TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 0.260nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 0.350nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membrane homogenatesMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 0.370nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 0.420nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 0.540nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membrane homogenatesMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 0.680nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 0.740nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membrane homogenatesMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 0.790nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membrane homogenatesMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 0.830nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 0.910nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 0.910nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membrane homogenatesMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 0.960nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 2.80nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 4.10nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 4.20nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 4.20nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 8.10nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 61nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 260nMAssay Description:Displacement of [3H]PK11195 from TSPO in rat heart membranes after 15 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
France; Inserm/CEA/Universit£ Paris Sud
Curated by ChEMBL
Affinity DataKi: 920nMAssay Description:Displacement of [3H]-PK11195 from rat heart membrane TSPOMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:"U"-bottomed Falcon plates are prepared by placing 5 uL of solutions of the compounds according to the invention at concentrations of 10, 1, 0.1, 0.0...More data for this Ligand-Target Pair