Compile Data Set for Download or QSAR
Found 1145 with Last Name = 'mullady' and Initial = 'el'
LigandPNGBDBM50401261(CHEMBL2206921 | US8772480, 384)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Inhibition of human N-terminal polyHis-tagged PI3K p110delta expressed in baculovirus infected Hi5 cells using Phosphatidylinositol-4,5-bisphosphate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7QNWPubMed
LigandPNGBDBM50357645(CHEMBL1738719)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Inhibition of N-terminus polyHis-tagged human recombinant PI3Kalpha expressed in baculovirus infected insect Sf9 cells using phosphoinositol-4,5-bisp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB53C5PubMed
LigandPNGBDBM50119621(CHEMBL3618245)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Inhibition of PI3Kdelta (unknown origin) by alpha screen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49SKCPubMed
LigandPNGBDBM50357674(CHEMBL1914739)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Inhibition of N-terminus polyHis-tagged human recombinant PI3Kalpha expressed in baculovirus infected insect Sf9 cells using phosphoinositol-4,5-bisp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB53C5PubMed
LigandPNGBDBM50401261(CHEMBL2206921 | US8772480, 384)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Inhibition of human N-terminal polyHis-tagged PI3K p110beta expressed in baculovirus infected Hi5 cells using Phosphatidylinositol-4,5-bisphosphate a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7QNWPubMed
LigandPNGBDBM50357652(CHEMBL1914726)copy SMILEScopy InChI
Affinity DataKi:  0.700nMAssay Description:Inhibition of N-terminus polyHis-tagged human recombinant PI3Kalpha expressed in baculovirus infected insect Sf9 cells using phosphoinositol-4,5-bisp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB53C5PubMed
LigandPNGBDBM50357665(CHEMBL1914728)copy SMILEScopy InChI
Affinity DataKi:  0.700nMAssay Description:Inhibition of N-terminus polyHis-tagged human recombinant PI3Kalpha expressed in baculovirus infected insect Sf9 cells using phosphoinositol-4,5-bisp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB53C5PubMed
LigandPNGBDBM50357670(CHEMBL1914734)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Inhibition of N-terminus polyHis-tagged human recombinant PI3Kalpha expressed in baculovirus infected insect Sf9 cells using phosphoinositol-4,5-bisp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB53C5PubMed
LigandPNGBDBM50351949(CHEMBL1822054)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Inhibition of human N-terminal His-tagged PI3Kdelta expressed in insect Sf9 cells using PI(4,5)P2 as substrate after 20 mins by alphascreen assay in ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V12567PubMed
LigandPNGBDBM50357668(CHEMBL1914731)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Inhibition of N-terminus polyHis-tagged human recombinant PI3Kalpha expressed in baculovirus infected insect Sf9 cells using phosphoinositol-4,5-bisp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB53C5PubMed
LigandPNGBDBM50357650(CHEMBL1914742)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Inhibition of N-terminus polyHis-tagged human recombinant PI3Kalpha expressed in baculovirus infected insect Sf9 cells using phosphoinositol-4,5-bisp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB53C5PubMed
LigandPNGBDBM50357653(CHEMBL1914727)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Inhibition of N-terminus polyHis-tagged human recombinant PI3Kalpha expressed in baculovirus infected insect Sf9 cells using phosphoinositol-4,5-bisp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB53C5PubMed
LigandPNGBDBM50357662(CHEMBL1914721)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:Inhibition of PI3Kalpha-mediated Akt phosphorylation at Ser 473 in human U87MG cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB53C5PubMed
LigandPNGBDBM50357651(CHEMBL1914724)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:Inhibition of N-terminus polyHis-tagged human recombinant PI3Kalpha expressed in baculovirus infected insect Sf9 cells using phosphoinositol-4,5-bisp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB53C5PubMed
LigandPNGBDBM50357673(CHEMBL1914738)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:Inhibition of N-terminus polyHis-tagged human recombinant PI3Kalpha expressed in baculovirus infected insect Sf9 cells using phosphoinositol-4,5-bisp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB53C5PubMed
