Compile Data Set for Download or QSAR
Found 69 with Last Name = 'weaver' and Initial = 'dr'
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM29611(2-Iodomelatonin | CHEMBL289233 | Melatonin,2-Iodo)copy SMILEScopy InChI
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8WXKPubMed
TargetMelatonin receptor type 1A(Sheep)
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM29611(2-Iodomelatonin | CHEMBL289233 | Melatonin,2-Iodo)copy SMILEScopy InChI
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8WXKPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM29611(2-Iodomelatonin | CHEMBL289233 | Melatonin,2-Iodo)copy SMILEScopy InChI
Affinity DataKi:  0.0900nMMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM29611(2-Iodomelatonin | CHEMBL289233 | Melatonin,2-Iodo)copy SMILEScopy InChI
Affinity DataKi:  0.170nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9GGMPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50034110(CHEMBL15060 | Melatonin,2-Phenyl | N-[2-(5-Methoxy...)copy SMILEScopy InChI
Affinity DataKi:  0.210nMMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50035179(Agomelatine | CHEMBL10878 | N-[2-(7-Methoxy-naphth...)copy SMILEScopy InChI
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9GGMPubMedDrugBank
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)copy SMILEScopy InChI
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8WXKPubMedDrugBank
TargetMelatonin receptor type 1A(Sheep)
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)copy SMILEScopy InChI
Affinity DataKi:  0.240nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8WXKPubMed
TargetMelatonin receptor type 1A(Sheep)
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50043289(CHEMBL34730 | N-[2-(6-Chloro-5-methoxy-1H-indol-3-...)copy SMILEScopy InChI
Affinity DataKi:  0.25nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8WXKPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50034110(CHEMBL15060 | Melatonin,2-Phenyl | N-[2-(5-Methoxy...)copy SMILEScopy InChI
Affinity DataKi:  0.260nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9GGMPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50043289(CHEMBL34730 | N-[2-(6-Chloro-5-methoxy-1H-indol-3-...)copy SMILEScopy InChI
Affinity DataKi:  0.660nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9GGMPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50035179(Agomelatine | CHEMBL10878 | N-[2-(7-Methoxy-naphth...)copy SMILEScopy InChI
Affinity DataKi:  0.720nMMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)copy SMILEScopy InChI
Affinity DataKi:  1.11nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9GGMPubMedDrugBank
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)copy SMILEScopy InChI
Affinity DataKi:  1.48nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9GGMPubMedDrugBank
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82509(Melatonin,6-Hydroxy | melatonin, 6-Hydroxy)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8WXKPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50043289(CHEMBL34730 | N-[2-(6-Chloro-5-methoxy-1H-indol-3-...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8WXKPubMed
TargetMelatonin receptor type 1A(Sheep)
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82509(Melatonin,6-Hydroxy | melatonin, 6-Hydroxy)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8WXKPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50043289(CHEMBL34730 | N-[2-(6-Chloro-5-methoxy-1H-indol-3-...)copy SMILEScopy InChI
Affinity DataKi:  6.78nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9GGMPubMed
TargetMelatonin receptor type 1A(Sheep)
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82271(CAS_260803 | NAS | NSC_260803)copy SMILEScopy InChI
Affinity DataKi:  140nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8WXKPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82271(CAS_260803 | NAS | NSC_260803)copy SMILEScopy InChI
Affinity DataKi:  170nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8WXKPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82271(CAS_260803 | NAS | NSC_260803)copy SMILEScopy InChI
Affinity DataKi:  595nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9GGMPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82271(CAS_260803 | NAS | NSC_260803)copy SMILEScopy InChI
Affinity DataKi:  986nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9GGMPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9GGMPubMed
TargetMelatonin receptor type 1A(Sheep)
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8WXKPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9GGMPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Massachusetts General Hospital

Curated by PDSP Ki Database
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9GGMPubMed
TargetEstrogen receptor beta(Rattus norvegicus)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Binding to Estrogen receptor- beta (ER beta) receptorMore data for this Ligand-Target Pair
TargetEstrogen receptor(RAT)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Binding to Estrogen receptor- alpha (ER alpha) receptorMore data for this Ligand-Target Pair
TargetEstrogen receptor(RAT)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM19441(2-(4-hydroxyphenyl)-3-({4-[2-(piperidin-1-yl)ethox...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Binding to Estrogen receptor- alpha (ER alpha) receptorMore data for this Ligand-Target Pair
TargetEstrogen receptor(RAT)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50118989((2-Chloro-phenyl)-(6-hydroxy-3-naphthalen-1-yl-ben...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Binding to Estrogen receptor- alpha (ER alpha) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F18Z2HPubMed
TargetEstrogen receptor beta(Rattus norvegicus)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50118989((2-Chloro-phenyl)-(6-hydroxy-3-naphthalen-1-yl-ben...)copy SMILEScopy InChI
Affinity DataIC50: 63nMAssay Description:Binding to Estrogen receptor- beta (ER beta) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F18Z2HPubMed
