Compile Data Set for Download or QSAR
Found 58 with Last Name = 'roll' and Initial = 'dm'
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50024382(CHEMBL189690)copy SMILEScopy InChI
Affinity DataKi:  0.0794nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50024388(CHEMBL190621)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50024390(CHEMBL372702)copy SMILEScopy InChI
Affinity DataKi:  0.310nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50024402(CHEMBL190232)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50024401(CHEMBL190712)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50024380(CHEMBL193124)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50024400(CHEMBL192719)copy SMILEScopy InChI
Affinity DataKi:  3.40nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50024393(CHEMBL426449)copy SMILEScopy InChI
Affinity DataKi:  3.80nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50024383(CHEMBL192121)copy SMILEScopy InChI
Affinity DataKi:  4.60nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50171860(((R)-3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin...)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50171860(((R)-3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin...)copy SMILEScopy InChI
Affinity DataKi:  5.10nMAssay Description:Inhibition constant for human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50024385(CHEMBL365588)copy SMILEScopy InChI
Affinity DataKi:  5.20nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50024389(CHEMBL370032)copy SMILEScopy InChI
Affinity DataKi:  6.40nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50024381(CHEMBL190713)copy SMILEScopy InChI
Affinity DataKi:  6.5nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50024397(CHEMBL372470)copy SMILEScopy InChI
Affinity DataKi:  6.60nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50024394(CHEMBL187733)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50024398(CHEMBL193080)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50024384(CHEMBL191318)copy SMILEScopy InChI
Affinity DataKi:  17nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50024391(CHEMBL364694)copy SMILEScopy InChI
Affinity DataKi:  32nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50024395(CHEMBL189945)copy SMILEScopy InChI
Affinity DataKi:  38nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50171864(((R)-3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin...)copy SMILEScopy InChI
Affinity DataKi:  42nMAssay Description:Inhibition constant for human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50171864(((R)-3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin...)copy SMILEScopy InChI
Affinity DataKi:  42nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50171862(((R)-3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin...)copy SMILEScopy InChI
Affinity DataKi:  43nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50171862(((R)-3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin...)copy SMILEScopy InChI
Affinity DataKi:  43nMAssay Description:Inhibition constant for human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50171863((4-Fluoro-phenyl)-((R)-3-hydroxycarbamoyl-3,4-dihy...)copy SMILEScopy InChI
Affinity DataKi:  52nMAssay Description:Inhibition constant for human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50171863((4-Fluoro-phenyl)-((R)-3-hydroxycarbamoyl-3,4-dihy...)copy SMILEScopy InChI
Affinity DataKi:  52nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50024399(CHEMBL364547)copy SMILEScopy InChI
Affinity DataKi:  59nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50024379(CHEMBL363351)copy SMILEScopy InChI
Affinity DataKi:  80nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50024386(CHEMBL189330)copy SMILEScopy InChI
Affinity DataKi:  95nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50024387(CHEMBL371362)copy SMILEScopy InChI
Affinity DataKi:  278nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50024392(CHEMBL190683)copy SMILEScopy InChI
Affinity DataKi:  316nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50171861(((S)-3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin...)copy SMILEScopy InChI
Affinity DataKi:  349nMAssay Description:Inhibition constant for human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
North Dakota State University

Curated by ChEMBL
LigandPNGBDBM50171861(((S)-3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin...)copy SMILEScopy InChI
Affinity DataKi:  349nMAssay Description:Inhibition of MOCAc-Pro-Leu-Gly-Leu-A2p (Dnp)-Ala-Arg-NH2 binding to human matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z89BZ5PubMed
TargetMineralocorticoid receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50228080(2',15'-dimethyl-5,5'-dioxo-(9'R)-spiro[tetrahydrof...)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at mineralocorticoid receptor ligand binding domain expressed in african green monkey COS7 cells co-transfected with Gal4-LBD by ...More data for this Ligand-Target Pair
TargetGlucocorticoid receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM18627((10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]...)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at glucocorticoid receptor ligand binding domain expressed in african green monkey COS7 cells co-transfected with Gal4-LBD by luc...More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50169743((13S,17S)-13-Methyl-7-[9-(4,4,5,5,5-pentafluoro-pe...)copy SMILEScopy InChI
