Compile Data Set for Download or QSAR
Found 180 with Last Name = 'pühler' and Initial = 'f'
LigandPNGBDBM218770(US9296757, 92)copy SMILES
Affinity DataIC50: 0.600nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DD7US Patent
LigandPNGBDBM218771(US9296757, 93)copy SMILES
Affinity DataIC50: 0.700nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DD7US Patent
LigandPNGBDBM218766(US9296757, 88)copy SMILES
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DD7US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1 [1-424](Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM227719(3-bromo-n-(6-methoxy-1h-indazol-5-yl)-1h-pyrazolo[...)copy SMILEScopy InChI
Affinity DataIC50: 1nMpH: 7.5Assay Description:TBDA recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accessio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2C53NTHUS Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
BAYER INTELLECTUAL PROPERTY GMBH

US Patent
LigandPNGBDBM333402(2-{[3-(Furo[3,2-c]pyridin-2-yl)imidazo[1,2-b]pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4S1HUS Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1 [1-424](Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM227732(3-bromo-n-(6-isopropoxy-1h-indazol-5-yl)-1h-pyrazo...)copy SMILEScopy InChI
Affinity DataIC50: 1nMpH: 7.5Assay Description:TBDA recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accessio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2C53NTHUS Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
BAYER INTELLECTUAL PROPERTY GMBH

US Patent
LigandPNGBDBM333401(2-{[3-(Furo[2,3-c]pyridin-2-yl)imidazo[1,2-b]pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4S1HUS Patent
LigandPNGBDBM218768(US9296757, 90)copy SMILES
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DD7US Patent
LigandPNGBDBM218767(US9296757, 89)copy SMILES
Affinity DataIC50: 1.90nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DD7US Patent
LigandPNGBDBM218765(US9296757, 87)copy SMILES
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DD7US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
BAYER INTELLECTUAL PROPERTY GMBH

US Patent
LigandPNGBDBM333382(3-[(1R)-1-{[3-(1- Benzofuran-2- yl)imidazo[1,2-b]p...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4S1HUS Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1 [1-424](Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM227719(3-bromo-n-(6-methoxy-1h-indazol-5-yl)-1h-pyrazolo[...)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 7.5Assay Description:TBDA recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accessio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2C53NTHUS Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1 [1-424](Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM227728(3-(4-fluorophenyl)-n-(6-methoxy-1h-indazol-5-yl)-1...)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 7.5Assay Description:TBDA recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accessio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2C53NTHUS Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
BAYER INTELLECTUAL PROPERTY GMBH

US Patent
LigandPNGBDBM333390(2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4S1HUS Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
BAYER INTELLECTUAL PROPERTY GMBH

US Patent
LigandPNGBDBM333403(2-{[3-(4-Methoxyfuro[3,2-c]pyridin-2-yl)imidazo[1,...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4S1HUS Patent
LigandPNGBDBM218764(US9296757, 86)copy SMILES
Affinity DataIC50: 3nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DD7US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1 [1-424](Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM227719(3-bromo-n-(6-methoxy-1h-indazol-5-yl)-1h-pyrazolo[...)copy SMILEScopy InChI
Affinity DataIC50: 3nMpH: 7.5Assay Description:TBDA recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accessio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2C53NTHUS Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
BAYER INTELLECTUAL PROPERTY GMBH

US Patent
LigandPNGBDBM333389(2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4S1HUS Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
BAYER INTELLECTUAL PROPERTY GMBH

US Patent
LigandPNGBDBM333391((−)-2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]p...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4S1HUS Patent
LigandPNGBDBM214639(US9284319, 7)copy SMILEScopy InChI
Affinity DataIC50: 4nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2765D6DUS Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
BAYER INTELLECTUAL PROPERTY GMBH

US Patent
LigandPNGBDBM333388(3-[(1R)-1-Hydroxy-2- {[3-(4-methoxy-1- benzofuran-...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4S1HUS Patent
LigandPNGBDBM218763(US9296757, 85)copy SMILES
Affinity DataIC50: 4nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DD7US Patent
LigandPNGBDBM218709(US9296757, 31)copy SMILES
Affinity DataIC50: 4nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DD7US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
BAYER INTELLECTUAL PROPERTY GMBH

US Patent
LigandPNGBDBM333404(2-{[3-(4-Ethoxyfuro[3,2-c]pyridin-2-yl)imidazo[1,2...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4S1HUS Patent
LigandPNGBDBM214635(US9284319, 3)copy SMILEScopy InChI
Affinity DataIC50: 6nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2765D6DUS Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1 [1-424](Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM227719(3-bromo-n-(6-methoxy-1h-indazol-5-yl)-1h-pyrazolo[...)copy SMILEScopy InChI
Affinity DataIC50: 6nMpH: 7.5Assay Description:TBDA recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accessio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2C53NTHUS Patent
LigandPNGBDBM214633(US9284319, 1)copy SMILEScopy InChI
Affinity DataIC50: 7nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2765D6DUS Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1 [1-424](Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM227721(3-bromo-n-(1h-indazol-5-yl)-1h-pyrazolo[3,4-d]pyri...)copy SMILEScopy InChI
Affinity DataIC50: 8nMpH: 7.5Assay Description:TBDA recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accessio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2C53NTHUS Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1 [1-424](Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM227720(3-bromo-n-(6-fluoro-1h-indazol-5-yl)-1h-pyrazolo[3...)copy SMILEScopy InChI
Affinity DataIC50: 8nMpH: 7.5Assay Description:TBDA recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accessio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2C53NTHUS Patent
LigandPNGBDBM218714(US9296757, 36)copy SMILES
Affinity DataIC50: 9nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DD7US Patent
LigandPNGBDBM218687(US9296757, 9)copy SMILES
Affinity DataIC50: 9nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DD7US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
BAYER INTELLECTUAL PROPERTY GMBH