LigandPNGBDBM50357666(CHEMBL1914729)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:Inhibition of N-terminus polyHis-tagged human recombinant PI3Kalpha expressed in baculovirus infected insect Sf9 cells using phosphoinositol-4,5-bisp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB53C5PubMed
LigandPNGBDBM50357667(CHEMBL1914730)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Inhibition of PI3Kalpha-mediated Akt phosphorylation at Ser 473 in human U87MG cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB53C5PubMed
LigandPNGBDBM50343210(CHEMBL1773732 | N-(6-(6-Chloro-5-(4-chlorophenylsu...)copy SMILEScopy InChI
Affinity DataKi: <1nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8N1KPubMed
LigandPNGBDBM50343203(CHEMBL1773604 | N-(6-(6-Chloro-5-(4-methoxyphenyls...)copy SMILEScopy InChI
Affinity DataKi: <1nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8N1KPubMed
LigandPNGBDBM50343213(CHEMBL1773735 | N-(6-(6-Chloro-5-(2-fluorophenylsu...)copy SMILEScopy InChI
Affinity DataKi: <1nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8N1KPubMed
LigandPNGBDBM50343212(CHEMBL1773734 | N-(6-(6-Chloro-5-(4-tert-butylphen...)copy SMILEScopy InChI
Affinity DataKi: <1nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8N1KPubMed
LigandPNGBDBM50343209(CHEMBL1773731 | N-(6-(6-Chloro-5-(3-chlorophenylsu...)copy SMILEScopy InChI
Affinity DataKi: <1nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8N1KPubMed
LigandPNGBDBM50343208(CHEMBL1773730 | N-(6-(6-Chloro-5-(2-chlorophenylsu...)copy SMILEScopy InChI
Affinity DataKi: <1nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8N1KPubMed
LigandPNGBDBM50343207(CHEMBL1773729 | N-(6-(6-Chloro-5-(4-(trifluorometh...)copy SMILEScopy InChI
Affinity DataKi: <1nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8N1KPubMed
LigandPNGBDBM50343206(CHEMBL1773728 | N-(6-(6-Chloro-5-(3-(trifluorometh...)copy SMILEScopy InChI
Affinity DataKi: <1nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8N1KPubMed
LigandPNGBDBM50357675(CHEMBL1914740)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Inhibition of N-terminus polyHis-tagged human recombinant PI3Kalpha expressed in baculovirus infected insect Sf9 cells using phosphoinositol-4,5-bisp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB53C5PubMed
LigandPNGBDBM50396808(CHEMBL2170081 | US8772480, 148)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Inhibition of human N-terminal polyHis-tagged PI3K p110gamma expressed in baculovirus infected Hi5 cells using ATP as substrate after 20 mins by spec...More data for this Ligand-Target Pair
LigandPNGBDBM50396820(CHEMBL2170088 | US8772480, 272)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Inhibition of human N-terminal polyHis-tagged PI3K p110alpha/p85alpha expressed in baculovirus infected Sf9 cells using phosphatidylinositol-4,5-bisp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028SPTPubMed
LigandPNGBDBM50343205(CHEMBL1773606 | N-(6-(6-Chloro-5-(2-(trifluorometh...)copy SMILEScopy InChI
Affinity DataKi: <1nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8N1KPubMed
LigandPNGBDBM50357664(CHEMBL1914723)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Inhibition of PI3Kalpha-mediated Akt phosphorylation at Ser 473 in human U87MG cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB53C5PubMed
LigandPNGBDBM50357644(CHEMBL1914947)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Inhibition of N-terminus polyHis-tagged human recombinant PI3Kalpha expressed in baculovirus infected insect Sf9 cells using phosphoinositol-4,5-bisp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB53C5PubMed
LigandPNGBDBM50343211(CHEMBL1773733 | N-(6-(5-(3-tert-Butylphenylsulfona...)copy SMILEScopy InChI
Affinity DataKi: <1nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8N1KPubMed
LigandPNGBDBM50396806(CHEMBL2170083 | US8772480, 270)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Inhibition of human N-terminal polyHis-tagged PI3K p110delta/p85alpha expressed in baculovirus infected Sf9 cells using phosphatidylinositol-4,5-bisp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028SPTPubMed
LigandPNGBDBM50396807(CHEMBL2170082 | US8772480, 316)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Inhibition of human N-terminal polyHis-tagged PI3K p110delta/p85alpha expressed in baculovirus infected Sf9 cells using phosphatidylinositol-4,5-bisp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028SPTPubMed
LigandPNGBDBM50396809(CHEMBL2170099 | US8772480, 147)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Inhibition of human N-terminal polyHis-tagged PI3K p110delta/p85alpha expressed in baculovirus infected Sf9 cells using phosphatidylinositol-4,5-bisp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2028SPTPubMed
LigandPNGBDBM50394838(CHEMBL2165007 | US8772480, 141)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Inhibition of human N-terminal poly-His tagged-PI3Kdelta expressed in Sf9 baculovirus system co-expressing p85alpha after 20 mins by AlphaScreen assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4QSJPubMed
LigandPNGBDBM50401261(CHEMBL2206921 | US8772480, 384)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Inhibition of human N-terminal polyHis-tagged PI3K p110gamma expressed in baculovirus infected Hi5 cells using Phosphatidylinositol-4,5-bisphosphate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7QNWPubMed
LigandPNGBDBM50343214(CHEMBL1773736 | N-(6-(6-Chloro-5-(3-fluorophenylsu...)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8N1KPubMed
LigandPNGBDBM50401256(CHEMBL2206904 | US8772480, 331)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Inhibition of human N-terminal polyHis-tagged PI3K p110delta expressed in baculovirus infected Hi5 cells using Phosphatidylinositol-4,5-bisphosphate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7QNWPubMed
LigandPNGBDBM50343200(CHEMBL1615189 | N-(6-(6-Chloro-5-(4-fluorophenylsu...)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Inhibition of human PI3Kalpha using PI(4,5)P2 as substrate after 20 mins by alphascreen assay in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V12567PubMed
LigandPNGBDBM50343200(CHEMBL1615189 | N-(6-(6-Chloro-5-(4-fluorophenylsu...)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8N1KPubMed
LigandPNGBDBM50343200(CHEMBL1615189 | N-(6-(6-Chloro-5-(4-fluorophenylsu...)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Inhibition of human PI3Kdelta expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8N1KPubMed
LigandPNGBDBM50343202(CHEMBL1773603 | N-(6-(5-(4-Methoxyphenylsulfonamid...)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8N1KPubMed
LigandPNGBDBM50401269(CHEMBL2206913)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Inhibition of human N-terminal polyHis-tagged PI3K p110delta expressed in baculovirus infected Hi5 cells using Phosphatidylinositol-4,5-bisphosphate ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7QNWPubMed
LigandPNGBDBM50351952(CHEMBL1822057)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Inhibition of human PI3Kalpha using PI(4,5)P2 as substrate after 20 mins by alphascreen assay in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V12567PubMed
LigandPNGBDBM50343200(CHEMBL1615189 | N-(6-(6-Chloro-5-(4-fluorophenylsu...)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Inhibition of PI3Kalpha-mediated Akt phosphorylation at Ser 473 in human U87MG cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB53C5PubMed
LigandPNGBDBM50357643(CHEMBL1914725)copy SMILEScopy InChI
Affinity DataKi:  1.30nMAssay Description:Inhibition of N-terminus polyHis-tagged human recombinant PI3Kalpha expressed in baculovirus infected insect Sf9 cells using phosphoinositol-4,5-bisp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB53C5PubMed
LigandPNGBDBM50343204(CHEMBL1773605 | N-(6-(6-Chloro-5-(phenylsulfonamid...)copy SMILEScopy InChI
Affinity DataKi:  1.40nMAssay Description:Inhibition of human PI3Kalpha expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8N1KPubMed
LigandPNGBDBM50351949(CHEMBL1822054)copy SMILEScopy InChI
Affinity DataKi:  1.40nMAssay Description:Inhibition of human PI3Kalpha using PI(4,5)P2 as substrate after 20 mins by alphascreen assay in presence of 20 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V12567PubMed
LigandPNGBDBM50357669(CHEMBL1914732)copy SMILEScopy InChI
Affinity DataKi:  1.40nMAssay Description:Inhibition of N-terminus polyHis-tagged human recombinant PI3Kalpha expressed in baculovirus infected insect Sf9 cells using phosphoinositol-4,5-bisp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB53C5PubMed
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