Compile Data Set for Download or QSAR
Found 289 with Last Name = 'quartieri' and Initial = 'f'
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Nerviano Medical Sciences Srl

LigandPNGBDBM31541(pyrazolo[4,3-h]quinazoline-3-carboxamide, 24)copy SMILEScopy InChI
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzymes and substrates, followed by quantitation of the phosphorylat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3JJPPubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Nerviano Medical Sciences Srl

LigandPNGBDBM31532(pyrazolo[4,3-h]quinazoline-3-carboxamide, 1)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzymes and substrates, followed by quantitation of the phosphorylat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3JJPPubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Nerviano Medical Sciences Srl

LigandPNGBDBM31539(pyrazolo[4,3-h]quinazoline-3-carboxamide, 22)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzymes and substrates, followed by quantitation of the phosphorylat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3JJPPubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Nerviano Medical Sciences Srl

LigandPNGBDBM31532(pyrazolo[4,3-h]quinazoline-3-carboxamide, 1)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of CDK2/Cyclin A assessed as [33P]-gamma-ATP incorporation into substrate by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R211RSPubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Nerviano Medical Sciences Srl

LigandPNGBDBM50318085(1-Methyl-8-[(2-methylphenyl)amino]-4,5-dihydro-1H-...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of CDK2/Cyclin A assessed as [33P]-gamma-ATP incorporation into substrate by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R211RSPubMed
TargetCholine kinase alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50579781(CHEMBL5094847)copy SMILES
Affinity DataIC50: 14nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1PFFPubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Nerviano Medical Sciences Srl

LigandPNGBDBM31542(pyrazolo[4,3-h]quinazoline-3-carboxamide, 25)copy SMILEScopy InChI
Affinity DataIC50: 14nMpH: 7.4 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzymes and substrates, followed by quantitation of the phosphorylat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3JJPPubMed
TargetCholine kinase alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50579779(CHEMBL5091519)copy SMILES
Affinity DataIC50: 14nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1PFFPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Nerviano Medical Sciences srl

Curated by ChEMBL
LigandPNGBDBM50318085(1-Methyl-8-[(2-methylphenyl)amino]-4,5-dihydro-1H-...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of PLK1 assessed as [33P]-gamma-ATP incorporation into substrate by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R211RSPubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Nerviano Medical Sciences Srl

LigandPNGBDBM31544(pyrazolo[4,3-h]quinazoline-3-carboxamide, 27)copy SMILEScopy InChI
Affinity DataIC50: 17nMpH: 7.4 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzymes and substrates, followed by quantitation of the phosphorylat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3JJPPubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Nerviano Medical Sciences Srl

LigandPNGBDBM31533(pyrazolo[4,3-h]quinazoline-3-carboxamide, 16)copy SMILEScopy InChI
Affinity DataIC50: 19nMpH: 7.4 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzymes and substrates, followed by quantitation of the phosphorylat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3JJPPubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Nerviano Medical Sciences Srl

LigandPNGBDBM31533(pyrazolo[4,3-h]quinazoline-3-carboxamide, 16)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of CDK2/Cyclin A assessed as [33P]-gamma-ATP incorporation into substrate by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R211RSPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Nerviano Medical Sciences srl

Curated by ChEMBL
LigandPNGBDBM50349092(CHEMBL1807303)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of MPS1 assessed as [33P]-gamma-ATP incorporation into substrate P38-betatide by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R211RSPubMed
TargetCholine kinase alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50579782(CHEMBL5078600)copy SMILES
Affinity DataIC50: 20nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1PFFPubMed
TargetCholine kinase alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50579773(CHEMBL5079663)copy SMILES
Affinity DataIC50: 20nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1PFFPubMed
TargetCholine kinase alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50579777(CHEMBL5090932)copy SMILES
Affinity DataIC50: 21nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1PFFPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Nerviano Medical Sciences srl

