Compile Data Set for Download or QSAR
Found 3290 with Last Name = 'de ceuninck' and Initial = 'f'
LigandPNGBDBM194644(US9206139, 3)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of human recombinant ADAMTS5 using synthetic peptide as substrate by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VBMPubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
University of Illinois at Chicago

LigandPNGBDBM379774(US9926281, Compound 279 | US9926281, Compound 448)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:MMP2: Protocol 2: The basis for the assay is the cleavage of the substrate 390 MMP FRET substrate I (Anaspec, Catalog n#: AS-27076) by human MMP2 (R&...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27S7R3TUS Patent
LigandPNGBDBM194644(US9206139, 3)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of human recombinant ADAMTS4 using synthetic peptide as substrate by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VBMPubMed
TargetADAMTS5(Rattus norvegicus (Rat))
University of Illinois at Chicago

LigandPNGBDBM379670(US9926281, Compound 194 | US9926281, Compound 413)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27S7R3TUS Patent
TargetADAMTS5(Rattus norvegicus (Rat))
University of Illinois at Chicago

LigandPNGBDBM379686(US9926281, Compound 212)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27S7R3TUS Patent
TargetCollagenase 3(Homo sapiens (Human))
University of Illinois at Chicago

LigandPNGBDBM379776(US9926281, Compound 234)copy SMILEScopy InChI
Affinity DataIC50: 5.60nMAssay Description:MMP-13:The basis for the assay is the cleavage of the substrate 390 MMP FRET Substrate I (Anaspec Cat # AS-27076) by human MMP13 (Chemicon, Cat #CC06...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27S7R3TUS Patent
TargetADAMTS5(Rattus norvegicus (Rat))
University of Illinois at Chicago

LigandPNGBDBM379681(US9926281, Compound 207 | US9926281, Compound 416)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27S7R3TUS Patent
TargetADAMTS5(Rattus norvegicus (Rat))
University of Illinois at Chicago

LigandPNGBDBM379668(US9926281, Compound 192 | US9926281, Compound 411)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27S7R3TUS Patent
TargetADAMTS5(Rattus norvegicus (Rat))
University of Illinois at Chicago

LigandPNGBDBM379669(US9926281, Compound 193 | US9926281, Compound 412)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27S7R3TUS Patent
TargetADAMTS5(Rattus norvegicus (Rat))
University of Illinois at Chicago

LigandPNGBDBM379653(US9926281, Compound 176)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27S7R3TUS Patent
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
University of Illinois at Chicago

LigandPNGBDBM379901(US9926281, Compound 396)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:MMP-14:The basis for the assay is the cleavage of the substrate 390 MMP FRET Substrate I (Anaspec Cat # AS-27076) by human MMP14 (Biomol, Cat #SE-259...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27S7R3TUS Patent
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
University of Illinois at Chicago

LigandPNGBDBM379776(US9926281, Compound 234)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:MMP-14:The basis for the assay is the cleavage of the substrate 390 MMP FRET Substrate I (Anaspec Cat # AS-27076) by human MMP14 (Biomol, Cat #SE-259...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27S7R3TUS Patent
LigandPNGBDBM50575720(CHEMBL4864283)copy SMILES
Affinity DataIC50: 8nMAssay Description:Inhibition of human recombinant ADAMTS5 using synthetic peptide as substrate by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VBMPubMed
TargetADAMTS5(Rattus norvegicus (Rat))
University of Illinois at Chicago

LigandPNGBDBM379645(US9926281, Compound 167 | US9926281, Compound 408)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27S7R3TUS Patent
LigandPNGBDBM379668(US9926281, Compound 192 | US9926281, Compound 411)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:ADAMTS-5:Protocol 2: The basis for the assay is the cleavage of the substrate TBIS-1 (5 FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27S7R3TUS Patent
LigandPNGBDBM379670(US9926281, Compound 194 | US9926281, Compound 413)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:ADAMTS-5:Protocol 2: The basis for the assay is the cleavage of the substrate TBIS-1 (5 FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27S7R3TUS Patent
TargetADAMTS5(Rattus norvegicus (Rat))
University of Illinois at Chicago

LigandPNGBDBM379667(US9926281, Compound 191)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27S7R3TUS Patent
LigandPNGBDBM379670(US9926281, Compound 194 | US9926281, Compound 413)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:ADAMTS-5:Protocol 2: The basis for the assay is the cleavage of the substrate TBIS-1 (5 FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27S7R3TUS Patent
TargetADAMTS5(Rattus norvegicus (Rat))
University of Illinois at Chicago

LigandPNGBDBM379649(US9926281, Compound 172 | US9926281, Compound 409)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27S7R3TUS Patent
LigandPNGBDBM379668(US9926281, Compound 192 | US9926281, Compound 411)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:ADAMTS-5:Protocol 2: The basis for the assay is the cleavage of the substrate TBIS-1 (5 FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27S7R3TUS Patent
TargetADAMTS5(Rattus norvegicus (Rat))
University of Illinois at Chicago

LigandPNGBDBM379678(US9926281, Compound 204)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:ADAMTS-4:The basis for the assay is the cleavage of the substrate TBIS-1 (5-FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMTS4For the do...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27S7R3TUS Patent
LigandPNGBDBM379681(US9926281, Compound 207 | US9926281, Compound 416)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:ADAMTS-5:Protocol 2: The basis for the assay is the cleavage of the substrate TBIS-1 (5 FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27S7R3TUS Patent
LigandPNGBDBM379686(US9926281, Compound 212)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:ADAMTS-5:Protocol 2: The basis for the assay is the cleavage of the substrate TBIS-1 (5 FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27S7R3TUS Patent
LigandPNGBDBM379686(US9926281, Compound 212)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of human recombinant ADAMTS-5 assessed as cleavage of fluorescent substrate using FAM-TBIS-1 by biochemical assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VBMPubMed
LigandPNGBDBM379975(US9926281, Compound 436)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of human recombinant ADAMTS-4 (AA1 to 520) assessed as cleavage of fluorescent substrate using as TBIS-1 substrate incubated for 180 mins ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VBMPubMed
LigandPNGBDBM379681(US9926281, Compound 207 | US9926281, Compound 416)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:ADAMTS-5:Protocol 2: The basis for the assay is the cleavage of the substrate TBIS-1 (5 FAM-TEGEARGSVILLK (5TAMRA)K-NH2) (SEQ ID No 2) by human ADAMT...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27S7R3TUS Patent
LigandPNGBDBM429689(5-(3-(4-(4- chloro-3,5- dimethoxy- phenyl)piperidi...)copy SMILEScopy InChI
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate 520 MMP FRET substrate XII by human ADAMTS6.The substrate contains sequence Arg-Pro-Lys-Pro-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D2211NUS Patent
LigandPNGBDBM429691(5-(3-(4-(4- chlorophenyl) piperidin-1- yl)-2-methy...)copy SMILEScopy InChI
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate 520 MMP FRET substrate XII by human ADAMTS6.The substrate contains sequence Arg-Pro-Lys-Pro-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D2211NUS Patent
LigandPNGBDBM429692(5-(3-(4-(3,5- dichlorophenyl) piperidin-1- yl)-2-m...)copy SMILEScopy InChI
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate 520 MMP FRET substrate XII by human ADAMTS6.The substrate contains sequence Arg-Pro-Lys-Pro-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D2211NUS Patent
LigandPNGBDBM429715(5-(3-(4-(4- chloro-3- methoxyl- phenyl)piperidin-1...)copy SMILEScopy InChI
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate 520 MMP FRET substrate XII by human ADAMTS6.The substrate contains sequence Arg-Pro-Lys-Pro-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D2211NUS Patent
LigandPNGBDBM429716(5-(3-(4-(4- chloro-5- methoxy-2- methylphenyl) pip...)copy SMILEScopy InChI
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate 520 MMP FRET substrate XII by human ADAMTS6.The substrate contains sequence Arg-Pro-Lys-Pro-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D2211NUS Patent
LigandPNGBDBM429723(5-(3-(4-(4- chloro-2- methoxyphenyl) piperidin-1- ...)copy SMILEScopy InChI
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate 520 MMP FRET substrate XII by human ADAMTS6.The substrate contains sequence Arg-Pro-Lys-Pro-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D2211NUS Patent
LigandPNGBDBM429724(5-(3-(4-(3,4- difluoro-5- methoxyphenyl) piperidin...)copy SMILEScopy InChI
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate 520 MMP FRET substrate XII by human ADAMTS6.The substrate contains sequence Arg-Pro-Lys-Pro-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D2211NUS Patent
LigandPNGBDBM429725((R)-5-(3-(4-(4- chloro-3- fluoro-5- methoxyphenyl)...)copy SMILEScopy InChI
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate 520 MMP FRET substrate XII by human ADAMTS6.The substrate contains sequence Arg-Pro-Lys-Pro-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D2211NUS Patent
LigandPNGBDBM429726(5-(3-(4-(4- chloro-3- fluoro-5- methoxyphenyl) pip...)copy SMILEScopy InChI
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate 520 MMP FRET substrate XII by human ADAMTS6.The substrate contains sequence Arg-Pro-Lys-Pro-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D2211NUS Patent
LigandPNGBDBM429740((R)-5-(3-(4- (4,5-dichloro- 2- methoxyphenyl) pipe...)copy SMILEScopy InChI
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate 520 MMP FRET substrate XII by human ADAMTS6.The substrate contains sequence Arg-Pro-Lys-Pro-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D2211NUS Patent
LigandPNGBDBM429741(5-(3-(4-(4,5- dichloro-2- methoxyphenyl) piperidin...)copy SMILEScopy InChI
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate 520 MMP FRET substrate XII by human ADAMTS6.The substrate contains sequence Arg-Pro-Lys-Pro-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D2211NUS Patent
LigandPNGBDBM429745((R)-5-(3-(4-(3- chloro-5- methoxyphenyl) piperidin...)copy SMILEScopy InChI
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate 520 MMP FRET substrate XII by human ADAMTS6.The substrate contains sequence Arg-Pro-Lys-Pro-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D2211NUS Patent
LigandPNGBDBM429747((R)-5-(3-(4- (3,4-dichloro-5- methoxyphenyl) piper...)copy SMILEScopy InChI
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate 520 MMP FRET substrate XII by human ADAMTS6.The substrate contains sequence Arg-Pro-Lys-Pro-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D2211NUS Patent
LigandPNGBDBM429748((R)-5-(3-(4- (3,4-dichloro-5- methoxyphenyl) piper...)copy SMILEScopy InChI
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate 520 MMP FRET substrate XII by human ADAMTS6.The substrate contains sequence Arg-Pro-Lys-Pro-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D2211NUS Patent
LigandPNGBDBM429750(5-(3-(4-(4,5- dichloro-2- methylphenyl) piperidin-...)copy SMILEScopy InChI
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate 520 MMP FRET substrate XII by human ADAMTS6.The substrate contains sequence Arg-Pro-Lys-Pro-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D2211NUS Patent
LigandPNGBDBM429751(5-(3-(4-(4- fluoro-3,5- dimethoxyphenyl) piperidin...)copy SMILEScopy InChI
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate 520 MMP FRET substrate XII by human ADAMTS6.The substrate contains sequence Arg-Pro-Lys-Pro-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D2211NUS Patent
LigandPNGBDBM429752(5-(3-(4-(3- chloro-4- fluoro-5- methoxyphenyl) pip...)copy SMILEScopy InChI
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate 520 MMP FRET substrate XII by human ADAMTS6.The substrate contains sequence Arg-Pro-Lys-Pro-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D2211NUS Patent
LigandPNGBDBM429758((5R)-5-[3-[4- (4-chloro-2- methoxy- phenyl)-1- pip...)copy SMILEScopy InChI
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate 520 MMP FRET substrate XII by human ADAMTS6.The substrate contains sequence Arg-Pro-Lys-Pro-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D2211NUS Patent
LigandPNGBDBM429759((5R)-5-[3-[4- (3-chloro-4- fluoro-5- methoxy- phen...)copy SMILEScopy InChI
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate 520 MMP FRET substrate XII by human ADAMTS6.The substrate contains sequence Arg-Pro-Lys-Pro-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D2211NUS Patent
LigandPNGBDBM429760((5R)-5-[3-[4- (4-fluoro-3,5- dimethoxy- phenyl)-1-...)copy SMILEScopy InChI
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate 520 MMP FRET substrate XII by human ADAMTS6.The substrate contains sequence Arg-Pro-Lys-Pro-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D2211NUS Patent
LigandPNGBDBM429761((5R)-5-[3-[4- (4-fluoro-3,5- dimethoxy- phenyl)-1-...)copy SMILEScopy InChI
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate 520 MMP FRET substrate XII by human ADAMTS6.The substrate contains sequence Arg-Pro-Lys-Pro-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D2211NUS Patent
LigandPNGBDBM429763((5R)-5-[3-[4- (4-chloro-3- fluoro-5- methoxy- phen...)copy SMILEScopy InChI
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate 520 MMP FRET substrate XII by human ADAMTS6.The substrate contains sequence Arg-Pro-Lys-Pro-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D2211NUS Patent
LigandPNGBDBM429765((5R)-5-[3-[4- (4-chloro-3- methoxy- phenyl)-1- pip...)copy SMILEScopy InChI
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate 520 MMP FRET substrate XII by human ADAMTS6.The substrate contains sequence Arg-Pro-Lys-Pro-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D2211NUS Patent
LigandPNGBDBM429767((5R)-5-[3-[4- (4-chloro-3- ethoxy-5- methoxy- phen...)copy SMILEScopy InChI
Affinity DataIC50: 12.5nMAssay Description:The basis for the assay is the cleavage of the substrate 520 MMP FRET substrate XII by human ADAMTS6.The substrate contains sequence Arg-Pro-Lys-Pro-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D2211NUS Patent
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