TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University of Texas Southwestern Medical Center at Dallas
University of Texas Southwestern Medical Center at Dallas
Affinity DataIC50: 19nMpH: 7.5 T: 2°CAssay Description:Kinase activity was assayed in reaction buffer containing substrate, enzyme, and inhibitor in the presence of 0.17 mM ATP/[gamma-32P] ATP. 32P incorp...More data for this Ligand-Target Pair
Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar
In DepthDetails
Article
BindingDB Entry DOI: 10.7270/Q2XP7351PubMedDrugBank
MMDB
PDB
3D Structure (crystal)
BindingDB Entry DOI: 10.7270/Q2XP7351PubMedDrugBank
MMDB
PDB
![3D 3D](/images/Docked_3d.png)
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University of Texas Southwestern Medical Center at Dallas
University of Texas Southwestern Medical Center at Dallas
Affinity DataIC50: 25nMpH: 7.5 T: 2°CAssay Description:Kinase activity was assayed in reaction buffer containing substrate, enzyme, and inhibitor in the presence of 0.17 mM ATP/[gamma-32P] ATP. 32P incorp...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University of Texas Southwestern Medical Center at Dallas
University of Texas Southwestern Medical Center at Dallas
Affinity DataIC50: 48nMpH: 7.5 T: 2°CAssay Description:Kinase activity was assayed in reaction buffer containing substrate, enzyme, and inhibitor in the presence of 0.17 mM ATP/[gamma-32P] ATP. 32P incorp...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University of Texas Southwestern Medical Center at Dallas
University of Texas Southwestern Medical Center at Dallas
Affinity DataIC50: 160nMpH: 7.5 T: 2°CAssay Description:Kinase activity was assayed in reaction buffer containing substrate, enzyme, and inhibitor in the presence of 0.17 mM ATP/[gamma-32P] ATP. 32P incorp...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system using MBP as substrate measured after 30 mins in p...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system using MBP as substrate measured after 30 mins in p...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Rattus norvegicus)
University of Texas Southwestern Medical Center
Curated by ChEMBL
University of Texas Southwestern Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of rat TAOK2 (1 to 320 residues) expressed in Baculovirus/insect cell expression system assessed as remaining activity using MBP as substr...More data for this Ligand-Target Pair
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