Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Vanderbilt University
Curated by PDSP Ki Database
Vanderbilt University
Curated by PDSP Ki Database
Affinity DataKi: 0.320nMAssay Description:Binding affinity was measured against 5-hydroxytryptamine 1A receptor by displacement of [3H]-8-OH-DPAT by lysergic acid amidesMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity was measured against 5-hydroxytryptamine 1A receptor by displacement of [3H]-8-OH-DPAT by lysergic acid amidesMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Vanderbilt University
Curated by PDSP Ki Database
Vanderbilt University
Curated by PDSP Ki Database
Affinity DataKi: 2nMAssay Description:Binding affinity was measured against 5-hydroxytryptamine 1A receptor by displacement of [3H]-8-OH-DPAT by lysergic acid amidesMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Vanderbilt University
Curated by PDSP Ki Database
Vanderbilt University
Curated by PDSP Ki Database
Affinity DataKi: 2.10nMAssay Description:Binding affinity was measured against 5-hydroxytryptamine 1A receptor by displacement of [3H]-8-OH-DPAT by lysergic acid amidesMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Binding affinity was measured against 5-hydroxytryptamine 1A receptor by displacement of [3H]-8-OH-DPAT by lysergic acid amidesMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Binding affinity was measured against 5-hydroxytryptamine 2A receptor by displacement of [3H]- ketanserin by lysergic acid amidesMore data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Binding affinity was measured against 5-hydroxytryptamine 2A receptor by displacement of [3H]- ketanserin by lysergic acid amidesMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Binding affinity was measured against 5-hydroxytryptamine 1A receptor by displacement of [3H]-8-OH-DPAT by lysergic acid amidesMore data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:Binding affinity was measured against 5-hydroxytryptamine 1A receptor by displacement of [3H]-8-OH-DPAT by lysergic acid amidesMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Binding affinity was measured against 5-hydroxytryptamine 1A receptor by displacement of [3H]-8-OH-DPAT by lysergic acid amidesMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity was measured against 5-hydroxytryptamine 2A receptor by displacement of [3H]- ketanserin by lysergic acid amidesMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity was measured against 5-hydroxytryptamine 1A receptor by displacement of [3H]-8-OH-DPAT by lysergic acid amidesMore data for this Ligand-Target Pair
Affinity DataKi: 8.80nMAssay Description:Binding affinity was measured against 5-hydroxytryptamine 2A receptor by displacement of [3H]- ketanserin by lysergic acid amidesMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity was measured against 5-hydroxytryptamine 1A receptor by displacement of [3H]-8-OH-DPAT by lysergic acid amidesMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding affinity was measured against 5-hydroxytryptamine 2A receptor by displacement of [3H]- ketanserin by lysergic acid amidesMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Vanderbilt University
Curated by PDSP Ki Database
Vanderbilt University
Curated by PDSP Ki Database
Affinity DataKi: 34nMAssay Description:Binding affinity was measured against 5-hydroxytryptamine 2A receptor by displacement of [3H]- ketanserin by lysergic acid amidesMore data for this Ligand-Target Pair
Affinity DataKi: 55nMAssay Description:Binding affinity was measured against 5-hydroxytryptamine 2A receptor by displacement of [3H]- ketanserin by lysergic acid amidesMore data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Agonist activity at cloned human 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Binding affinity was measured against 5-hydroxytryptamine 2A receptor by displacement of [3H]- ketanserin by lysergic acid amidesMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Vanderbilt University
Curated by PDSP Ki Database
Vanderbilt University
Curated by PDSP Ki Database
Affinity DataKi: 105nMAssay Description:Binding affinity was measured against 5-hydroxytryptamine 2A receptor by displacement of [3H]- ketanserin by lysergic acid amidesMore data for this Ligand-Target Pair
Affinity DataKi: 118nMAssay Description:Agonist activity at cloned human 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 177nMAssay Description:Agonist activity at cloned human 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 205nMAssay Description:Antagonist activity at cloned human 5-hydroxytryptamine 2B receptor using [3H]- rauwolscine radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 216nMAssay Description:Agonist activity at cloned human 5-hydroxytryptamine 2A receptor using [125I]-DOI radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 302nMAssay Description:Agonist activity at cloned human 5-hydroxytryptamine 2B receptor using [3H]-5-HT radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 303nMAssay Description:Agonist activity at cloned human 5-hydroxytryptamine 2C receptor using [125I]-DOI radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 311nMAssay Description:Antagonist activity at cloned human 5-hydroxytryptamine 2B receptor using [3H]-rauwolscine radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 335nMAssay Description:Agonist activity at cloned human 5-hydroxytryptamine 2A receptor using [125I]-DOI radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 357nMAssay Description:Binding affinity was measured against 5-hydroxytryptamine 2A receptor by displacement of [3H]- ketanserin by lysergic acid amidesMore data for this Ligand-Target Pair
Affinity DataKi: 368nMAssay Description:Agonist activity at cloned human 5-hydroxytryptamine 2A receptor using [125I]-DOI radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 368nMAssay Description:Agonist activity at cloned human 5-hydroxytryptamine 2A receptor using [125I]-DOI radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 523nMAssay Description:Agonist activity at cloned human 5-hydroxytryptamine 2B receptor using [3H]-5-HT radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 551nMAssay Description:Agonist activity at cloned human 5-hydroxytryptamine 2A receptor using [125I]-DOI radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 555nMAssay Description:Agonist activity at cloned human 5-hydroxytryptamine 2B receptor using [3H]-5-HT radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 654nMAssay Description:Antagonist activity at cloned human 5-hydroxytryptamine 2C receptor using [3H]-mesulergine radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 795nMAssay Description:Agonist activity at cloned human 5-hydroxytryptamine 2B receptor using [3H]-5-HT radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.11E+3nMAssay Description:Antagonist activity at cloned human 5-hydroxytryptamine 2C receptor using [3H]-mesulergine radioligandMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Vanderbilt University
Curated by PDSP Ki Database
Vanderbilt University
Curated by PDSP Ki Database
Affinity DataKi: 2.10E+3nMAssay Description:Ability to displace [3H]-ketanserin from rat cortical homogenate 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:Ability to displace [3H]-ketanserin from rat cortical homogenate 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Vanderbilt University
Curated by PDSP Ki Database
Vanderbilt University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Vanderbilt University
Curated by PDSP Ki Database
Vanderbilt University
Curated by PDSP Ki Database
Affinity DataKi: 4.44E+3nMAssay Description:Antagonist activity at cloned human 5-hydroxytryptamine 2A receptor using [3H]-Ketanserin radioligandMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Vanderbilt University
Curated by PDSP Ki Database
Vanderbilt University
Curated by PDSP Ki Database
Affinity DataKi: 5.50E+3nMAssay Description:Ability to displace [3H]-ketanserin from rat cortical homogenate 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
![](/img/powered_by_small.gif)