Affinity DataKi: 1.90nMAssay Description:Competitive inhibition of recombinant furin (unknown origin) using as substrate after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Competitive inhibition of recombinant furin (unknown origin) using as substrate after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Competitive inhibition of recombinant furin (unknown origin) using as substrate after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Competitive inhibition of recombinant furin (unknown origin) using as substrate after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Competitive inhibition of recombinant furin (unknown origin) using as substrate after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Competitive inhibition of recombinant furin (unknown origin) using as substrate after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Competitive inhibition of recombinant furin (unknown origin) using as substrate after 60 minsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University of Li£ge
Curated by ChEMBL
University of Li£ge
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:Displacement of [125I]-apamin from cloned SK3 channel expressed in human HEK293 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 89nMAssay Description:Competitive inhibition of recombinant furin (unknown origin) using as substrate after 60 minsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 2(Homo sapiens (Human))
University of Li£ge
Curated by ChEMBL
University of Li£ge
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Displacement of [125I]-apamin from cloned SK2 channel expressed in human HEK293 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 123nMAssay Description:Competitive inhibition of recombinant furin (unknown origin) using as substrate after 60 minsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 2(Homo sapiens (Human))
University of Li£ge
Curated by ChEMBL
University of Li£ge
Curated by ChEMBL
Affinity DataKi: 194nMAssay Description:Displacement of [125I]-apamin from cloned SK2 channel expressed in human HEK293 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University of Li£ge
Curated by ChEMBL
University of Li£ge
Curated by ChEMBL
Affinity DataKi: 214nMAssay Description:Displacement of [125I]-apamin from cloned SK3 channel expressed in human HEK293 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 2(Homo sapiens (Human))
University of Li£ge
Curated by ChEMBL
University of Li£ge
Curated by ChEMBL
Affinity DataKi: 397nMAssay Description:Displacement of [125I]-apamin from cloned SK2 channel expressed in human HEK293 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University of Li£ge
Curated by ChEMBL
University of Li£ge
Curated by ChEMBL
Affinity DataKi: 575nMAssay Description:Displacement of [125I]-apamin from cloned SK3 channel expressed in human HEK293 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 591nMAssay Description:Competitive inhibition of recombinant furin (unknown origin) using as substrate after 60 minsMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 2(Homo sapiens (Human))
University of Li£ge
Curated by ChEMBL
University of Li£ge
Curated by ChEMBL
Affinity DataKi: 593nMAssay Description:Displacement of [125I]-apamin from cloned SK2 channel expressed in human HEK293 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University of Li£ge
Curated by ChEMBL
University of Li£ge
Curated by ChEMBL
Affinity DataKi: 837nMAssay Description:Displacement of [125I]-apamin from cloned SK3 channel expressed in human HEK293 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 2(Homo sapiens (Human))
University of Li£ge
Curated by ChEMBL
University of Li£ge
Curated by ChEMBL
Affinity DataKi: 878nMAssay Description:Displacement of [125I]-apamin from cloned SK2 channel expressed in human HEK293 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University of Li£ge
Curated by ChEMBL
University of Li£ge
Curated by ChEMBL
Affinity DataKi: 1.27E+3nMAssay Description:Displacement of [125I]-apamin from cloned SK3 channel expressed in human HEK293 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
PSL Research University
Curated by ChEMBL
PSL Research University
Curated by ChEMBL
Affinity DataIC50: 0.770nMAssay Description:Inhibition of recombinant His-tagged human Axl (473 to end residues) cytoplasmic domain expressed in insect system using poly (Glu-Ala-Tyr) peptide a...More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of recombinant GST-tagged human Mer (578 to 872 residues) cytoplasmic domain expressed in Baculovirus system using poly (Glu-Ala-Tyr) pept...More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant GST-tagged human Mer (578 to 872 residues) cytoplasmic domain expressed in Baculovirus system using poly (Glu-Ala-Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
PSL Research University
Curated by ChEMBL
PSL Research University
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of recombinant His-tagged human Axl (473 to end residues) cytoplasmic domain expressed in insect system using poly (Glu-Ala-Tyr) peptide a...More data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of recombinant GST-tagged human Mer (578 to 872 residues) cytoplasmic domain expressed in Baculovirus system using poly (Glu-Ala-Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
PSL Research University
Curated by ChEMBL
PSL Research University
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Inhibition of recombinant GST-tagged human Tyro3 (451 to 890 residues) cytoplasmic domain expressed in Baculovirus expression system using poly (Glu-...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
PSL Research University
Curated by ChEMBL
PSL Research University
Curated by ChEMBL
Affinity DataIC50: 690nMAssay Description:Inhibition of recombinant GST-tagged human Tyro3 (451 to 890 residues) cytoplasmic domain expressed in Baculovirus expression system using poly (Glu-...More data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 2(Rattus norvegicus (Rat))
University of Li£ge
Curated by ChEMBL
University of Li£ge
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of cloned rat SK2 channel expressed in human HEK293 cells by patch clamp assay in the presence of 1 uM intracellular Ca2+More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
PSL Research University
Curated by ChEMBL
PSL Research University
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of recombinant His-tagged human Axl (473 to end residues) cytoplasmic domain expressed in insect system using poly (Glu-Ala-Tyr) peptide a...More data for this Ligand-Target Pair
TargetSmall conductance calcium-activated potassium channel protein 3(Homo sapiens (Human))
University of Li£ge
Curated by ChEMBL
University of Li£ge
Curated by ChEMBL
Affinity DataIC50: 2.97E+3nMAssay Description:Inhibition of cloned human SK3 channel expressed in human HEK293 cells by patch clamp assay in the presence of 1 uM intracellular Ca2+More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
PSL Research University
Curated by ChEMBL
PSL Research University
Curated by ChEMBL
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of recombinant GST-tagged human Tyro3 (451 to 890 residues) cytoplasmic domain expressed in Baculovirus expression system using poly (Glu-...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant GST-tagged human Mer (578 to 872 residues) cytoplasmic domain expressed in Baculovirus system using poly (Glu-Ala-Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
PSL Research University
Curated by ChEMBL
PSL Research University
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant His-tagged human Axl (473 to end residues) cytoplasmic domain expressed in insect system using poly (Glu-Ala-Tyr) peptide a...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor TYRO3(Homo sapiens (Human))
PSL Research University
Curated by ChEMBL
PSL Research University
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant GST-tagged human Tyro3 (451 to 890 residues) cytoplasmic domain expressed in Baculovirus expression system using poly (Glu-...More data for this Ligand-Target Pair
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