Curated by ChEMBL
LigandPNGBDBM50349094(CHEMBL1807305)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of MPS1 assessed as [33P]-gamma-ATP incorporation into substrate P38-betatide by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R211RSPubMed
TargetCholine kinase alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50579771(CHEMBL5077194)copy SMILES
Affinity DataIC50: 22nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1PFFPubMed
TargetCholine kinase alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50579769(CHEMBL5075042)copy SMILES
Affinity DataIC50: 23nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1PFFPubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Nerviano Medical Sciences Srl

LigandPNGBDBM31543(pyrazolo[4,3-h]quinazoline-3-carboxamide, 26)copy SMILEScopy InChI
Affinity DataIC50: 24nMpH: 7.4 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzymes and substrates, followed by quantitation of the phosphorylat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3JJPPubMed
TargetCholine kinase alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50579780(CHEMBL5089356)copy SMILES
Affinity DataIC50: 27nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1PFFPubMed
TargetCholine kinase alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50579775(CHEMBL5085262)copy SMILES
Affinity DataIC50: 28nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1PFFPubMed
TargetCholine kinase alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50579757(CHEMBL5084844)copy SMILES
Affinity DataIC50: 28nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1PFFPubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Nerviano Medical Sciences Srl

LigandPNGBDBM31549(pyrazolo[4,3-h]quinazoline-3-carboxamide, 32)copy SMILEScopy InChI
Affinity DataIC50: 29nMpH: 7.4 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzymes and substrates, followed by quantitation of the phosphorylat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3JJPPubMed
TargetCholine kinase alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50579770(CHEMBL5090132)copy SMILES
Affinity DataIC50: 29nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1PFFPubMed
TargetAurora kinase A(Homo sapiens (Human))
Nerviano Medical Sciences Srl

LigandPNGBDBM31541(pyrazolo[4,3-h]quinazoline-3-carboxamide, 24)copy SMILEScopy InChI
Affinity DataIC50: 30nMT: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzymes and substrates, followed by quantitation of the phosphorylat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3JJPPubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Nerviano Medical Sciences Srl

LigandPNGBDBM31546(pyrazolo[4,3-h]quinazoline-3-carboxamide, 29)copy SMILEScopy InChI
Affinity DataIC50: 31nMpH: 7.4 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzymes and substrates, followed by quantitation of the phosphorylat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3JJPPubMed
TargetCholine kinase alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50579786(CHEMBL5093152)copy SMILES
Affinity DataIC50: 31nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1PFFPubMed
TargetCholine kinase alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50579785(CHEMBL5075110)copy SMILES
Affinity DataIC50: 31nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1PFFPubMed
TargetCholine kinase alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50579774(CHEMBL5081222)copy SMILES
Affinity DataIC50: 31nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1PFFPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Nerviano Medical Sciences srl

Curated by ChEMBL
LigandPNGBDBM50349103(CHEMBL1808341)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Inhibition of MPS1 assessed as [33P]-gamma-ATP incorporation into substrate P38-betatide by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R211RSPubMed
TargetCholine kinase alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50579772(CHEMBL5088776)copy SMILES
Affinity DataIC50: 33nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1PFFPubMed
TargetCholine kinase alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50579784(CHEMBL5091201)copy SMILES
Affinity DataIC50: 34nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1PFFPubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Nerviano Medical Sciences Srl

LigandPNGBDBM31557(pyrazolo[4,3-h]quinazoline-3-carboxamide, 40)copy SMILEScopy InChI
Affinity DataIC50: 35nMpH: 7.4 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzymes and substrates, followed by quantitation of the phosphorylat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3JJPPubMed
TargetDual specificity protein kinase TTK(Homo sapiens (Human))
Nerviano Medical Sciences srl

Curated by ChEMBL
LigandPNGBDBM50349099(CHEMBL1808338)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Inhibition of MPS1 assessed as [33P]-gamma-ATP incorporation into substrate P38-betatide by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R211RSPubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Nerviano Medical Sciences Srl

LigandPNGBDBM31553(pyrazolo[4,3-h]quinazoline-3-carboxamide, 36)copy SMILEScopy InChI
Affinity DataIC50: 36nMpH: 7.4 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzymes and substrates, followed by quantitation of the phosphorylat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3JJPPubMed
TargetCholine kinase alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50579764(CHEMBL5086885)copy SMILES
Affinity DataIC50: 40nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1PFFPubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Nerviano Medical Sciences srl