US Patent
LigandPNGBDBM333384(2-{[3-(1- Benzofuran-2- yl)imidazo[1,2-b]pyridazi...)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4S1HUS Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
BAYER INTELLECTUAL PROPERTY GMBH

US Patent
LigandPNGBDBM333393(1-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6...)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4S1HUS Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
BAYER INTELLECTUAL PROPERTY GMBH

US Patent
LigandPNGBDBM333394(1-{[3-(4-Methoxyfuro[3,2-c]pyridin-2-yl)imidazo[1,...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4S1HUS Patent
LigandPNGBDBM214649(US9284319, R7 | US9730929, Example R7 | US9783543,...)copy SMILEScopy InChI
Affinity DataIC50: 11nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2765D6DUS Patent
LigandPNGBDBM218688(US9296757, 10)copy SMILES
Affinity DataIC50: 11nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8DD7US Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1 [1-424](Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM227720(3-bromo-n-(6-fluoro-1h-indazol-5-yl)-1h-pyrazolo[3...)copy SMILEScopy InChI
Affinity DataIC50: 12nMpH: 7.5Assay Description:TBDA recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accessio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2C53NTHUS Patent
LigandPNGBDBM214638(US9284319, 6)copy SMILEScopy InChI
Affinity DataIC50: 12nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2765D6DUS Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1 [1-424](Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM227727(3-(4-fluorophenyl)-n-(1h-indazol-5-yl)-1h-pyrazolo...)copy SMILEScopy InChI
Affinity DataIC50: 12nMpH: 7.5Assay Description:TBDA recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accessio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2C53NTHUS Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1 [1-424](Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM227729(US9556181, 14 | n-(6-fluoro-1h-indazol-5-yl)-3-(4-...)copy SMILEScopy InChI
Affinity DataIC50: 12nMpH: 7.5Assay Description:TBDA recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accessio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2C53NTHUS Patent
LigandPNGBDBM214637(US9284319, 5)copy SMILEScopy InChI
Affinity DataIC50: 13nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2765D6DUS Patent
LigandPNGBDBM214649(US9284319, R7 | US9730929, Example R7 | US9783543,...)copy SMILEScopy InChI
Affinity DataIC50: 13nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2765D6DUS Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
BAYER INTELLECTUAL PROPERTY GMBH

US Patent
LigandPNGBDBM214649(US9284319, R7 | US9730929, Example R7 | US9783543,...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:A recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accession n...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28S4S1HUS Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1 [1-424](Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM227721(3-bromo-n-(1h-indazol-5-yl)-1h-pyrazolo[3,4-d]pyri...)copy SMILEScopy InChI
Affinity DataIC50: 14nMpH: 7.5Assay Description:TBDA recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accessio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2C53NTHUS Patent
LigandPNGBDBM214639(US9284319, 7)copy SMILEScopy InChI
Affinity DataIC50: 14nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2765D6DUS Patent
TargetMAP kinase-interacting serine/threonine-protein kinase 1 [1-424](Homo sapiens (Human))
BAYER PHARMA AKTIENGESELLSCHAFT

US Patent
LigandPNGBDBM227720(3-bromo-n-(6-fluoro-1h-indazol-5-yl)-1h-pyrazolo[3...)copy SMILEScopy InChI
Affinity DataIC50: 15nMpH: 7.5Assay Description:TBDA recombinant fusion protein of Glutathione-S-Transferase (GST, N-terminally) and human full-length MKNK1 (amino acids 1-424 and T344D of accessio...More data for this Ligand-Target Pair
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BindingDB Entry DOI: 10.7270/Q2C53NTHUS Patent
LigandPNGBDBM214640(US9284319, 8)copy SMILEScopy InChI
Affinity DataIC50: 15nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
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BindingDB Entry DOI: 10.7270/Q2765D6DUS Patent
LigandPNGBDBM214636(US9284319, 4)copy SMILEScopy InChI
Affinity DataIC50: 15nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2765D6DUS Patent
LigandPNGBDBM214641(US9284319, 9)copy SMILEScopy InChI
Affinity DataIC50: 15nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2765D6DUS Patent
LigandPNGBDBM218708(US9296757, 30 | US9296757, 33)copy SMILES
Affinity DataIC50: 15nMpH: 7.5 T: 2°CAssay Description:For the assay 50 nL of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a black low volume 384 well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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BindingDB Entry DOI: 10.7270/Q2XK8DD7US Patent
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