Compile Data Set for Download or QSAR
Found 201 with Last Name = 'darout' and Initial = 'e'
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424575(CHEMBL2312159)copy SMILEScopy InChI
Affinity DataKi:  7nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Daegu University

Curated by ChEMBL
LigandPNGBDBM50327038((3aR,5R,6S,7R,7aR)-5-(hydroxymethyl)-2-methyl-5,6,...)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Inhibition of human O-GlcNAcase after 5 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8S2RPubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424576(CHEMBL2312158)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424564(CHEMBL2312506)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424577(CHEMBL2312157)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424579(CHEMBL2312156)copy SMILEScopy InChI
Affinity DataKi:  21nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50341309(CHEMBL1766081 | isopropyl 4-(5-methyl-6-(2-methylp...)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Displacement of [3H]isopropyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yloxy)piperidine-1-carboxylate/tert-butyl 4-(1-(4-(methyl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ37G0PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50341310(CHEMBL1766082 | Isopropyl 9-anti-({5-Methyl-6-[(2-...)copy SMILEScopy InChI
Affinity DataKi:  33nMAssay Description:Displacement of [3H]isopropyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yloxy)piperidine-1-carboxylate/tert-butyl 4-(1-(4-(methyl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ37G0PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424573(CHEMBL2312161)copy SMILEScopy InChI
Affinity DataKi:  33nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50341310(CHEMBL1766082 | Isopropyl 9-anti-({5-Methyl-6-[(2-...)copy SMILEScopy InChI
Affinity DataKi:  33nMAssay Description:Displacement of [3H]isopropyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yloxy)piperidine-1-carboxylate/tert-butyl 4-(1-(4-(methyl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ37G0PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424548(CHEMBL2312517)copy SMILEScopy InChI
Affinity DataKi:  41nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424580(CHEMBL2312516)copy SMILEScopy InChI
Affinity DataKi:  48nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50364541(CHEMBL1951011)copy SMILEScopy InChI
Affinity DataKi:  53nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424581(CHEMBL2312515)copy SMILEScopy InChI
Affinity DataKi:  94nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424563(CHEMBL2312505)copy SMILEScopy InChI
Affinity DataKi:  123nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Rattus norvegicus)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50341310(CHEMBL1766082 | Isopropyl 9-anti-({5-Methyl-6-[(2-...)copy SMILEScopy InChI
Affinity DataKi:  125nMAssay Description:Displacement of [3H]isopropyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yloxy)piperidine-1-carboxylate/tert-butyl 4-(1-(4-(methyl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ37G0PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424578(CHEMBL2311545)copy SMILEScopy InChI
Affinity DataKi:  125nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Rattus norvegicus)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50341310(CHEMBL1766082 | Isopropyl 9-anti-({5-Methyl-6-[(2-...)copy SMILEScopy InChI
Affinity DataKi:  125nMAssay Description:Displacement of [3H]isopropyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yloxy)piperidine-1-carboxylate/tert-butyl 4-(1-(4-(methyl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ37G0PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424550(CHEMBL2312519)copy SMILEScopy InChI
Affinity DataKi:  131nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424583(CHEMBL2312513)copy SMILEScopy InChI
Affinity DataKi:  133nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424559(CHEMBL2312528)copy SMILEScopy InChI
Affinity DataKi:  136nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Rattus norvegicus)
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50341309(CHEMBL1766081 | isopropyl 4-(5-methyl-6-(2-methylp...)copy SMILEScopy InChI
Affinity DataKi:  140nMAssay Description:Displacement of [3H]isopropyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yloxy)piperidine-1-carboxylate/tert-butyl 4-(1-(4-(methyl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ37G0PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424549(CHEMBL2312518)copy SMILEScopy InChI
Affinity DataKi:  141nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424569(CHEMBL2312511)copy SMILEScopy InChI
Affinity DataKi:  163nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424562(CHEMBL2312504)copy SMILEScopy InChI
Affinity DataKi:  197nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424555(CHEMBL2312525)copy SMILEScopy InChI
Affinity DataKi:  231nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424552(CHEMBL2312526)copy SMILEScopy InChI
Affinity DataKi:  290nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424582(CHEMBL2312514)copy SMILEScopy InChI
Affinity DataKi:  294nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424558(CHEMBL2312524)copy SMILEScopy InChI
Affinity DataKi:  486nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424553(CHEMBL2312527)copy SMILEScopy InChI
Affinity DataKi:  493nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424571(CHEMBL2312501)copy SMILEScopy InChI
Affinity DataKi:  507nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424556(CHEMBL2312522)copy SMILEScopy InChI
Affinity DataKi:  586nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424557(CHEMBL2312523)copy SMILEScopy InChI
Affinity DataKi:  682nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Daegu University

Curated by ChEMBL
LigandPNGBDBM50327039((3aR,5R,6S,7R,7aR)-5-(Hydroxymethyl)-2-methyl-5,6,...)copy SMILEScopy InChI
Affinity DataKi:  700nMAssay Description:Inhibition of human O-GlcNAcase after 5 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8S2RPubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424566(CHEMBL2312508)copy SMILEScopy InChI
Affinity DataKi:  814nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetCollagenase 3(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50361639(CHEMBL1371684)copy SMILEScopy InChI
Affinity DataKi:  824nMAssay Description:Noncompetitive inhibition of human full length recombinant MMP13 using triple-helical fTHP-15 as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424570(CHEMBL2312512)copy SMILEScopy InChI
Affinity DataKi:  912nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424572(CHEMBL2312162)copy SMILEScopy InChI
Affinity DataKi:  948nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424574(CHEMBL2312160)copy SMILEScopy InChI
Affinity DataKi:  1.15E+3nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50341312((1R,5R,8R)-Isopropyl 8-(5-Methyl-6-(2-methylpyridi...)copy SMILEScopy InChI
Affinity DataKi:  1.18E+3nMAssay Description:Displacement of [3H]isopropyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yloxy)piperidine-1-carboxylate/tert-butyl 4-(1-(4-(methyl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ37G0PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424567(CHEMBL2312509)copy SMILEScopy InChI
Affinity DataKi:  1.50E+3nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetCollagenase 3(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM50361640(CHEMBL1515648)copy SMILEScopy InChI
Affinity DataKi:  1.53E+3nMAssay Description:Noncompetitive inhibition of human full length recombinant MMP13 using triple-helical fTHP-15 as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2VKNPubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50341311((+/-)-isopropyl 8-(5-methyl-6-(2-methylpyridin-3-y...)copy SMILEScopy InChI
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [3H]isopropyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yloxy)piperidine-1-carboxylate/tert-butyl 4-(1-(4-(methyl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ37G0PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424554(CHEMBL2312521)copy SMILEScopy InChI
Affinity DataKi:  1.97E+3nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424551(CHEMBL2312520)copy SMILEScopy InChI
Affinity DataKi:  2.23E+3nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50341313((1S,5S,8S)-Isopropyl 8-(5-Methyl-6-(2-methylpyridi...)copy SMILEScopy InChI
Affinity DataKi:  2.27E+3nMAssay Description:Displacement of [3H]isopropyl 4-(1-(4-(methylsulfonyl)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yloxy)piperidine-1-carboxylate/tert-butyl 4-(1-(4-(methyl...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ37G0PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424568(CHEMBL2312510)copy SMILEScopy InChI
Affinity DataKi:  3.12E+3nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetCollagenase 3(Homo sapiens (Human))
Scripps Florida

Curated by ChEMBL
LigandPNGBDBM40467(2-[(4-chlorobenzyl)thio]-1,5,6,7-tetrahydrocyclope...)copy SMILEScopy InChI
Affinity DataKi:  3.80E+3nMAssay Description:Noncompetitive inhibition of human full length recombinant MMP13 using triple-helical fTHP-15 as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2VKNPubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424565(CHEMBL2312507)copy SMILEScopy InChI
Affinity DataKi: >7.32E+3nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Pfizer Inc.

Curated by ChEMBL
LigandPNGBDBM50424561(CHEMBL2312503)copy SMILEScopy InChI
Affinity DataKi: >8.15E+3nMAssay Description:Binding affinity to human GPR119 in HEK293FT cell membrane by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q91PubMed
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