol-4-y...)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Inhibition of active form of human recombinant TAFI assessed as substrate turnover every 15 seconds for 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1038RPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50226610((2S)-5-AMINO-2-[(1-PROPYL-1H-IMIDAZOL-4-YL)METHYL]...)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:Inhibition of active form of human recombinant TAFI assessed as substrate turnover every 15 seconds for 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1038RPubMed
TargetCarboxypeptidase B(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50305346((S)-2-(2-aminoethoxy)-3-(1-phenyl-1H-imidazol-4-yl...)copy SMILEScopy InChI
Affinity DataKi:  27nMAssay Description:Inhibition of human pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1038RPubMed
TargetCarboxypeptidase B(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50305348((S)-2-(2-aminoethoxy)-3-(1-(2-cyclohexylethyl)-1H-...)copy SMILEScopy InChI
Affinity DataKi:  27nMAssay Description:Inhibition of human pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1038RPubMed
TargetCarboxypeptidase B(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50305347((S)-2-(2-aminoethoxy)-3-(1-(4-tert-butylphenyl)-1H...)copy SMILEScopy InChI
Affinity DataKi:  49nMAssay Description:Inhibition of human pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1038RPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50305350((+/-)-2-(2-aminoethoxy)-3-(1-o-tolyl-1H-imidazol-4...)copy SMILEScopy InChI
Affinity DataKi:  65nMAssay Description:Inhibition of active form of human recombinant TAFI assessed as substrate turnover every 15 seconds for 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1038RPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50226606((S)-2-(2-aminoethylamino)-3-(1-propyl-1H-imidazol-...)copy SMILEScopy InChI
Affinity DataKi:  150nMAssay Description:Inhibition of active form of human recombinant TAFI assessed as substrate turnover every 15 seconds for 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1038RPubMed
TargetCarboxypeptidase B(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50226610((2S)-5-AMINO-2-[(1-PROPYL-1H-IMIDAZOL-4-YL)METHYL]...)copy SMILEScopy InChI
Affinity DataKi:  206nMAssay Description:Inhibition of human pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1038RPubMed
TargetCarboxypeptidase B(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50305345((S)-2-(2-aminoethoxy)-3-(1-propyl-1H-imidazol-4-yl...)copy SMILEScopy InChI
Affinity DataKi:  238nMAssay Description:Inhibition of human pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1038RPubMed
TargetCarboxypeptidase B(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50305352((S)-2-((R)-1-aminopropan-2-yloxy)-3-(1-phenyl-1H-i...)copy SMILEScopy InChI
Affinity DataKi:  240nMAssay Description:Inhibition of human pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1038RPubMed
TargetCarboxypeptidase B(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50305351((S)-2-((R)-1-aminopropan-2-yloxy)-3-(1-(pyridin-2-...)copy SMILEScopy InChI
Affinity DataKi:  265nMAssay Description:Inhibition of human pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1038RPubMed
TargetCarboxypeptidase B(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50305349((+/-)-2-(2-aminoethoxy)-3-(1-butyl-1H-imidazol-4-y...)copy SMILEScopy InChI
Affinity DataKi:  360nMAssay Description:Inhibition of human pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1038RPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50305353((+/-)-2-(2-(methylamino)ethoxy)-3-(1-propyl-1H-imi...)copy SMILEScopy InChI
Affinity DataKi:  407nMAssay Description:Inhibition of active form of human recombinant TAFI assessed as substrate turnover every 15 seconds for 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1038RPubMed
TargetCarboxypeptidase B2(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50305354((R)-2-(2-aminoethoxy)-3-(1-propyl-1H-imidazol-4-yl...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of active form of human recombinant TAFI assessed as substrate turnover every 15 seconds for 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1038RPubMed
TargetCarboxypeptidase B(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50226606((S)-2-(2-aminoethylamino)-3-(1-propyl-1H-imidazol-...)copy SMILEScopy InChI
Affinity DataKi:  1.16E+3nMAssay Description:Inhibition of human pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1038RPubMed
TargetCarboxypeptidase B(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50305350((+/-)-2-(2-aminoethoxy)-3-(1-o-tolyl-1H-imidazol-4...)copy SMILEScopy InChI
Affinity DataKi:  2.72E+3nMAssay Description:Inhibition of human pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1038RPubMed
TargetCarboxypeptidase B(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50305353((+/-)-2-(2-(methylamino)ethoxy)-3-(1-propyl-1H-imi...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1038RPubMed
TargetCarboxypeptidase B(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50305354((R)-2-(2-aminoethoxy)-3-(1-propyl-1H-imidazol-4-yl...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human pancreatic carboxypeptidase BMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1038RPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50033236(8,9-Dichloro-2-methyl-5-[4-(2-methyl-imidazo[4,5-c...)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50033242(3-Cyclohexyl-6-[4-(2-methyl-imidazo[4,5-c]pyridin-...)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50033257(1,8-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50033240(1-Methyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50033238(3-(4-Chloro-phenyl)-1,8-dimethyl-5-[4-(2-methyl-im...)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50033264(3-Cyclohexyl-1,8-dimethyl-5-[4-(2-methyl-imidazo[4...)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50033260(3-Isobutoxymethyl-1,8-dimethyl-5-[4-(2-methyl-imid...)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50033234(1,3-Dimethyl-7-[4-(2-methyl-imidazo[4,5-c]pyridin-...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50033233(8,9-Dichloro-1-methyl-5-[4-(2-methyl-imidazo[4,5-c...)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50033229(8,9-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50033249(5,7,9-Trimethyl-2-[4-(2-methyl-imidazo[4,5-c]pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50033245(8-Bromo-5-methyl-2-[4-(2-methyl-imidazo[4,5-c]pyri...)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50033255(1,8-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50033232(8,9-Dichloro-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50033263(8,9-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)copy SMILEScopy InChI
Affinity DataIC50: 2.30nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50033231(1,8,9-Trimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50033251(1,8-Dimethyl-5-[4-(2-methyl-imidazo[4,5-c]pyridin-...)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50033246(5-Methyl-2-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50033243(1-Methyl-7-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 2.70nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50033230(5-Methyl-2-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50033241(3-Isopropyl-1,8-dimethyl-5-[4-(2-methyl-imidazo[4,...)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50033268(5-Methyl-2-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50033254(8-Bromo-2-[4-(2-methyl-imidazo[4,5-c]pyridin-1-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50033239(8-Bromo-1-methyl-4-[4-(2-methyl-imidazo[4,5-c]pyri...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50033235(7-[4-(2-Methyl-imidazo[4,5-c]pyridin-1-yl)-phenyl]...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Pfizer Central Research

Curated by ChEMBL
LigandPNGBDBM50004633((S)-4-(2-Chloro-phenyl)-6-methyl-2-[4-(2-methyl-im...)copy SMILEScopy InChI
Affinity DataIC50: 4.30nMAssay Description:In vitro antagonist activity against platelet activating factor (PAF) receptor, using washed rabbit plateletsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JS9R2XPubMed
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