TargetEstrogen receptor(RAT)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50118987((2,4-Dimethyl-phenyl)-(6-hydroxy-3-naphthalen-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 75nMAssay Description:Binding to Estrogen receptor- alpha (ER alpha) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F18Z2HPubMed
TargetEstrogen receptor beta(Rattus norvegicus)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50118993((6-Hydroxy-3-naphthalen-1-yl-benzofuran-2-yl)-(4-h...)copy SMILEScopy InChI
Affinity DataIC50: 79nMAssay Description:Binding to Estrogen receptor- beta (ER beta) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F18Z2HPubMed
TargetEstrogen receptor(RAT)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50119003(Biphenyl-4-yl-(6-hydroxy-3-naphthalen-1-yl-benzofu...)copy SMILEScopy InChI
Affinity DataIC50: 99nMAssay Description:Binding to Estrogen receptor- alpha (ER alpha) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F18Z2HPubMed
TargetEstrogen receptor beta(Rattus norvegicus)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50118999((6-Hydroxy-3-naphthalen-1-yl-benzofuran-2-yl)-phen...)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Binding to Estrogen receptor- beta (ER beta) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F18Z2HPubMed
TargetEstrogen receptor(RAT)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50119000((2,3-Dihydro-benzo[1,4]dioxin-6-yl)-(6-hydroxy-3-n...)copy SMILEScopy InChI
Affinity DataIC50: 140nMAssay Description:Binding to Estrogen receptor- alpha (ER alpha) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F18Z2HPubMed
TargetEstrogen receptor(RAT)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50118999((6-Hydroxy-3-naphthalen-1-yl-benzofuran-2-yl)-phen...)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Binding to Estrogen receptor- alpha (ER alpha) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F18Z2HPubMed
TargetEstrogen receptor(RAT)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50118993((6-Hydroxy-3-naphthalen-1-yl-benzofuran-2-yl)-(4-h...)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Binding to Estrogen receptor- alpha (ER alpha) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F18Z2HPubMed
TargetEstrogen receptor(RAT)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50119006((3,4-Dihydro-2H-benzo[b][1,4]dioxepin-7-yl)-(6-hyd...)copy SMILEScopy InChI
Affinity DataIC50: 190nMAssay Description:Binding affinity for Estrogen receptor alpha (ER alpha) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F18Z2HPubMed
TargetEstrogen receptor(RAT)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50119004((3-Fluoro-phenyl)-(6-hydroxy-3-naphthalen-1-yl-ben...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Binding to Estrogen receptor- alpha (ER alpha) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F18Z2HPubMed
TargetEstrogen receptor(RAT)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50118998((3-Bromo-phenyl)-(6-hydroxy-3-naphthalen-1-yl-benz...)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Binding to Estrogen receptor- alpha (ER alpha) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F18Z2HPubMed
TargetEstrogen receptor beta(Rattus norvegicus)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50118987((2,4-Dimethyl-phenyl)-(6-hydroxy-3-naphthalen-1-yl...)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Binding to Estrogen receptor- beta (ER beta) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F18Z2HPubMed
TargetEstrogen receptor(RAT)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50118997((4-Difluoromethoxy-phenyl)-(6-hydroxy-3-naphthalen...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Binding to Estrogen receptor- alpha (ER alpha) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F18Z2HPubMed
TargetEstrogen receptor beta(Rattus norvegicus)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50119002((4-Fluoro-phenyl)-(6-hydroxy-3-naphthalen-1-yl-ben...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Binding to Estrogen receptor- beta (ER beta) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F18Z2HPubMed
TargetEstrogen receptor beta(Rattus norvegicus)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50119004((3-Fluoro-phenyl)-(6-hydroxy-3-naphthalen-1-yl-ben...)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:Binding to Estrogen receptor- beta (ER beta) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F18Z2HPubMed
TargetEstrogen receptor(RAT)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50119002((4-Fluoro-phenyl)-(6-hydroxy-3-naphthalen-1-yl-ben...)copy SMILEScopy InChI
Affinity DataIC50: 360nMAssay Description:Binding to Estrogen receptor- alpha (ER alpha) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F18Z2HPubMed
TargetEstrogen receptor(RAT)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50118990((4-Bromo-phenyl)-(6-hydroxy-3-naphthalen-1-yl-benz...)copy SMILEScopy InChI
Affinity DataIC50: 380nMAssay Description:Binding to Estrogen receptor- alpha (ER alpha) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F18Z2HPubMed
TargetEstrogen receptor(RAT)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50118992((2-Chloro-phenyl)-[6-hydroxy-3-(2-methoxy-benzyl)-...)copy SMILEScopy InChI
Affinity DataIC50: 380nMAssay Description:Binding to Estrogen receptor- alpha (ER alpha) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F18Z2HPubMed
TargetEstrogen receptor(RAT)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50119001((2,4-Dimethyl-phenyl)-[6-hydroxy-3-(2-methoxy-benz...)copy SMILEScopy InChI
Affinity DataIC50: 380nMAssay Description:Binding to Estrogen receptor- alpha (ER alpha) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F18Z2HPubMed
TargetEstrogen receptor(RAT)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50118988((2-Chloro-phenyl)-(6-hydroxy-3-phenyl-benzofuran-2...)copy SMILEScopy InChI
Affinity DataIC50: 390nMAssay Description:Binding to Estrogen receptor- alpha (ER alpha) receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F18Z2HPubMed
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