Compile Data Set for Download or QSAR
Found 197 with Last Name = 'glover' and Initial = 'dm'
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81438(CDK Inhibitor, 11)copy SMILEScopy InChI
Affinity DataKi:  0.110nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81433(CDK Inhibitor, 6)copy SMILEScopy InChI
Affinity DataKi:  0.290nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81441(CDK Inhibitor, 14)copy SMILEScopy InChI
Affinity DataKi:  0.380nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetAurora kinase A(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319623(4-(2,4-Dimethylthiazol-5-yl)-N-(3,4,5-trimethoxyph...)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Inhibition of human recombinant Aurora A after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81439(CDK Inhibitor, 12)copy SMILEScopy InChI
Affinity DataKi:  0.520nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81440(CDK Inhibitor, 13)copy SMILEScopy InChI
Affinity DataKi:  0.560nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81430(CDK Inhibitor, 3)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81434(CDK Inhibitor, 7)copy SMILEScopy InChI
Affinity DataKi:  0.960nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetAurora kinase A(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319622(CHEMBL1083152 | N,4-Dimethyl-5-(2-(3,4,5-trimethox...)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Inhibition of human recombinant Aurora A after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM8061(2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 32 | 4...)copy SMILEScopy InChI
Affinity DataKi: <1nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81433(CDK Inhibitor, 6)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81439(CDK Inhibitor, 12)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM50229973((4-(2-Amino-4-methylthiazol-5-yl)pyrimidin-2-yl)-(...)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Inhibition of CDK2More data for this Ligand-Target Pair
TargetAurora kinase B(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319623(4-(2,4-Dimethylthiazol-5-yl)-N-(3,4,5-trimethoxyph...)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Inhibition of human recombinant Aurora B after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81441(CDK Inhibitor, 14)copy SMILEScopy InChI
Affinity DataKi:  2.30nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81430(CDK Inhibitor, 3)copy SMILEScopy InChI
Affinity DataKi:  2.40nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81440(CDK Inhibitor, 13)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetAurora kinase B(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319622(CHEMBL1083152 | N,4-Dimethyl-5-(2-(3,4,5-trimethox...)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Inhibition of human recombinant Aurora B after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetAurora kinase A(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319621(CHEMBL1086088 | N-Ethyl-4-methyl-5-(2-(3,4,5-trime...)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Inhibition of human recombinant Aurora A after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetAurora kinase B(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319616(1-(4-(4-(4-(2-Amino-4-methylthiazol-5-yl)pyrimidin...)copy SMILEScopy InChI
Affinity DataKi:  3.80nMAssay Description:Inhibition of human recombinant Aurora B after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM50229973((4-(2-Amino-4-methylthiazol-5-yl)pyrimidin-2-yl)-(...)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Inhibition of CDK9More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetAurora kinase B(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319620(CHEMBL1084715 | N-(4-(4-(2-(Ethylamino)-4-methylth...)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Inhibition of human recombinant Aurora B after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetAurora kinase A(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319619(4-(2,4-Dimethylthiazol-5-yl)-N-(4-morpholinophenyl...)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Inhibition of human recombinant Aurora A after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81438(CDK Inhibitor, 11)copy SMILEScopy InChI
Affinity DataKi:  4.10nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81431(CDK Inhibitor, 4)copy SMILEScopy InChI
Affinity DataKi:  4.30nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81432(CDK Inhibitor, 5)copy SMILEScopy InChI
Affinity DataKi:  4.30nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81429(CDK Inhibitor, 2)copy SMILEScopy InChI
Affinity DataKi:  4.5nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM8061(2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 32 | 4...)copy SMILEScopy InChI
