Compile Data Set for Download or QSAR
Found 21 with Last Name = 'thomas' and Initial = 'dj'
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Kalypsys, Inc.

Curated by ChEMBL
LigandPNGBDBM50317611(4-(3,5-dichloropyridin-4-ylamino)-8-(3-(dimethylam...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZMFPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Kalypsys, Inc.

Curated by ChEMBL
LigandPNGBDBM14775(3-(cyclopentyloxy)-N-(3,5-dichloropyridin-4-yl)-4-...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hrMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Kalypsys, Inc.

Curated by ChEMBL
LigandPNGBDBM50317610(9-(4-(3,5-dichloropyridin-4-ylamino)-7-methoxy-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZMFPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Kalypsys, Inc.

Curated by ChEMBL
LigandPNGBDBM50317616(4-(3,5-dichloropyridin-4-ylamino)-8-(8-(dimethylam...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZMFPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Kalypsys, Inc.

Curated by ChEMBL
LigandPNGBDBM50317609(8-(4-(3,5-dichloropyridin-4-ylamino)-7-methoxy-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZMFPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Kalypsys, Inc.

Curated by ChEMBL
LigandPNGBDBM50317615(4-(3,5-dichloropyridin-4-ylamino)-8-(7-(dimethylam...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZMFPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Kalypsys, Inc.

Curated by ChEMBL
LigandPNGBDBM50317603(8-(cyclopentyloxy)-4-(3,5-dichloropyridin-4-ylamin...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hrMore data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Kalypsys, Inc.

Curated by ChEMBL
LigandPNGBDBM50317604(2-(4-(3,5-dichloropyridin-4-ylamino)-7-methoxy-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZMFPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Kalypsys, Inc.

Curated by ChEMBL
LigandPNGBDBM50317614(4-(3,5-dichloropyridin-4-ylamino)-8-(6-(dimethylam...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZMFPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Kalypsys, Inc.

Curated by ChEMBL
LigandPNGBDBM50317608(7-(4-(3,5-dichloropyridin-4-ylamino)-7-methoxy-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZMFPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Kalypsys, Inc.

Curated by ChEMBL
LigandPNGBDBM50317613(4-(3,5-dichloropyridin-4-ylamino)-8-(5-(dimethylam...)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZMFPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Kalypsys, Inc.

Curated by ChEMBL
LigandPNGBDBM50317607(6-(4-(3,5-dichloropyridin-4-ylamino)-7-methoxy-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZMFPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Kalypsys, Inc.

Curated by ChEMBL
LigandPNGBDBM50317612(4-(3,5-dichloropyridin-4-ylamino)-8-(4-(dimethylam...)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZMFPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Kalypsys, Inc.

Curated by ChEMBL
LigandPNGBDBM50317606(5-(4-(3,5-dichloropyridin-4-ylamino)-7-methoxy-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 80nMAssay Description:Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZMFPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Kalypsys, Inc.

Curated by ChEMBL
LigandPNGBDBM50092350((5-Cyclopentyloxy-6-methoxy-phthalazin-1-yl)-(3,5-...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZMFPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Kalypsys, Inc.

Curated by ChEMBL
LigandPNGBDBM50317599(5-(cyclopentyloxy)-N-(3,5-dichloropyridin-4-yl)-6-...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZMFPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Kalypsys, Inc.

Curated by ChEMBL
LigandPNGBDBM50317605(4-(4-(3,5-dichloropyridin-4-ylamino)-7-methoxy-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZMFPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Kalypsys, Inc.

Curated by ChEMBL
LigandPNGBDBM50317600(8-(cyclopentyloxy)-N-(3,5-dichloropyridin-4-yl)-7-...)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZMFPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Kalypsys, Inc.

Curated by ChEMBL
LigandPNGBDBM50317598(8-(cyclopentyloxy)-N-(3,5-dichloropyridin-4-yl)-7-...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZMFPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Kalypsys, Inc.

Curated by ChEMBL
LigandPNGBDBM50317601(3,5-dichloro-N-(7-(cyclopentyloxy)-6-methoxybenzof...)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZMFPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Kalypsys, Inc.

Curated by ChEMBL
LigandPNGBDBM50317602(3,5-dichloro-N-(8-(cyclopentyloxy)-7-methoxychroma...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human His6-tagged PDE4B (152-487) expressed in Escherichia coli BL21 (DE3) after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD6ZMFPubMed