Compile Data Set for Download or QSAR
Found 107 with Last Name = 'riegler' and Initial = 'e'
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545768(CHEMBL4641127)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545779(CHEMBL4642563)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545782(CHEMBL4637695)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545769(CHEMBL4645325)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545771(CHEMBL4639600)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545778(CHEMBL4637143)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545762(CHEMBL4647117)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545770(CHEMBL4641595)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545777(CHEMBL4634054)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545781(CHEMBL4633133)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545773(CHEMBL4633494)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545759(CHEMBL4647188)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545760(CHEMBL4636749)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545778(CHEMBL4637143)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Antagonist activity at CCR4 in human Treg cells assessed as inhibition of CCL22-mediated chemotaxis preincubated for 30 mins followed by CCL22 additi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545766(CHEMBL4645037)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545779(CHEMBL4642563)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Antagonist activity at CCR4 in human CCRF-CEM cells assessed as inhibition of CCL22-mediated chemotaxis preincubated for 30 mins followed by CCL22 ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545776(CHEMBL4641873)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Mus musculus)
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545778(CHEMBL4637143)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Antagonist activity at CCR4 in mouse Treg cells assessed as inhibition of CCL22-mediated chemotaxis preincubated for 30 mins followed by CCL22 additi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545768(CHEMBL4641127)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Antagonist activity at CCR4 in human CCRF-CEM cells assessed as inhibition of CCL22-mediated chemotaxis preincubated for 30 mins followed by CCL22 ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545767(CHEMBL4640439)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545765(CHEMBL4639418)copy SMILEScopy InChI
Affinity DataIC50: 47nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545778(CHEMBL4637143)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Antagonist activity at CCR4 in human CCRF-CEM cells assessed as inhibition of CCL22-mediated chemotaxis preincubated for 30 mins followed by CCL22 ad...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545769(CHEMBL4645325)copy SMILEScopy InChI
Affinity DataIC50: 59nMAssay Description:Antagonist activity at CCR4 in human CCRF-CEM cells assessed as inhibition of CCL22-mediated chemotaxis preincubated for 30 mins followed by CCL22 ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545778(CHEMBL4637143)copy SMILEScopy InChI
Affinity DataIC50: 64nMAssay Description:Antagonist activity at CCR4 in human CCRF-CEM cells assessed as inhibition of CCL17-mediated chemotaxis preincubated for 30 mins followed by CCL17 ad...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545763(CHEMBL4638846)copy SMILEScopy InChI
Affinity DataIC50: 69nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545777(CHEMBL4634054)copy SMILEScopy InChI
Affinity DataIC50: 74nMAssay Description:Antagonist activity at CCR4 in human CCRF-CEM cells assessed as inhibition of CCL22-mediated chemotaxis preincubated for 30 mins followed by CCL22 ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545761(CHEMBL4633920)copy SMILEScopy InChI
Affinity DataIC50: 77nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545758(CHEMBL4643609)copy SMILEScopy InChI
Affinity DataIC50: 84nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545764(CHEMBL4643158)copy SMILEScopy InChI
Affinity DataIC50: 91nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545771(CHEMBL4639600)copy SMILEScopy InChI
Affinity DataIC50: 97nMAssay Description:Antagonist activity at CCR4 in human CCRF-CEM cells assessed as inhibition of CCL22-mediated chemotaxis preincubated for 30 mins followed by CCL22 ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545776(CHEMBL4641873)copy SMILEScopy InChI
Affinity DataIC50: 109nMAssay Description:Antagonist activity at CCR4 in human CCRF-CEM cells assessed as inhibition of CCL22-mediated chemotaxis preincubated for 30 mins followed by CCL22 ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545760(CHEMBL4636749)copy SMILEScopy InChI
