Compile Data Set for Download or QSAR
Found 520 with Last Name = 'lorrain' and Initial = 'ds'
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549891(CHEMBL4790083)copy SMILES
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]NMS from human recombinant muscarinic receptor M1 expressed in CHO-K1 cell membranes assessed as inhibition constant incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))TBA
LigandPNGBDBM50549891(CHEMBL4790083)copy SMILES
Affinity DataKi:  0.840nMAssay Description:Displacement of [3H]NMS from human recombinant muscarinic receptor M3 expressed in CHO-K1 cell membranes assessed as inhibition constant incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50549891(CHEMBL4790083)copy SMILES
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]NMS from human recombinant muscarinic receptor M4 expressed in CHO-K1 cell membranes assessed as inhibition constant incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549891(CHEMBL4790083)copy SMILES
Affinity DataKi:  19nMAssay Description:Displacement of [3H]NMS from human recombinant muscarinic receptor M2 expressed in CHO-K1 cell membranes assessed as inhibition constant incubated fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50296979(2-((3R)-3-(4-fluoro-N-methylphenylsulfonamido)-3,4...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Displacement of [3H]PGD2 from human prostaglandin D2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3KHBPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50335958(2-(2'-(((benzyloxycarbonyl)(ethyl)amino)methyl)-4'...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Displacement of [3H]PGD2 from human CRTh2 receptor expressed in 293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8ZNTPubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50304887((S)-3-(5-((1-acetylindolin-2-yl)methoxy)-3-(tert-b...)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Binding affinity to FLAP in human PMN derived membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2H78PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549891(CHEMBL4790083)copy SMILES
Affinity DataIC50: 1.58nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549891(CHEMBL4790083)copy SMILES
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50304898((S)-3-(5-((1-acetylindolin-2-yl)methoxy)-3-(tert-b...)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Binding affinity to FLAP in human PMN derived membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2H78PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50335954(CHEMBL1668898 | Sodium [2'-[(cyclopropanecarbonyl-...)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Antagonist activity against CRTh2 receptor in human eosinophils assessed as cell shape change after 4 hrs by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8ZNTPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50357310(CHEMBL1916710)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Displacement of [3H]-PGD2 from human prostanoid DP2 receptor expressed in human 293T cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2513ZM9PubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50322851(CHEMBL1210423 | sodium 3-(3-(tert-butylthio)-1-(4-...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Binding affinity to FLAP in human PMN by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76CRRPubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
USA.

Curated by ChEMBL
LigandPNGBDBM50335954(CHEMBL1668898 | Sodium [2'-[(cyclopropanecarbonyl-...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of human CYP3A4 by time-dependent inhibition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8ZNTPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50357308(CHEMBL1916707)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Displacement of [3H]-PGD2 from human prostanoid DP2 receptor expressed in human 293T cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2513ZM9PubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50304903((S)-3-(5-((1-acetylindolin-2-yl)methoxy)-3-(tert-b...)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Binding affinity to FLAP in human PMN derived membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2H78PubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50304899((S)-3-(5-((1-acetylindolin-2-yl)methoxy)-3-(tert-b...)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Binding affinity to FLAP in human PMN derived membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2H78PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50013729(CHEMBL3264919)copy SMILEScopy InChI
Affinity DataIC50: 2.70nMAssay Description:Antagonist activity at human PPAR-alpha assessed as inhibition of GW7647-induced effect after overnight incubation by cell-based luciferase reporter ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GX4D33PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50013730(CHEMBL3264920)copy SMILEScopy InChI
Affinity DataIC50: 2.80nMAssay Description:Antagonist activity at human PPAR-alpha assessed as inhibition of GW7647-induced effect after overnight incubation by cell-based luciferase reporter ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GX4D33PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50335957(2-(2'-(((benzyloxycarbonyl)(ethyl)amino)methyl)-4'...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]PGD2 from human CRTh2 receptor expressed in 293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8ZNTPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50013734(CHEMBL3264924)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Antagonist activity at human PPAR-alpha assessed as inhibition of GW7647-induced effect after overnight incubation by cell-based luciferase reporter ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GX4D33PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50357307(CHEMBL1916706)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]-PGD2 from human prostanoid DP2 receptor expressed in human 293T cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2513ZM9PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50357311(CHEMBL1916711)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]-PGD2 from human prostanoid DP2 receptor expressed in human 293T cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2513ZM9PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50357289(CHEMBL1916708)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]-PGD2 from human prostanoid DP2 receptor expressed in human 293T cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2513ZM9PubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50304902((S)-3-(5-((1-acetylindolin-2-yl)methoxy)-3-(tert-b...)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Binding affinity to FLAP in human PMN derived membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2H78PubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50304901((S)-3-(5-((1-acetylindolin-2-yl)methoxy)-3-(tert-b...)copy SMILEScopy InChI
