Compile Data Set for Download or QSAR
Found 19 with Last Name = 'martel' and Initial = 'f'
TargetSolute carrier family 22 member 1(RAT)
University of Heidelberg

Curated by ChEMBL
LigandPNGBDBM50420215(CHEMBL339858)copy SMILEScopy InChI
Affinity DataKi:  110nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7QSPPubMed
TargetSolute carrier family 22 member 1(RAT)
University of Heidelberg

Curated by ChEMBL
LigandPNGBDBM39687((2E)-1-ethyl-2-[(1-ethyl-2-quinolin-1-iumyl)methyl...)copy SMILEScopy InChI
Affinity DataKi:  500nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7QSPPubMed
TargetSolute carrier family 22 member 1(RAT)
University of Heidelberg

Curated by ChEMBL
LigandPNGBDBM50420192(CHEMBL2074851)copy SMILEScopy InChI
Affinity DataKi:  670nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7QSPPubMed
TargetSolute carrier family 22 member 1(RAT)
University of Heidelberg

Curated by ChEMBL
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)copy SMILEScopy InChI
Affinity DataKi:  1.40E+3nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7QSPPubMed
TargetSolute carrier family 22 member 1(RAT)
University of Heidelberg

Curated by ChEMBL
LigandPNGBDBM50367247(QUININE | Quinamm | Quinsan | cid_3034034)copy SMILEScopy InChI
Affinity DataKi:  4.30E+3nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7QSPPubMed
TargetSolute carrier family 22 member 1(RAT)
University of Heidelberg

Curated by ChEMBL
LigandPNGBDBM50017681((1S,2R,4S,5R)-2-[(S)-Hydroxy-(6-methoxy-quinolin-4...)copy SMILEScopy InChI
Affinity DataKi:  6.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7QSPPubMed
TargetSolute carrier family 22 member 1(RAT)
University of Heidelberg

Curated by ChEMBL
LigandPNGBDBM50420217(METIPRENALINE)copy SMILEScopy InChI
Affinity DataKi:  2.50E+4nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7QSPPubMed
TargetSolute carrier family 22 member 1(RAT)
University of Heidelberg

Curated by ChEMBL
LigandPNGBDBM50170653((11beta)-11,21-dihydroxypregn-4-ene-3,20-dione | 1...)copy SMILEScopy InChI
Affinity DataKi:  7.20E+4nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in OCT1-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7QSPPubMed
TargetSolute carrier family 22 member 3(Homo sapiens (Human))
Universidade do Porto

Curated by ChEMBL
LigandPNGBDBM50420192(CHEMBL2074851)copy SMILEScopy InChI
Affinity DataIC50: 1.76E+3nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake (MPP+: 0.2 uM) in OCT3-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ702RPubMed
TargetSolute carrier family 22 member 3(Homo sapiens (Human))
Universidade do Porto

Curated by ChEMBL
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)copy SMILEScopy InChI
Affinity DataIC50: 7.93E+4nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake (MPP+: 0.2 uM) in OCT3-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ702RPubMed
TargetATP-dependent RNA helicase DDX1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50537057(CHEMBL4551611)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of human DDX1 helicase activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06BJKPubMed
TargetATP-dependent RNA helicase DDX1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50537055(CHEMBL4591917)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of human DDX1 helicase activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06BJKPubMed
TargetATP-dependent RNA helicase DDX1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50537056(CHEMBL4571759)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of human DDX1 helicase activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06BJKPubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50537055(CHEMBL4591917)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of human DDX3X ATPase activity using DDX3 as substrate by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06BJKPubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50537056(CHEMBL4571759)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of human DDX3X ATPase activity using DDX3 as substrate by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06BJKPubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50537057(CHEMBL4551611)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of human DDX3X ATPase activity using DDX3 as substrate by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06BJKPubMed
TargetATP-dependent RNA helicase DDX1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50537058(CHEMBL4531719)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of human DDX1 helicase activityMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06BJKPubMed
TargetATP-dependent RNA helicase DDX3X(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50537058(CHEMBL4531719)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of human DDX3X ATPase activity using DDX3 as substrate by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06BJKPubMed
TargetSolute carrier family 22 member 3(Homo sapiens (Human))
Universidade do Porto

Curated by ChEMBL
LigandPNGBDBM50149890(CHEMBL9324 | tetraethylammonium)copy SMILEScopy InChI
Affinity DataIC50: 1.03E+7nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake (MPP+: 0.2 uM) in OCT3-expressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ702RPubMed