Compile Data Set for Download or QSAR
Found 69 with Last Name = 'el-fakahany' and Initial = 'ee'
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM85817(NNC 11-1585)copy SMILEScopy InChI
Affinity DataKi:  0.0790nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26M35D8PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM85817(NNC 11-1585)copy SMILEScopy InChI
Affinity DataKi:  0.129nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26M35D8PubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM86231(ATR | ATROPINE | Atropine,(-) | CAS_51-55-8 | CHEM...)copy SMILEScopy InChI
Affinity DataKi:  0.550nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GX492DPubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM86231(ATR | ATROPINE | Atropine,(-) | CAS_51-55-8 | CHEM...)copy SMILEScopy InChI
Affinity DataKi:  1.64nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GX492DPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM85816(NNC 11-1607)copy SMILEScopy InChI
Affinity DataKi:  2.40nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26M35D8PubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM85817(NNC 11-1585)copy SMILEScopy InChI
Affinity DataKi:  2.57nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26M35D8PubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50176065(4-DAMP | 4-Diphenylacetoxy-1,1-dimethyl-piperidini...)copy SMILEScopy InChI
Affinity DataKi:  3.74nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GX492DPubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM85817(NNC 11-1585)copy SMILEScopy InChI
Affinity DataKi:  4.68nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26M35D8PubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM85817(NNC 11-1585)copy SMILEScopy InChI
Affinity DataKi:  5.25nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26M35D8PubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM85816(NNC 11-1607)copy SMILEScopy InChI
Affinity DataKi:  5.75nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26M35D8PubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM85816(NNC 11-1607)copy SMILEScopy InChI
Affinity DataKi:  6.03nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26M35D8PubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)copy SMILEScopy InChI
Affinity DataKi:  6.99nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GX492DPubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM85816(NNC 11-1607)copy SMILEScopy InChI
Affinity DataKi:  8.13nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26M35D8PubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM85816(NNC 11-1607)copy SMILEScopy InChI
Affinity DataKi:  8.13nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26M35D8PubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM85816(NNC 11-1607)copy SMILEScopy InChI
Affinity DataKi:  9.55nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26M35D8PubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50072228(3-[4-(3-Phenyl-prop-2-ynyloxy)-[1,2,5]thiadiazol-3...)copy SMILEScopy InChI
Affinity DataKi:  14.8nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26M35D8PubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM81799(CAS_98299-40-2 | HHSiD | NSC_3602 | hexahydrosilad...)copy SMILEScopy InChI
Affinity DataKi:  14.8nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GX492DPubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50064176(CHEMBL27673 | CHEMBL500996 | METHOCTRAMINE | N,N''...)copy SMILEScopy InChI
Affinity DataKi:  16.7nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GX492DPubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)copy SMILEScopy InChI
Affinity DataKi:  33.9nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GX492DPubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50064176(CHEMBL27673 | CHEMBL500996 | METHOCTRAMINE | N,N''...)copy SMILEScopy InChI
Affinity DataKi:  34.7nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GX492DPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50072228(3-[4-(3-Phenyl-prop-2-ynyloxy)-[1,2,5]thiadiazol-3...)copy SMILEScopy InChI
Affinity DataKi:  41.7nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26M35D8PubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50072228(3-[4-(3-Phenyl-prop-2-ynyloxy)-[1,2,5]thiadiazol-3...)copy SMILEScopy InChI
Affinity DataKi:  49nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26M35D8PubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM81799(CAS_98299-40-2 | HHSiD | NSC_3602 | hexahydrosilad...)copy SMILEScopy InChI
Affinity DataKi:  50.2nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GX492DPubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50072228(3-[4-(3-Phenyl-prop-2-ynyloxy)-[1,2,5]thiadiazol-3...)copy SMILEScopy InChI
Affinity DataKi:  58.9nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26M35D8PubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50072228(3-[4-(3-Phenyl-prop-2-ynyloxy)-[1,2,5]thiadiazol-3...)copy SMILEScopy InChI
Affinity DataKi:  77.6nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26M35D8PubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)copy SMILEScopy InChI
Affinity DataKi:  180nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GX492DPubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)copy SMILEScopy InChI
Affinity DataKi:  219nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GX492DPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50003359(5-(4-Hexyloxy-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2...)copy SMILEScopy InChI
Affinity DataIC50: 18nMpH: 6.0Assay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells at pH 6 in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VNCPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50003351(3-(4-butoxy-1,2,5-thiadiazol-3-yl)-1-methyl-1,2,5,...)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VNCPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50003359(5-(4-Hexyloxy-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2...)copy SMILEScopy InChI
Affinity DataIC50: 29nMpH: 8.0Assay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells at pH 8 in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VNCPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50003366(1-Methyl-5-(4-pentyloxy-[1,2,5]thiadiazol-3-yl)-1,...)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VNCPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50072215(1-Methyl-5-[4-(3-phenyl-prop-2-ynyloxy)-[1,2,5]thi...)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VNCPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50003369(1-Methyl-5-(4-propoxy-[1,2,5]thiadiazol-3-yl)-1,2,...)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VNCPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423615(CHEMBL405125)copy SMILEScopy InChI
Affinity DataIC50: 59nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VNCPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50003359(5-(4-Hexyloxy-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2...)copy SMILEScopy InChI
Affinity DataIC50: 81nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VNCPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50003365(3-(3-(ethoxy)-1,2,5-thiadiazol-4-yl)-1,2,5,6-tetra...)copy SMILEScopy InChI
Affinity DataIC50: 141nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VNCPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50072234(1-Methyl-5-[4-(4-phenyl-butoxy)-[1,2,5]thiadiazol-...)copy SMILEScopy InChI
Affinity DataIC50: 145nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VNCPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423611(CHEMBL270031)copy SMILEScopy InChI
Affinity DataIC50: 162nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VNCPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423607(CHEMBL408822)copy SMILEScopy InChI
Affinity DataIC50: 219nMpH: 8.0Assay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells at pH 8 in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VNCPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423607(CHEMBL408822)copy SMILEScopy InChI
Affinity DataIC50: 275nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VNCPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423614(CHEMBL403829)copy SMILEScopy InChI
Affinity DataIC50: 309nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VNCPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423607(CHEMBL408822)copy SMILEScopy InChI
Affinity DataIC50: 407nMpH: 6.0Assay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells at pH 6 in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VNCPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423613(CHEMBL271774)copy SMILEScopy InChI
Affinity DataIC50: 617nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VNCPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423609(CHEMBL406802)copy SMILEScopy InChI
Affinity DataIC50: 646nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VNCPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423608(CHEMBL272468)copy SMILEScopy InChI
Affinity DataIC50: 871nMpH: 8.0Assay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells at pH 8 in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VNCPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423608(CHEMBL272468)copy SMILEScopy InChI
Affinity DataIC50: 871nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VNCPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50003359(5-(4-Hexyloxy-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2...)copy SMILEScopy InChI
Affinity DataIC50: 955nMpH: 8.0Assay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells at pH 8 by wash-resistant binding methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VNCPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423612(CHEMBL406570)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VNCPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423619(CHEMBL257683)copy SMILEScopy InChI
Affinity DataIC50: 1.07E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VNCPubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Melbourne

Curated by PDSP Ki Database
LigandPNGBDBM50423610(CHEMBL255791)copy SMILEScopy InChI
Affinity DataIC50: 1.91E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 receptor expressed in CHO cells in continuous presence of radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VNCPubMed
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