Compile Data Set for Download or QSAR
Found 91 with Last Name = 'sarukhanyan' and Initial = 'e'
TargetGlycine receptor subunit alpha-1(RAT)
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Displacement of [3H]strychnine from glycine receptor alpha 1 in rat brain synaptic membranesMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(RAT)
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232884(CHEMBL4060962)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Displacement of [3H]strychnine from glycine receptor alpha 1 in rat brain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Displacement of [3H]strychnine from recombinant human glycine receptor alpha 1 expressed in HEK293 cell membranes after 30 mins by liquid scintillati...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232885(CHEMBL4089150)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Displacement of [3H]strychnine from recombinant human glycine receptor alpha 1 expressed in HEK293 cell membranes after 30 mins by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232888(CHEMBL4096857)copy SMILEScopy InChI
Affinity DataKi:  67nMAssay Description:Displacement of [3H]strychnine from recombinant human glycine receptor alpha 1 expressed in HEK293 cell membranes after 30 mins by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232890(CHEMBL4102677)copy SMILEScopy InChI
Affinity DataKi:  189nMAssay Description:Displacement of [3H]strychnine from recombinant human glycine receptor alpha 1 expressed in HEK293 cell membranes after 30 mins by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232897(CHEMBL4068867)copy SMILEScopy InChI
Affinity DataKi:  241nMAssay Description:Displacement of [3H]strychnine from recombinant human glycine receptor alpha 1 expressed in HEK293 cell membranes after 30 mins by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232896(CHEMBL4079657)copy SMILEScopy InChI
Affinity DataKi:  370nMAssay Description:Displacement of [3H]strychnine from recombinant human glycine receptor alpha 1 expressed in HEK293 cell membranes after 30 mins by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232889(CHEMBL4103909)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in HEK293 cells assessed as inhibition of glycine-induced current at...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232896(CHEMBL4079657)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in HEK293 cells assessed as inhibition of glycine-induced current at...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232896(CHEMBL4079657)copy SMILEScopy InChI
Affinity DataIC50: 49nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232889(CHEMBL4103909)copy SMILEScopy InChI
Affinity DataIC50: 51nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)copy SMILEScopy InChI
Affinity DataIC50: 51nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232889(CHEMBL4103909)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232890(CHEMBL4102677)copy SMILEScopy InChI
Affinity DataIC50: 56nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in HEK293 cells assessed as inhibition of glycine-induced current at...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)copy SMILEScopy InChI
Affinity DataIC50: 58nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in HEK293 cells assessed as inhibition of glycine-induced current at...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232889(CHEMBL4103909)copy SMILEScopy InChI
Affinity DataIC50: 59nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232890(CHEMBL4102677)copy SMILEScopy InChI
Affinity DataIC50: 75nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232884(CHEMBL4060962)copy SMILEScopy InChI
Affinity DataIC50: 76nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232884(CHEMBL4060962)copy SMILEScopy InChI
Affinity DataIC50: 77nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232884(CHEMBL4060962)copy SMILEScopy InChI
Affinity DataIC50: 78nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232885(CHEMBL4089150)copy SMILEScopy InChI
Affinity DataIC50: 80nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in HEK293 cells assessed as inhibition of glycine-induced current at...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232885(CHEMBL4089150)copy SMILEScopy InChI
Affinity DataIC50: 82nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)copy SMILEScopy InChI
Affinity DataIC50: 93nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232896(CHEMBL4079657)copy SMILEScopy InChI
Affinity DataIC50: 95nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232885(CHEMBL4089150)copy SMILEScopy InChI
Affinity DataIC50: 97nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232884(CHEMBL4060962)copy SMILEScopy InChI
Affinity DataIC50: 97nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in HEK293 cells assessed as inhibition of glycine-induced current at...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232885(CHEMBL4089150)copy SMILEScopy InChI
Affinity DataIC50: 98nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232890(CHEMBL4102677)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232890(CHEMBL4102677)copy SMILEScopy InChI
Affinity DataIC50: 105nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232897(CHEMBL4068867)copy SMILEScopy InChI
Affinity DataIC50: 109nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232897(CHEMBL4068867)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232897(CHEMBL4068867)copy SMILEScopy InChI
Affinity DataIC50: 115nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232897(CHEMBL4068867)copy SMILEScopy InChI
Affinity DataIC50: 116nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in HEK293 cells assessed as inhibition of glycine-induced current at...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232896(CHEMBL4079657)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in human tsA201 cells assessed as inhibition of glycine-induced rece...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232896(CHEMBL4079657)copy SMILEScopy InChI
Affinity DataIC50: 158nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in human tsA201 cells assessed as inhibition of glycine-induced rece...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232891(CHEMBL4086212)copy SMILEScopy InChI
Affinity DataIC50: 166nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232891(CHEMBL4086212)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in human tsA201 cells assessed as inhibition of glycine-induced rece...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)copy SMILEScopy InChI
Affinity DataIC50: 182nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in human tsA201 cells assessed as inhibition of glycine-induced rece...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232888(CHEMBL4096857)copy SMILEScopy InChI
Affinity DataIC50: 201nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232885(CHEMBL4089150)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in human tsA201 cells assessed as inhibition of glycine-induced rece...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232890(CHEMBL4102677)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in human tsA201 cells assessed as inhibition of glycine-induced rece...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232890(CHEMBL4102677)copy SMILEScopy InChI
Affinity DataIC50: 214nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in human tsA201 cells assessed as inhibition of glycine-induced rece...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232885(CHEMBL4089150)copy SMILEScopy InChI
Affinity DataIC50: 214nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in human tsA201 cells assessed as inhibition of glycine-induced rece...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232887(CHEMBL4096505)copy SMILEScopy InChI
Affinity DataIC50: 220nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232887(CHEMBL4096505)copy SMILEScopy InChI
Affinity DataIC50: 224nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232889(CHEMBL4103909)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in human tsA201 cells assessed as inhibition of glycine-induced rece...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232895(CHEMBL4087535)copy SMILEScopy InChI
Affinity DataIC50: 245nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232895(CHEMBL4087535)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
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