Affinity DataKi: 0.110nMAssay Description:Reversible binding affinity to human EGFR L858R/ T790M double mutant expressed in baculovirus by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of EGFR T790M/L858R double mutant (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Reversible binding affinity to human EGFR L858R/ T790M double mutant expressed in baculovirus by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Reversible binding affinity to human EGFR L858R/ T790M double mutant expressed in baculovirus by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of EGFR T790M/L858R double mutant (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibition of EGFR T790M/L858R double mutant (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibition of EGFR T790M/L858R double mutant (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Reversible binding affinity to human EGFR L858R/ T790M double mutant expressed in baculovirus by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Reversible binding affinity to human EGFR L858R/ T790M double mutant expressed in baculovirus by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Reversible binding affinity to human EGFR L858R/ T790M double mutant expressed in baculovirus by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Inhibition of EGFR T790M/L858R double mutant (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity of compound towards 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Reversible binding affinity to human EGFR L858R/ T790M double mutant expressed in baculovirus by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Reversible binding affinity to human EGFR L858R/ T790M double mutant expressed in baculovirus by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Affinity at D2 dopamine receptor on CHO cell membranes by [3H]-PNU-86170 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Binding affinity of the compound towards 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Affinity at D2 dopamine receptor on CHO cell membranes by [3H]-PNU-86170 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Inhibition of EGFR T790M/L858R double mutant (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 6.10nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Reversible binding affinity to human EGFR L858R/ T790M double mutant expressed in baculovirus by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Reversible binding affinity to human EGFR L858R/ T790M double mutant expressed in baculovirus by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Inhibition of EGFR T790M/L858R double mutant (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Inhibition of EGFR T790M/L858R double mutant (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Reversible binding affinity to human EGFR L858R/ T790M double mutant expressed in baculovirus by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition of EGFR T790M/L858R double mutant (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Reversible binding affinity to human EGFR L858R/ T790M double mutant expressed in baculovirus by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Affinity at rat D3 dopamine receptor on CHO cell membranes by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Affinity at rat D3 dopamine receptor on CHO cell membranes by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Reversible binding affinity to human EGFR L858R/ T790M double mutant expressed in baculovirus by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Inhibition of EGFR T790M/L858R double mutant (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Inhibition of EGFR T790M/L858R double mutant (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Inhibition of EGFR T790M/L858R double mutant (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligand.More data for this Ligand-Target Pair