TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Frederick National Laboratory for Cancer Research
Curated by ChEMBL
Frederick National Laboratory for Cancer Research
Curated by ChEMBL
Affinity DataIC50: 6.90nMAssay Description:Inhibition of PARP-1 (unknown origin) assessed as incorporation of biotinylated poly ADP-ribose onto histone proteins by colorimetric analysis in pre...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Frederick National Laboratory for Cancer Research
Curated by ChEMBL
Frederick National Laboratory for Cancer Research
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of PARP-1 (unknown origin) assessed as incorporation of biotinylated poly ADP-ribose onto histone proteins by colorimetric analysis in pre...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Frederick National Laboratory for Cancer Research
Curated by ChEMBL
Frederick National Laboratory for Cancer Research
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of PARP-1 (unknown origin) assessed as incorporation of biotinylated poly ADP-ribose onto histone proteins by colorimetric analysis in pre...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Frederick National Laboratory for Cancer Research
Curated by ChEMBL
Frederick National Laboratory for Cancer Research
Curated by ChEMBL
Affinity DataIC50: 58nMAssay Description:Inhibition of PARP-1 (unknown origin) assessed as incorporation of biotinylated poly ADP-ribose onto histone proteins measured without activation by ...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Frederick National Laboratory for Cancer Research
Curated by ChEMBL
Frederick National Laboratory for Cancer Research
Curated by ChEMBL
Affinity DataIC50: 123nMAssay Description:Inhibition of PARP-1 (unknown origin) assessed as incorporation of biotinylated poly ADP-ribose onto histone proteins measured without activation by ...More data for this Ligand-Target Pair
TargetCell division control protein 42 homolog(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of GEF-independent nucleotide exchange activity of prenylated Cdc42 after 3 mins in presence of 4 mM Mg2+ chelator EDTAMore data for this Ligand-Target Pair
TargetCell division control protein 42 homolog(Homo sapiens (Human))
Harvard Medical School
Curated by ChEMBL
Harvard Medical School
Curated by ChEMBL
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of GEF-independent nucleotide exchange activity of prenylated Cdc42 after 3 mins in presence of 4 mM Mg2+ chelator EDTAMore data for this Ligand-Target Pair