Affinity DataIC50: 115nMAssay Description:Antagonist activity at CCR4 in human CCRF-CEM cells assessed as inhibition of CCL22-mediated chemotaxis preincubated for 30 mins followed by CCL22 ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545783(CHEMBL4649666)copy SMILEScopy InChI
Affinity DataIC50: 121nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545770(CHEMBL4641595)copy SMILEScopy InChI
Affinity DataIC50: 133nMAssay Description:Antagonist activity at CCR4 in human CCRF-CEM cells assessed as inhibition of CCL22-mediated chemotaxis preincubated for 30 mins followed by CCL22 ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545759(CHEMBL4647188)copy SMILEScopy InChI
Affinity DataIC50: 136nMAssay Description:Antagonist activity at CCR4 in human CCRF-CEM cells assessed as inhibition of CCL22-mediated chemotaxis preincubated for 30 mins followed by CCL22 ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545767(CHEMBL4640439)copy SMILEScopy InChI
Affinity DataIC50: 247nMAssay Description:Antagonist activity at CCR4 in human CCRF-CEM cells assessed as inhibition of CCL22-mediated chemotaxis preincubated for 30 mins followed by CCL22 ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545762(CHEMBL4647117)copy SMILEScopy InChI
Affinity DataIC50: 259nMAssay Description:Antagonist activity at CCR4 in human CCRF-CEM cells assessed as inhibition of CCL22-mediated chemotaxis preincubated for 30 mins followed by CCL22 ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545764(CHEMBL4643158)copy SMILEScopy InChI
Affinity DataIC50: 370nMAssay Description:Antagonist activity at CCR4 in human CCRF-CEM cells assessed as inhibition of CCL22-mediated chemotaxis preincubated for 30 mins followed by CCL22 ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545775(CHEMBL4640909)copy SMILEScopy InChI
Affinity DataIC50: 370nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545782(CHEMBL4637695)copy SMILEScopy InChI
Affinity DataIC50: 379nMAssay Description:Antagonist activity at CCR4 in human CCRF-CEM cells assessed as inhibition of CCL22-mediated chemotaxis preincubated for 30 mins followed by CCL22 ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545765(CHEMBL4639418)copy SMILEScopy InChI
Affinity DataIC50: 409nMAssay Description:Antagonist activity at CCR4 in human CCRF-CEM cells assessed as inhibition of CCL22-mediated chemotaxis preincubated for 30 mins followed by CCL22 ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545781(CHEMBL4633133)copy SMILEScopy InChI
Affinity DataIC50: 446nMAssay Description:Antagonist activity at CCR4 in human CCRF-CEM cells assessed as inhibition of CCL22-mediated chemotaxis preincubated for 30 mins followed by CCL22 ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545784(CHEMBL4642090)copy SMILEScopy InChI
Affinity DataIC50: 455nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545774(CHEMBL4644412)copy SMILEScopy InChI
Affinity DataIC50: 505nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545773(CHEMBL4633494)copy SMILEScopy InChI
Affinity DataIC50: 523nMAssay Description:Antagonist activity at CCR4 in human CCRF-CEM cells assessed as inhibition of CCL22-mediated chemotaxis preincubated for 30 mins followed by CCL22 ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545763(CHEMBL4638846)copy SMILEScopy InChI
Affinity DataIC50: 559nMAssay Description:Antagonist activity at CCR4 in human CCRF-CEM cells assessed as inhibition of CCL22-mediated chemotaxis preincubated for 30 mins followed by CCL22 ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545761(CHEMBL4633920)copy SMILEScopy InChI
Affinity DataIC50: 575nMAssay Description:Antagonist activity at CCR4 in human CCRF-CEM cells assessed as inhibition of CCL22-mediated chemotaxis preincubated for 30 mins followed by CCL22 ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545756(CHEMBL4643066)copy SMILEScopy InChI
Affinity DataIC50: 596nMAssay Description:Antagonist activity at human CCR4 expressed in rat chem-5 cells assessed as inhibition of CCL22-induced calcium flux measured at 2.5 secs time interv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545758(CHEMBL4643609)copy SMILEScopy InChI
Affinity DataIC50: 717nMAssay Description:Antagonist activity at CCR4 in human CCRF-CEM cells assessed as inhibition of CCL22-mediated chemotaxis preincubated for 30 mins followed by CCL22 ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
RAPT Therapeutics

Curated by ChEMBL
LigandPNGBDBM50545766(CHEMBL4645037)copy SMILEScopy InChI
Affinity DataIC50: 775nMAssay Description:Antagonist activity at CCR4 in human CCRF-CEM cells assessed as inhibition of CCL22-mediated chemotaxis preincubated for 30 mins followed by CCL22 ad...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ0CW6PubMed
Displayed 1 to 50 (of 107 total ) | Next | Last >>
Jump to: