Compile Data Set for Download or QSAR
Found 121 with Last Name = 'cohen' and Initial = 'ds'
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003780(4-(3-Pyridin-3-yl-propyl)-8-(toluene-4-sulfonylami...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F47N3WPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003784(8-(4-Chloro-benzenesulfonylamino)-4-[3-(4-methyl-p...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F47N3WPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003792(8-(4-Fluoro-benzenesulfonylamino)-4-(3-pyridin-3-y...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F47N3WPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003803(8-(Naphthalene-2-sulfonylamino)-4-(3-pyridin-3-yl-...)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F47N3WPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003776(8-(4-Chloro-benzenesulfonylamino)-4-(3-pyridin-3-y...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:In vitro inhibition of the compound against thromboxane synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53KS7
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003776(8-(4-Chloro-benzenesulfonylamino)-4-(3-pyridin-3-y...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:The compound was tested in vitro for its inhibitory activity against thromboxane synthase A2 (TXA2)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JW8CVBPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003776(8-(4-Chloro-benzenesulfonylamino)-4-(3-pyridin-3-y...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:In vitro inhibition of thromboxane synthasase in microsomal platelet preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XS5TFKPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003781(CHEMBL341686 | [5-(4-Chloro-benzenesulfonylamino)-...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F47N3WPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003801(4-(3-Pyridin-3-yl-propyl)-8-(4-trifluoromethyl-ben...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F47N3WPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003776(8-(4-Chloro-benzenesulfonylamino)-4-(3-pyridin-3-y...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:In vitro inhibition of thromboxane synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GX4BG6
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003797(8-(4-Chloro-benzenesulfonylamino)-4-[2-(pyridin-3-...)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:In vitro inhibition of thromboxane synthasase in microsomal platelet preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XS5TFKPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003798(8-(4-Chloro-benzenesulfonylamino)-4-(3-imidazol-1-...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F47N3WPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003800(8-(4-Methoxy-benzenesulfonylamino)-4-(3-pyridin-3-...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F47N3WPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003796(8-(4-Chloro-benzenesulfonylamino)-4-[3-(1-oxy-pyri...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F47N3WPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003795(5-[1-Pyridin-3-yl-1-(3-trifluoromethyl-phenyl)-met...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F47N3WPubMedDrugBank
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50025953(6-Imidazo[1,5-a]pyridin-5-yl-hexanoic acid | CGS-1...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of thromboxane synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GX4BG6
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003799(8-(4-Chloro-benzenesulfonylamino)-2-methyl-4-(3-py...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F47N3WPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003797(8-(4-Chloro-benzenesulfonylamino)-4-[2-(pyridin-3-...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F47N3WPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003795(5-[1-Pyridin-3-yl-1-(3-trifluoromethyl-phenyl)-met...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of the compound against thromboxane synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53KS7DrugBank
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50008790(5-[Pyridin-4-yl-(3-trifluoromethyl-phenyl)-methyle...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Compound was evaluated in vitro for the inhibition of Thromboxane synthase using [14C]-arachidonic acid as radioligandMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2BR8R47PubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50046312(8-(4-Chloro-benzenesulfonylamino)-4-[2-(pyridin-3-...)copy SMILEScopy InChI
Affinity DataIC50: 3.5nMAssay Description:In vitro inhibition of thromboxane synthasase in microsomal platelet preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XS5TFKPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003777(8-(4-Chloro-benzenesulfonylamino)-2-(5-pyridin-3-y...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:The compound was tested in vitro for its inhibitory activity against thromboxane synthase A2 (TXA2)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JW8CVBPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003789(8-(4-Methanesulfonyl-benzenesulfonylamino)-4-(3-py...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F47N3WPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003794(8-(4-Azido-benzenesulfonylamino)-4-(3-pyridin-3-yl...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F47N3WPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50283051((Z)-7-[(2S,3R,4R)-4-(Biphenyl-4-ylmethoxy)-2-pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 4.30nMAssay Description:In vitro inhibition of the compound against thromboxane synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53KS7
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50283051((Z)-7-[(2S,3R,4R)-4-(Biphenyl-4-ylmethoxy)-2-pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 4.30nMAssay Description:In vitro inhibition against thromboxane synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53KS7
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50046311(8-(4-Chloro-benzenesulfonylamino)-4-(3-pyridin-3-y...)copy SMILEScopy InChI