Affinity DataIC50: 3.80nMAssay Description:Antagonist activity at estrogen receptor beta ligand binding domain expressed in african green monkey COS7 cells co-transfected with Gal4-LBD by luci...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49RQRPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50169743((13S,17S)-13-Methyl-7-[9-(4,4,5,5,5-pentafluoro-pe...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Antagonist activity at estrogen receptor alpha ligand binding domain expressed in african green monkey COS7 cells co-transfected with Gal4-LBD by luc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49RQRPubMed
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50312006(CHEMBL1076438 | Lecanindole D)copy SMILEScopy InChI
Affinity DataIC50: 5.5nMAssay Description:Displacement of progesterone from progesterone receptor in human T47D cells after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49RQRPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM35909(2-Hydroxy-2-methyl-N-(4-nitro-3-trifluoromethyl-ph...)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Antagonist activity at androgen receptor ligand binding domain expressed in african green monkey COS7 cells co-transfected with Gal4-LBD by luciferas...More data for this Ligand-Target Pair
TargetProgesterone receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50312006(CHEMBL1076438 | Lecanindole D)copy SMILEScopy InChI
Affinity DataIC50: 57.3nMAssay Description:Displacement of [3H]progesterone from progesterone receptor in human T47D cells after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49RQRPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50312006(CHEMBL1076438 | Lecanindole D)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at glucocorticoid receptor ligand binding domain expressed in african green monkey COS7 cells co-transfected with Gal4-LBD by luc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49RQRPubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50312006(CHEMBL1076438 | Lecanindole D)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at estrogen receptor beta ligand binding domain expressed in african green monkey COS7 cells co-transfected with Gal4-LBD by luci...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49RQRPubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50312005(CHEMBL1087512 | Lecanindole B)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at estrogen receptor beta ligand binding domain expressed in african green monkey COS7 cells co-transfected with Gal4-LBD by luci...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49RQRPubMed
TargetEstrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50312006(CHEMBL1076438 | Lecanindole D)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at estrogen receptor alpha ligand binding domain expressed in african green monkey COS7 cells co-transfected with Gal4-LBD by luc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49RQRPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50312005(CHEMBL1087512 | Lecanindole B)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at androgen receptor ligand binding domain expressed in african green monkey COS7 cells co-transfected with Gal4-LBD by luciferas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49RQRPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50312006(CHEMBL1076438 | Lecanindole D)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at androgen receptor ligand binding domain expressed in african green monkey COS7 cells co-transfected with Gal4-LBD by luciferas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49RQRPubMed
TargetMineralocorticoid receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50312006(CHEMBL1076438 | Lecanindole D)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+6nMAssay Description:Antagonist activity at mineralocorticoid receptor ligand binding domain expressed in african green monkey COS7 cells co-transfected with Gal4-LBD by ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49RQRPubMed
TargetMineralocorticoid receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50312005(CHEMBL1087512 | Lecanindole B)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+7nMAssay Description:Antagonist activity at mineralocorticoid receptor ligand binding domain expressed in african green monkey COS7 cells co-transfected with Gal4-LBD by ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49RQRPubMed
TargetAndrogen receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM18161((1S,2S,7S,10R,11S,14S,15S)-14-hydroxy-2,15-dimethy...)copy SMILEScopy InChI
Affinity DataEC50:  20nMAssay Description:Agonist activity at androgen receptor ligand binding domain expressed in african green monkey COS7 cells co-transfected with Gal4-DBD by luciferase r...More data for this Ligand-Target Pair
TargetGlucocorticoid receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM18207((1R,2S,10S,11S,13R,14R,15S,17S)-1-fluoro-14,17-dih...)copy SMILEScopy InChI
Affinity DataEC50:  7.20nMAssay Description:Agonist activity at glucocorticoid receptor ligand binding domain expressed in african green monkey COS7 cells co-transfected with Gal4-LBD by lucife...More data for this Ligand-Target Pair
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