Affinity DataKi:  4.60nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetAurora kinase A(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319620(CHEMBL1084715 | N-(4-(4-(2-(Ethylamino)-4-methylth...)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Inhibition of human recombinant Aurora A after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81435(CDK Inhibitor, 8)copy SMILEScopy InChI
Affinity DataKi:  5.90nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81440(CDK Inhibitor, 13)copy SMILEScopy InChI
Affinity DataKi:  5.90nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetAurora kinase B(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319617(CHEMBL1084630 | N-Ethyl-4-methyl-5-(2-(4-morpholin...)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Inhibition of human recombinant Aurora B after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM50319622(CHEMBL1083152 | N,4-Dimethyl-5-(2-(3,4,5-trimethox...)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Inhibition of CDK9More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetAurora kinase B(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319621(CHEMBL1086088 | N-Ethyl-4-methyl-5-(2-(3,4,5-trime...)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Inhibition of human recombinant Aurora B after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81436(CDK Inhibitor, 9)copy SMILEScopy InChI
Affinity DataKi:  6.70nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81439(CDK Inhibitor, 12)copy SMILEScopy InChI
Affinity DataKi:  6.80nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetAurora kinase A(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM8066(2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 37 | 4...)copy SMILEScopy InChI
Affinity DataKi:  6.90nMAssay Description:Inhibition of human recombinant Aurora A after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetAurora kinase A(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319616(1-(4-(4-(4-(2-Amino-4-methylthiazol-5-yl)pyrimidin...)copy SMILEScopy InChI
Affinity DataKi:  7.60nMAssay Description:Inhibition of human recombinant Aurora A after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81434(CDK Inhibitor, 7)copy SMILEScopy InChI
Affinity DataKi:  7.60nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetAurora kinase A(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50277583(2-amino-4-methyl-1,3-thiazol-5-yl)-N-[4-(morpholin...)copy SMILEScopy InChI
Affinity DataKi:  8nMAssay Description:Inhibition of human recombinant Aurora A after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetAurora kinase A(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319627(1-(4-(4-(4-(2,4-Dimethylthiazol-5-yl)pyrimidin-2-y...)copy SMILEScopy InChI
Affinity DataKi:  8.20nMAssay Description:Inhibition of human recombinant Aurora A after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81437(CDK Inhibitor, 10)copy SMILEScopy InChI
Affinity DataKi:  8.5nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM50319620(CHEMBL1084715 | N-(4-(4-(2-(Ethylamino)-4-methylth...)copy SMILEScopy InChI
Affinity DataKi:  9nMAssay Description:Inhibition of CDK9More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetAurora kinase B(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319619(4-(2,4-Dimethylthiazol-5-yl)-N-(4-morpholinophenyl...)copy SMILEScopy InChI
Affinity DataKi:  9nMAssay Description:Inhibition of human recombinant Aurora B after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM81430(CDK Inhibitor, 3)copy SMILEScopy InChI
Affinity DataKi:  9.10nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F3QPubMed
TargetAurora kinase B(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50277583(2-amino-4-methyl-1,3-thiazol-5-yl)-N-[4-(morpholin...)copy SMILEScopy InChI
Affinity DataKi:  9.20nMAssay Description:Inhibition of human recombinant Aurora B after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetAurora kinase A(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319626(4-(2,4-Dimethylthiazol-5-yl)-N-(4-(4-(methylsulfon...)copy SMILEScopy InChI
Affinity DataKi:  9.20nMAssay Description:Inhibition of human recombinant Aurora A after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetAurora kinase B(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319618(CHEMBL1084629 | N,4-Dimethyl-5-(2-(4-morpholinophe...)copy SMILEScopy InChI
Affinity DataKi:  9.40nMAssay Description:Inhibition of human recombinant Aurora B after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetAurora kinase B(Homo sapiens (Human))
Cyclacel Ltd.

Curated by ChEMBL
LigandPNGBDBM50319615(1-(4-(4-(4-(4-Methyl-2-(methylamino)thiazol-5-yl)p...)copy SMILEScopy InChI
Affinity DataKi:  9.70nMAssay Description:Inhibition of human recombinant Aurora B after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Cyclacel Limited

LigandPNGBDBM50319623(4-(2,4-Dimethylthiazol-5-yl)-N-(3,4,5-trimethoxyph...)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Inhibition of CDK9More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2930T9DPubMed
Displayed 1 to 50 (of 197 total ) | Next | Last >>
Jump to: