Compile Data Set for Download or QSAR
Found 184 with Last Name = 'buckley' and Initial = 'dl'
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50458963(CHEMBL4209902)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM25121(4-{[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50458971(CHEMBL4215729)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50458969(CHEMBL4207165)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50458968(CHEMBL4216442)copy SMILEScopy InChI
Affinity DataIC50: 8.40nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50458967(CHEMBL4202820)copy SMILEScopy InChI
Affinity DataIC50: 8.60nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50458960(CHEMBL4216875)copy SMILEScopy InChI
Affinity DataIC50: 8.70nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50458962(CHEMBL4213276)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50458951(CHEMBL4206171)copy SMILEScopy InChI
Affinity DataIC50: 9.90nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Dana Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50503068(CHEMBL4483587)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Displacement of biotinylated probe from human TAF1 bromodomain 2 (1522 to 1656 residues) expressed in Escherichia coli BL21 (DE3) by alphascreen assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63T8PubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Dana Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50503091(CHEMBL4589721)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Displacement of biotinylated probe from human TAF1 bromodomain 2 (1522 to 1656 residues) expressed in Escherichia coli BL21 (DE3) by alphascreen assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63T8PubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50458965(CHEMBL4210571)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50458964(CHEMBL4206052)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50458952(CHEMBL4203571)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50458966(CHEMBL4207437)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Dana Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50503081(CHEMBL4534000)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Displacement of biotinylated probe from human TAF1 bromodomain 2 (1522 to 1656 residues) expressed in Escherichia coli BL21 (DE3) by alphascreen assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63T8PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50112336(CHEMBL3609305)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50112344(CHEMBL3609314)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Displacement of Bio-JQ1 from recombinant human His6 tagged BRD4 bromodomain 1 by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63T8PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50503091(CHEMBL4589721)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:Displacement of Bio-JQ1 from recombinant human His6 tagged BRD4 bromodomain 1 by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63T8PubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50458959(CHEMBL4214823)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Dana Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50503078(CHEMBL4542872)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Displacement of biotinylated probe from human TAF1 bromodomain 2 (1522 to 1656 residues) expressed in Escherichia coli BL21 (DE3) by alphascreen assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63T8PubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50458966(CHEMBL4207437)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50458955(CHEMBL4209192)copy SMILEScopy InChI
Affinity DataIC50: 47nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50503090(CHEMBL4466613)copy SMILEScopy InChI
Affinity DataIC50: 47nMAssay Description:Displacement of Bio-JQ1 from recombinant human His6 tagged BRD4 bromodomain 1 by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63T8PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50503081(CHEMBL4534000)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Displacement of Bio-JQ1 from recombinant human His6 tagged BRD4 bromodomain 1 by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63T8PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50503068(CHEMBL4483587)copy SMILEScopy InChI
Affinity DataIC50: 49nMAssay Description:Displacement of Bio-JQ1 from recombinant human His6 tagged BRD4 bromodomain 1 by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63T8PubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50112335(CHEMBL3609304)copy SMILEScopy InChI
Affinity DataIC50: 54nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50458970(CHEMBL4206381)copy SMILEScopy InChI
Affinity DataIC50: 59nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50503085(CHEMBL4437749)copy SMILEScopy InChI
Affinity DataIC50: 62nMAssay Description:Displacement of Bio-JQ1 from recombinant human His6 tagged BRD4 bromodomain 1 by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63T8PubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Dana Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50503087(CHEMBL4573352)copy SMILEScopy InChI
Affinity DataIC50: 63nMAssay Description:Displacement of biotinylated probe from human TAF1 bromodomain 2 (1522 to 1656 residues) expressed in Escherichia coli BL21 (DE3) by alphascreen assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50503086(CHEMBL4468126)copy SMILEScopy InChI
Affinity DataIC50: 63nMAssay Description:Displacement of Bio-JQ1 from recombinant human His6 tagged BRD4 bromodomain 1 by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63T8PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50503084(CHEMBL4440443)copy SMILEScopy InChI
Affinity DataIC50: 68nMAssay Description:Displacement of Bio-JQ1 from recombinant human His6 tagged BRD4 bromodomain 1 by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63T8PubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Dana Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50503079(CHEMBL4556917)copy SMILEScopy InChI
Affinity DataIC50: 72nMAssay Description:Displacement of biotinylated probe from human TAF1 bromodomain 2 (1522 to 1656 residues) expressed in Escherichia coli BL21 (DE3) by alphascreen assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63T8PubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50458958(CHEMBL4215910)copy SMILEScopy InChI
Affinity DataIC50: 78nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Dana Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50503074(CHEMBL4474288)copy SMILEScopy InChI
Affinity DataIC50: 82nMAssay Description:Displacement of biotinylated probe from human TAF1 bromodomain 2 (1522 to 1656 residues) expressed in Escherichia coli BL21 (DE3) by alphascreen assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50458963(CHEMBL4209902)copy SMILEScopy InChI
Affinity DataIC50: 84nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Dana Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50503084(CHEMBL4440443)copy SMILEScopy InChI
Affinity DataIC50: 87nMAssay Description:Displacement of biotinylated probe from human TAF1 bromodomain 2 (1522 to 1656 residues) expressed in Escherichia coli BL21 (DE3) by alphascreen assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63T8PubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Dana Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50503070(CHEMBL4539891)copy SMILEScopy InChI
Affinity DataIC50: 89nMAssay Description:Displacement of biotinylated probe from human TAF1 bromodomain 2 (1522 to 1656 residues) expressed in Escherichia coli BL21 (DE3) by alphascreen assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Dana Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50503090(CHEMBL4466613)copy SMILEScopy InChI
Affinity DataIC50: 93nMAssay Description:Displacement of biotinylated probe from human TAF1 bromodomain 2 (1522 to 1656 residues) expressed in Escherichia coli BL21 (DE3) by alphascreen assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63T8PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50458956(CHEMBL4202678)copy SMILEScopy InChI
Affinity DataIC50: 94nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50458968(CHEMBL4216442)copy SMILEScopy InChI
Affinity DataIC50: 95nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50458956(CHEMBL4202678)copy SMILEScopy InChI
Affinity DataIC50: 95nMAssay Description:Inhibition of human recombinant PLK1 by Z-Lyte assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50503083(CHEMBL4583926)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Displacement of Bio-JQ1 from recombinant human His6 tagged BRD4 bromodomain 1 by alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Dana Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50112344(CHEMBL3609314)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Displacement of biotinylated probe from human TAF1 bromodomain 2 (1522 to 1656 residues) expressed in Escherichia coli BL21 (DE3) by alphascreen assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P63T8PubMed
TargetBromodomain testis-specific protein(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50458966(CHEMBL4207437)copy SMILEScopy InChI
Affinity DataIC50: 102nMAssay Description:Inhibition of BRDT-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetBromodomain testis-specific protein(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50365262((+)-JQ1 | (S)-JQ1 (1) | CHEMBL1957266 | JQ1 | US10...)copy SMILEScopy InChI
Affinity DataIC50: 103nMAssay Description:Inhibition of BRDT-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50458965(CHEMBL4210571)copy SMILEScopy InChI
Affinity DataIC50: 104nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50458961(CHEMBL4210414)copy SMILEScopy InChI
Affinity DataIC50: 107nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University of Massachusetts-Boston

Curated by ChEMBL
LigandPNGBDBM50458960(CHEMBL4216875)copy SMILEScopy InChI
Affinity DataIC50: 107nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) incubated for 1 hr by AlphaScreen biotin-JQ1 competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP55WQPubMed
Displayed 1 to 50 (of 184 total ) | Next | Last >>
Jump to: