Compile Data Set for Download or QSAR
Found 101 with Last Name = 'imamiya' and Initial = 'e'
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115243((S)-N-[7-(5-fluoro-2-methylphenyl)-4-methyl-(7S)-5...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115239((S)-N-[7-(2,5-dichloro-3-thienyl)-4-methyl-(7S)-5,...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115271(CHEMBL556009 | N-[7-(2,5-dichloro-3-thienyl)-4-met...)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115246(CHEMBL543867 | N-[7-(2-chloro-5-fluorophenyl)-4-me...)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115248(CHEMBL552723 | N-[7-(3-chloro-2-thienyl)-4-methyl-...)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115267(CHEMBL102546 | N-[7-(2-chlorophenyl)-4-methyl-(7S)...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115268(CHEMBL554001 | N-[7-(2-chloro-3-thienyl)-4-methyl-...)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115238(CHEMBL552865 | N-[7-(2-chlorophenyl)-4-methyl-5,6,...)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115245(CHEMBL554215 | N-[4-methyl-7-(3-thienyl)-5,6,7,8-t...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50044403(2-Methoxy-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylme...)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of specific binding of [125 I ] Angiotensin-II (0.2 nM) to bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z73X8PubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115236(CHEMBL542925 | N-[7-(5-fluoro-2-methoxyphenyl)-4-m...)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115233(CHEMBL541577 | N-[7-(2-fluorophenyl)-4-methyl-5,6,...)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115270((R)-N-[7-(2,5-dichloro-3-thienyl)-4-methyl-(7R)-5,...)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115264(CHEMBL552934 | N-[3-methyl-6-(2-methylphenyl)-4,5,...)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115258(CHEMBL555535 | N-[7-(5-fluoro-2-methylphenyl)-4-me...)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50044379(2-Propylamino-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-...)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Inhibition of specific binding of [125 I ] Angiotensin-II (0.2 nM) to bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z73X8PubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115257(CHEMBL542687 | N-[7-(2,5-difluorophenyl)-4-methyl-...)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115256(CHEMBL543148 | N-[7-(2-chlorophenyl)-4-methyl-5,6,...)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50285002(2-Ethylamino-3-[2'-(5-oxo-4,5-dihydro-[1,2,4]oxadi...)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:Displacement of [125 I]-AII (0.2 nM) from bovine adrenal cortical membrane angiotensin II (AII) receptor at 10e-7 MMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M36SM
TargetType-1 angiotensin II receptor(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50044410(2-Ethyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Inhibition of specific binding of [125 I ] Angiotensin-II (0.2 nM) to bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z73X8PubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115252(CHEMBL552827 | N-[4-methyl-7-(2-thienyl)-5,6,7,8-t...)copy SMILEScopy InChI
Affinity DataIC50: 47nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115260(CHEMBL545732 | N-[7-(3,5-dichloro-2-thienyl)-4-met...)copy SMILEScopy InChI
Affinity DataIC50: 49nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115234(CHEMBL105412 | N-[7-(2-chlorophenyl)-4-methoxy-5,6...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115241(CHEMBL541918 | N-[6-(2-chlorophenyl)-3-methyl-4,5,...)copy SMILEScopy InChI
Affinity DataIC50: 55nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115259(CHEMBL554422 | N-[7-(2-bromophenyl)-4-methyl-5,6,7...)copy SMILEScopy InChI
Affinity DataIC50: 56nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115228(CHEMBL552540 | N-[4-methyl-7-(2-methylphenyl)-5,6,...)copy SMILEScopy InChI
Affinity DataIC50: 57nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115255(CHEMBL540813 | N-[7-(2,5-dichlorophenyl)-4-methyl-...)copy SMILEScopy InChI
Affinity DataIC50: 58nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115229(CHEMBL553754 | N-[7-(3-chlorophenyl)-4-methyl-5,6,...)copy SMILEScopy InChI
Affinity DataIC50: 61nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50044414(2-Ethylamino-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 62nMAssay Description:Inhibition of specific binding of [125 I ] Angiotensin-II (0.2 nM) to bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z73X8PubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50044396(2-Ethoxy-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)copy SMILEScopy InChI
Affinity DataIC50: 66nMAssay Description:Inhibition of specific binding of [125 I ] Angiotensin-II (0.2 nM) to bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z73X8PubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50058759(CHEMBL436559 | CHEMBL462831 | Cariporide | N-(4-Is...)copy SMILEScopy InChI
Affinity DataIC50: 75nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115235(CHEMBL541833 | N-[6-(2-chlorophenyl)-3-methyl-4,5,...)copy SMILEScopy InChI
Affinity DataIC50: 82nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50044386(2-Isopropyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-yl...)copy SMILEScopy InChI
Affinity DataIC50: 82nMAssay Description:Inhibition of specific binding of [125 I ] Angiotensin-II (0.2 nM) to bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z73X8PubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50044389(2-Cyclopropyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-...)copy SMILEScopy InChI
Affinity DataIC50: 84nMAssay Description:Inhibition of specific binding of [125 I ] Angiotensin-II (0.2 nM) to bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z73X8PubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115269(CHEMBL554686 | N-[7-(2,3-dichlorophenyl)-4-methyl-...)copy SMILEScopy InChI
Affinity DataIC50: 89nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115261(CHEMBL543865 | N-(4-methyl-7-phenyl-5,6,7,8-tetrah...)copy SMILEScopy InChI
Affinity DataIC50: 91nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50044388(2-Ethanesulfinyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of specific binding of [125 I ] Angiotensin-II (0.2 nM) to bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z73X8PubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115253(CHEMBL555103 | N-[7-(2-methoxyphenyl)-4-methyl-5,6...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50240609(2-Ethoxy-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibition of specific binding of [125 I ] Angiotensin-II (0.2 nM) to bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z73X8PubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50240609(2-Ethoxy-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Displacement of [125 I]-AII (0.2 nM) from bovine adrenal cortical membrane angiotensin II (AII) receptor at 10e-7 MMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M36SM
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115242(CHEMBL554125 | N-[7-(2-furyl)-4-methyl-5,6,7,8-tet...)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50044413(2-Propylsulfanyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of specific binding of [125 I ] Angiotensin-II (0.2 nM) to bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z73X8PubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50044377(2-Methylsulfanyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of specific binding of [125 I ] Angiotensin-II (0.2 nM) to bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z73X8PubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50009714(CHEMBL191 | {2-Butyl-5-chloro-3-[2'-(2H-tetrazol-5...)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Displacement of [125 I]-AII (0.2 nM) from bovine adrenal cortical membrane angiotensin II (AII) receptor at 10e-7 MMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26M36SM
TargetType-1 angiotensin II receptor(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50044406(2-Methylsulfanylmethyl-3-[2'-(1H-tetrazol-5-yl)-bi...)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Inhibition of specific binding of [125 I ] Angiotensin-II (0.2 nM) to bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z73X8PubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50406795(Cozaar | LOSARTAN POTASSIUM)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Inhibition of specific binding of [125 I ] Angiotensin-II (0.2 nM) to bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z73X8PubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50044408(2-Methylamino-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-...)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Inhibition of specific binding of [125 I ] Angiotensin-II (0.2 nM) to bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z73X8PubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50044375(2-Propyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Inhibition of specific binding of [125 I ] Angiotensin-II (0.2 nM) to bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z73X8PubMed
TargetType-1 angiotensin II receptor(Bos taurus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50044382(2-Ethylsulfanyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-...)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Inhibition of specific binding of [125 I ] Angiotensin-II (0.2 nM) to bovine adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20Z73X8PubMed
TargetSodium/hydrogen exchanger 1(Rattus norvegicus)
Takeda Chemical Industries, Ltd.

Curated by ChEMBL
LigandPNGBDBM50115249(CHEMBL545502 | N-(2,4-dimethyl-7-phenyl-5,6,7,8-te...)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:In vitro inhibition of acid induced swelling in rat platelets by 50% as a measure of NHE-1 inhibitionMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V40VZNPubMed
Displayed 1 to 50 (of 101 total ) | Next | Last >>
Jump to: