Compile Data Set for Download or QSAR
Found 600 with Last Name = 'herold' and Initial = 'f'
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM194780(7-(4-(4-(1-benzothiophen-4-yl)piperazin-1-yl)butox...)copy SMILEScopy InChI
Affinity DataKi:  0.120nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W0996HPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279520(2-{4-[4-(1H-Indol-3-yl)-piperidin-1-yl]-butyl}-4-p...)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]citalopram from 5HTT in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N5249PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM194780(7-(4-(4-(1-benzothiophen-4-yl)piperazin-1-yl)butox...)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cells incubated for 1 hr by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W0996HPubMedDrugBank
TargetD(2) dopamine receptor(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)copy SMILEScopy InChI
Affinity DataKi:  0.340nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cells incubated for 1 hr by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W0996HPubMedDrugBank
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM194780(7-(4-(4-(1-benzothiophen-4-yl)piperazin-1-yl)butox...)copy SMILEScopy InChI
Affinity DataKi:  0.398nMAssay Description:Binding affinity to 5-HT2BR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W0996HPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50558342(CHEMBL4754231)copy SMILES
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H] Spiperone from rat striatum dopamine D2 receptor measured after 30 mins by liquid scintillation counter methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52T9KPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50558348(CHEMBL4743158)copy SMILES
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H] Spiperone from rat striatum dopamine D2 receptor measured after 30 mins by liquid scintillation counter methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52T9KPubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM194780(7-(4-(4-(1-benzothiophen-4-yl)piperazin-1-yl)butox...)copy SMILEScopy InChI
Affinity DataKi:  0.470nMAssay Description:Displacement of [3H]-Ketanserin from human 5-HT2A receptor expressed in rat cortex tissue incubated for 30 mins by liquid scintillation counting meth...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W0996HPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50443101(Cariprazine | RGH-188)copy SMILEScopy InChI
Affinity DataKi:  0.490nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cells incubated for 1 hr by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W0996HPubMedDrugBank
TargetD(2) dopamine receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50366495((+)butaclamol | CHEMBL1255588)copy SMILEScopy InChI
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat straitum tissue after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z0395DPubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM85222(CAS_441351-20-8 | Lurasidone | SM 13496)copy SMILEScopy InChI
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]-5-CT from human 5HT7 receptor expressed in HEK293 cells incubated for 1 hr by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W0996HPubMedDrugBank
TargetD(2) dopamine receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50558345(CHEMBL4788843)copy SMILES
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H] Spiperone from rat striatum dopamine D2 receptor measured after 30 mins by liquid scintillation counter methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52T9KPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50279541(2-(4-(4-(1H-indol-3-yl)piperidin-1-yl)butyl)-4-(2-...)copy SMILEScopy InChI
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]citalopram from 5HTT in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N5249PubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM30708((6aR,9R)-4,7-dimethyl-N-[(1S)-1-methylolpropyl]-6,...)copy SMILEScopy InChI
Affinity DataKi:  0.794nMAssay Description:Binding affinity to 5-HT2CR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W0996HPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM85222(CAS_441351-20-8 | Lurasidone | SM 13496)copy SMILEScopy InChI
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cells incubated for 1 hr by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W0996HPubMedDrugBank
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)copy SMILEScopy InChI
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50001888((chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)...)copy SMILEScopy InChI
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]-raclopride from human D2 receptor expressed in HEK cells incubated for 1 hr by Cheng-Prusoff analysis based microbeta scintillat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B63H7PubMedDrugBank
TargetD(2) dopamine receptor(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50001888((chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)...)copy SMILEScopy InChI
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]-raclopride from recombinant human D2 receptor expressed in HEK293 cells measured after 1 hr by microbeta scintillation counting ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61PPWPubMedDrugBank
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50151982(5-{4-[4-(5-Cyano-1H-indol-3-yl)-butyl]-piperazin-1...)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]-imipramine from human serotonin transporter expressed in HEK293 cells membranes incubated for 30 mins by microbeta scintillation...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM30708((6aR,9R)-4,7-dimethyl-N-[(1S)-1-methylolpropyl]-6,...)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Binding affinity to 5-HT2BR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W0996HPubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM85222(CAS_441351-20-8 | Lurasidone | SM 13496)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-Ketanserin from human 5-HT2A receptor expressed in rat cortex tissue incubated for 30 mins by liquid scintillation counting meth...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W0996HPubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))TBA
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)copy SMILEScopy InChI
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]-8-OH-DPAT from rat cerebral cortex 5HT1A receptor measured after 15 mins by liquid scintillation counter methodMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50504436(CHEMBL4591440)copy SMILEScopy InChI
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W0996HPubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50010859(CHEMBL11 | IMIPRAMINE HYDROCHLORIDE | IMIPRAMINE P...)copy SMILEScopy InChI
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]-imipramine from human serotonin transporter expressed in HEK293 cells membranes incubated for 30 mins by microbeta scintillation...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50354102(CHEMBL1836107)copy SMILEScopy InChI
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z0395DPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50443101(Cariprazine | RGH-188)copy SMILEScopy InChI
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W0996HPubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))TBA
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)copy SMILEScopy InChI
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]8OH-DPAT from 5HT1A in rat brain cerebral cortex after 15 mins by scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50222218(CHEBI:51137 | Mianserin)copy SMILEScopy InChI
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]-ketanserin from recombinant human 5HT2A receptor expressed in HEK293 cells measured after 1.5 hrs by microbeta scintillation cou...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61PPWPubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50222218(CHEBI:51137 | Mianserin)copy SMILEScopy InChI
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]ketanserin from human 5HT2A receptor expressed in HEK293 cells incubated for 1.5 hrs by Cheng-Prusoff analysis based microbeta sc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B63H7PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50504435(CHEMBL4454176)copy SMILEScopy InChI
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W0996HPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50558349(CHEMBL4764971)copy SMILES
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H] Spiperone from rat striatum dopamine D2 receptor measured after 30 mins by liquid scintillation counter methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52T9KPubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)copy SMILEScopy InChI
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]-Ketanserin from human 5-HT2A receptor expressed in rat cortex tissue incubated for 30 mins by liquid scintillation counting meth...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W0996HPubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50558343(CHEMBL4748723)copy SMILES
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H] Spiperone from rat striatum dopamine D2 receptor measured after 30 mins by liquid scintillation counter methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52T9KPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)copy SMILEScopy InChI
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM194780(7-(4-(4-(1-benzothiophen-4-yl)piperazin-1-yl)butox...)copy SMILEScopy InChI
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]-5-CT from human 5HT7 receptor expressed in HEK293 cells incubated for 1 hr by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W0996HPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50062156(CHEMBL3397081)copy SMILEScopy InChI
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]citalopram from rat brain cerebral cortex SERT by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ34CBPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)copy SMILEScopy InChI
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]-raclopride from recombinant human D2 receptor expressed in HEK293 cells measured after 1 hr by microbeta scintillation counting ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61PPWPubMedDrugBank
TargetD(2) dopamine receptor(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)copy SMILEScopy InChI
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]-raclopride from human D2 receptor expressed in HEK cells incubated for 1 hr by Cheng-Prusoff analysis based microbeta scintillat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B63H7PubMedDrugBank
TargetD(2) dopamine receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50558339(CHEMBL4744722)copy SMILES
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H] Spiperone from rat striatum dopamine D2 receptor measured after 30 mins by liquid scintillation counter methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52T9KPubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM35254(2-methyl-4-(4-methylpiperazin-1-yl)-10H-thieno[2,3...)copy SMILEScopy InChI
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]ketanserin from human 5HT2A receptor expressed in HEK293 cells incubated for 1.5 hrs by Cheng-Prusoff analysis based microbeta sc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B63H7PubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM35254(2-methyl-4-(4-methylpiperazin-1-yl)-10H-thieno[2,3...)copy SMILEScopy InChI
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]-ketanserin from recombinant human 5HT2A receptor expressed in HEK293 cells measured after 1.5 hrs by microbeta scintillation cou...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M61PPWPubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))TBA
LigandPNGBDBM50279541(2-(4-(4-(1H-indol-3-yl)piperidin-1-yl)butyl)-4-(2-...)copy SMILEScopy InChI
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N5249PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM78940(METHIOTHEPIN | MLS000859918 | Methiothepin mesylat...)copy SMILEScopy InChI
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23B63H7PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50504438(CHEMBL4571321)copy SMILEScopy InChI
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W0996HPubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM31005(2-methyl-1,2,3,4,10,14b-hexahydrodibenzo[c,f]pyraz...)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Displacement of [3H]ketanserin from 5HT2A in rat brain cerebral cortex after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z0395DPubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM50062173(CHEMBL3397082)copy SMILEScopy InChI
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]citalopram from rat brain cerebral cortex SERT by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ34CBPubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)copy SMILEScopy InChI
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))TBA
LigandPNGBDBM50062241(CHEMBL3397075)copy SMILEScopy InChI
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]8-OH-DPAT from rat brain hippocampus 5-HT1A receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ34CBPubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))TBA
LigandPNGBDBM50279520(2-{4-[4-(1H-Indol-3-yl)-piperidin-1-yl]-butyl}-4-p...)copy SMILEScopy InChI
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22N5249PubMed
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