Curated by ChEMBL
LigandPNGBDBM50318081(8-[(2-Methoxyphenyl)amino]-1-methyl-4,5-dihydro-1H...)copy SMILEScopy InChI
Affinity DataIC50: 42nMAssay Description:Inhibition of PLK1 assessed as [33P]-gamma-ATP incorporation into substrate by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R211RSPubMed
TargetCholine kinase alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50579778(CHEMBL5078057)copy SMILES
Affinity DataIC50: 43nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1PFFPubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Nerviano Medical Sciences Srl

LigandPNGBDBM31545(Milciclib | pyrazolo[4,3-h]quinazoline-3-carboxami...)copy SMILEScopy InChI
Affinity DataIC50: 45nMpH: 7.4 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzymes and substrates, followed by quantitation of the phosphorylat...More data for this Ligand-Target Pair
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Nerviano Medical Sciences Srl

LigandPNGBDBM31540(pyrazolo[4,3-h]quinazoline-3-carboxamide, 23)copy SMILEScopy InChI
Affinity DataIC50: 45nMpH: 7.4 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzymes and substrates, followed by quantitation of the phosphorylat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3JJPPubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Nerviano Medical Sciences Srl

LigandPNGBDBM31550(pyrazolo[4,3-h]quinazoline-3-carboxamide, 33)copy SMILEScopy InChI
Affinity DataIC50: 47nMpH: 7.4 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzymes and substrates, followed by quantitation of the phosphorylat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3JJPPubMed
TargetCholine kinase alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50579783(CHEMBL5088850)copy SMILES
Affinity DataIC50: 49nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1PFFPubMed
TargetCholine kinase alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50579758(CHEMBL5085127)copy SMILES
Affinity DataIC50: 49nMAssay Description:Inhibition of ChoKalpha (unknown origin) by HTS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1PFFPubMed
TargetAurora kinase A(Homo sapiens (Human))
Nerviano Medical Sciences Srl

LigandPNGBDBM31532(pyrazolo[4,3-h]quinazoline-3-carboxamide, 1)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of Aur-A assessed as [33P]-gamma-ATP incorporation into substrate by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R211RSPubMed
TargetAurora kinase A(Homo sapiens (Human))
Nerviano Medical Sciences Srl

LigandPNGBDBM31532(pyrazolo[4,3-h]quinazoline-3-carboxamide, 1)copy SMILEScopy InChI
Affinity DataIC50: 50nMT: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzymes and substrates, followed by quantitation of the phosphorylat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3JJPPubMed
TargetAurora kinase A(Homo sapiens (Human))
Nerviano Medical Sciences Srl

LigandPNGBDBM31542(pyrazolo[4,3-h]quinazoline-3-carboxamide, 25)copy SMILEScopy InChI
Affinity DataIC50: 51nMT: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzymes and substrates, followed by quantitation of the phosphorylat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3JJPPubMed
TargetAurora kinase A(Homo sapiens (Human))
Nerviano Medical Sciences Srl

LigandPNGBDBM31539(pyrazolo[4,3-h]quinazoline-3-carboxamide, 22)copy SMILEScopy InChI
Affinity DataIC50: 53nMT: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzymes and substrates, followed by quantitation of the phosphorylat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3JJPPubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Nerviano Medical Sciences Srl

LigandPNGBDBM31545(Milciclib | pyrazolo[4,3-h]quinazoline-3-carboxami...)copy SMILEScopy InChI
Affinity DataIC50: 53nMpH: 7.5 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzymes and substrates, followed by quantitation of the phosphorylat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3JJPPubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Nerviano Medical Sciences Srl

LigandPNGBDBM31551(pyrazolo[4,3-h]quinazoline-3-carboxamide, 34)copy SMILEScopy InChI
Affinity DataIC50: 55nMpH: 7.4 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzymes and substrates, followed by quantitation of the phosphorylat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3JJPPubMed
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