Affinity DataIC50: 3.80nMAssay Description:Binding affinity to FLAP in human PMN derived membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2H78PubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50304882((S)-3-(3-(tert-butylthio)-1-(4-chlorobenzyl)-5-((1...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Binding affinity to FLAP in human PMN derived membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2H78PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50296979(2-((3R)-3-(4-fluoro-N-methylphenylsulfonamido)-3,4...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]PGD2 from human prostaglandin D2 receptor in presence of human serum albuminMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3KHBPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50335951(2-(2'-((N-ethylcyclopropanecarboxamido)methyl)-6-m...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Antagonist activity against CRTh2 receptor in human eosinophils assessed as cell shape change by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8ZNTPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50357304(CHEMBL1916702)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]-PGD2 from human prostanoid DP2 receptor expressed in human 293T cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2513ZM9PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50357303(CHEMBL1916701)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]-PGD2 from human prostanoid DP2 receptor expressed in human 293T cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2513ZM9PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50357310(CHEMBL1916710)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of human prostanoid DP2 receptor in human whole bood assessed as eosinophil shape change preincubated for 15 mins before addition of PGD2 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2513ZM9PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50357309(CHEMBL1916709)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]-PGD2 from human prostanoid DP2 receptor expressed in human 293T cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2513ZM9PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50357302(CHEMBL1916699)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]-PGD2 from human prostanoid DP2 receptor expressed in human 293T cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2513ZM9PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50357286(CHEMBL1916700)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]-PGD2 from human prostanoid DP2 receptor expressed in human 293T cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2513ZM9PubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50304897((S)-3-(5-((1-acetylindolin-2-yl)methoxy)-3-(tert-b...)copy SMILEScopy InChI
Affinity DataIC50: 4.5nMAssay Description:Binding affinity to FLAP in human PMN derived membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2H78PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Inception Sciences

Curated by ChEMBL
LigandPNGBDBM50013735(CHEMBL3264925)copy SMILEScopy InChI
Affinity DataIC50: 4.60nMAssay Description:Antagonist activity at human PPAR-alpha assessed as inhibition of GW7647-induced effect after overnight incubation by cell-based luciferase reporter ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GX4D33PubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50304895((S)-3-(5-((1-acetylindolin-2-yl)methoxy)-1-(4-chlo...)copy SMILEScopy InChI
Affinity DataIC50: 4.70nMAssay Description:Binding affinity to FLAP in human PMN derived membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2H78PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50357311(CHEMBL1916711)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of human prostanoid DP2 receptor in human whole bood assessed as eosinophil shape change preincubated for 15 mins before addition of PGD2 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2513ZM9PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50335959(2-(2'-(((benzyloxycarbonyl)(ethyl)amino)methyl)-6-...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]PGD2 from human CRTh2 receptor expressed in 293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8ZNTPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50335954(CHEMBL1668898 | Sodium [2'-[(cyclopropanecarbonyl-...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Antagonist activity against CRTh2 receptor in human eosinophils assessed as cell shape change by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8ZNTPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50357286(CHEMBL1916700)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of human prostanoid DP2 receptor in human whole bood assessed as eosinophil shape change preincubated for 15 mins before addition of PGD2 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2513ZM9PubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))TBA
LigandPNGBDBM50366775(BENZTROPINE | Benzatropine)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M4 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549901(CHEMBL4799006)copy SMILES
Affinity DataIC50: 5.80nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50549908(CHEMBL4760610)copy SMILES
Affinity DataIC50: 5.80nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M1 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445R41PubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50304907((S)-3-(5-((1-acetylpyrrolidin-2-yl)methoxy)-3-(ter...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Binding affinity to FLAP in human PMN derived membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2H78PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50357289(CHEMBL1916708)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of human prostanoid DP2 receptor in human whole bood assessed as eosinophil shape change preincubated for 15 mins before addition of PGD2 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2513ZM9PubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50335954(CHEMBL1668898 | Sodium [2'-[(cyclopropanecarbonyl-...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Displacement of [3H]PGD2 from human CRTh2 receptor expressed in 293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P8ZNTPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50296980((R)-2-(7-(4-fluoro-N-methylphenylsulfonamido)-6,7,...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Displacement of [3H]PGD2 from human prostaglandin D2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3KHBPubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50296977(2-(5-fluoro-2-methyl-3-(quinolin-2-ylmethyl)-1H-in...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Displacement of [3H]PGD2 from human prostaglandin D2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3KHBPubMed
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