Affinity DataIC50: 4.5nMAssay Description:In vitro inhibition of thromboxane synthasase in microsomal platelet preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XS5TFKPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50046309(8-(4-Chloro-benzenesulfonylamino)-4-(3-pyridin-3-y...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:In vitro inhibition of thromboxane synthasase in microsomal platelet preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XS5TFKPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003787(4-Chloro-N-{8-pyridin-3-yl-5-[2-(5H-tetrazol-5-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F47N3WPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50280267(CHEMBL295121 | [3-[3-(4-Chloro-benzenesulfonylamin...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibitory concentration of the compound against thromboxane synthase enzyme from human microsomal platelet preparationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M36QQ
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003804(7-(4-Chloro-benzenesulfonylamino)-3-(3-pyridin-3-y...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F47N3WPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003790(CHEMBL136880 | Potassium; 8-(4-chloro-benzenesulfo...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F47N3WPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50008798(7-(3-Pyridin-3-yl-bicyclo[2.2.1]hept-2-yl)-heptano...)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:In vitro inhibition of thromboxane synthase using [14C]-arachidonic acidMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2BR8R47PubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50280268(3-[3-[2-(4-Chloro-benzenesulfonylamino)-ethyl]-5-(...)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibitory concentration of the compound against thromboxane synthase enzyme from human microsomal platelet preparationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M36QQ
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50283046((Z)-7-[(2S,3S,4S)-4-(Biphenyl-4-ylmethoxy)-2-pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:In vitro thromboxane receptor antagonist activity was determined by inhibition of U-46619 induced aggregation of washed human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GX4BG6
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003793(8-(4-Chloro-benzenesulfonylamino)-4-(3-pyridin-3-y...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F47N3WPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50283042((Z)-7-[(2S,3S,4R)-4-(Biphenyl-4-ylmethoxy)-2-pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:In vitro inhibition of thromboxane synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GX4BG6
TargetThromboxane A2 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283049((Z)-7-[(1R,2R,3S,5S)-5-(Biphenyl-4-ylmethoxy)-3-hy...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:In vitro thromboxane receptor antagonist activity was determined by inhibition of U-46619 induced aggregation of washed human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GX4BG6
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50283046((Z)-7-[(2S,3S,4S)-4-(Biphenyl-4-ylmethoxy)-2-pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:In vitro inhibition of thromboxane synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GX4BG6
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50046310(8-(4-Chloro-benzenesulfonylamino)-4-[2-(pyridin-3-...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:In vitro inhibition of thromboxane synthasase in microsomal platelet preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XS5TFKPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50283046((Z)-7-[(2S,3S,4S)-4-(Biphenyl-4-ylmethoxy)-2-pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:In vitro inhibition of thromboxane synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GX4BG6
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003779(8-(4-Chloro-benzenesulfonylamino)-6-pyridin-3-ylme...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:The compound was tested in vitro for its inhibitory activity against thromboxane synthase A2 (TXA2)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JW8CVBPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50280260(7-{4-[3-(4-Chloro-benzenesulfonylamino)-propyl]-py...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibitory concentration of the compound against thromboxane synthase enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC3ZF2
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50280264(3-[5-[2-(4-Chloro-benzenesulfonylamino)-ethyl]-2-(...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibitory concentration of the compound against thromboxane synthase enzyme from human microsomal platelet preparationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M36QQ
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50283051((Z)-7-[(2S,3R,4R)-4-(Biphenyl-4-ylmethoxy)-2-pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:In vitro inhibition of the compound against thromboxane synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53KS7
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003791(CHEMBL343535 | [5-(4-Chloro-benzenesulfonylamino)-...)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2F47N3WPubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50003776(8-(4-Chloro-benzenesulfonylamino)-4-(3-pyridin-3-y...)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:In vitro thromboxane receptor antagonist activity was determined by inhibition of U-46619 induced aggregation of washed human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GX4BG6
TargetThromboxane A2 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283047((Z)-7-[(2S,3S,4S)-4-(Biphenyl-4-ylmethoxy)-1,1-dio...)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:In vitro thromboxane receptor antagonist activity was determined by inhibition of U-46619 induced aggregation of washed human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GX4BG6
TargetThromboxane A2 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50003776(8-(4-Chloro-benzenesulfonylamino)-4-(3-pyridin-3-y...)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:In vitro thromboxane receptor antagonist against U-46619 induced aggregation of washed human plateletsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53KS7
TargetThromboxane-A synthase(Homo sapiens (Human))
CIBA-GEIGY Corporation

Curated by ChEMBL
LigandPNGBDBM50003773(8-(4-Chloro-benzenesulfonylamino)-5-(2-pyridin-3-y...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:The compound was tested in vitro for its inhibitory activity against thromboxane synthase A2 (TXA2)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JW8CVBPubMed
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