Compile Data Set for Download or QSAR
Found 365 with Last Name = 'suzenet' and Initial = 'f'
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50139844(CHEMBL3763503)copy SMILEScopy InChI
Affinity DataKi:  0.0300nMAssay Description:Displacement of [125I]2-Iodomelatonin from human MT2 receptor expressed in HEK293 cells after 120 mins by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC6318PubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50139843(CHEMBL3765540)copy SMILEScopy InChI
Affinity DataKi:  0.0400nMAssay Description:Displacement of [125I]2-Iodomelatonin from human MT1 receptor expressed in HEK293 cells after 120 mins by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC6318PubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50139842(CHEMBL3765401)copy SMILEScopy InChI
Affinity DataKi:  0.0800nMAssay Description:Displacement of [125I]2-Iodomelatonin from human MT2 receptor expressed in HEK293 cells after 120 mins by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC6318PubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50139847(CHEMBL3764765)copy SMILEScopy InChI
Affinity DataKi:  0.0900nMAssay Description:Displacement of [125I]2-Iodomelatonin from human MT2 receptor expressed in HEK293 cells after 120 mins by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC6318PubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50139843(CHEMBL3765540)copy SMILEScopy InChI
Affinity DataKi:  0.140nMAssay Description:Displacement of [125I]2-Iodomelatonin from human MT2 receptor expressed in HEK293 cells after 120 mins by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC6318PubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50037242(CHEMBL323332 | N-(2-(5-methoxybenzofuran-3-yl)ethy...)copy SMILEScopy InChI
Affinity DataKi:  0.150nMAssay Description:Displacement of [125I]2-Iodomelatonin from human MT1 receptor expressed in HEK293 cells after 120 mins by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC6318PubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50139844(CHEMBL3763503)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]2-Iodomelatonin from human MT1 receptor expressed in HEK293 cells after 120 mins by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC6318PubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50139842(CHEMBL3765401)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]2-Iodomelatonin from human MT1 receptor expressed in HEK293 cells after 120 mins by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC6318PubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50340329(4-azamelatonin | CHEMBL1760944)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1JWMPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50513620(CHEMBL4563574)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in Wistar rat brain membrane incubated for 3 hrs by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49V3XPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50340329(4-azamelatonin | CHEMBL1760944)copy SMILEScopy InChI
Affinity DataKi:  0.240nMAssay Description:Displacement of [125I]2-Iodomelatonin from human MT1 receptor expressed in HEK293 cells after 120 mins by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC6318PubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)copy SMILEScopy InChI
Affinity DataKi:  0.25nMAssay Description:Displacement of [125I]2-Iodomelatonin from human MT1 receptor expressed in HEK293 cells after 120 mins by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC6318PubMedDrugBank
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)copy SMILEScopy InChI
Affinity DataKi:  0.25nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1JWMPubMedDrugBank
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50340324(CHEMBL1760946 | N-(2-(6-Methoxy-1H-pyrrolo[2,3-b]p...)copy SMILEScopy InChI
Affinity DataKi:  0.280nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1JWMPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50340329(4-azamelatonin | CHEMBL1760944)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1JWMPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50340338(CHEMBL1760947 | N-(2-(6-Methoxy-1H-pyrrolo[2,3-b]p...)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1JWMPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50513605(CHEMBL4563839)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in Wistar rat brain membrane incubated for 3 hrs by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49V3XPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50513617(CHEMBL4459802)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in Wistar rat brain membrane incubated for 3 hrs by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49V3XPubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50307501((6S)-N,N-dipropyl-5,6,7,8-tetrahydro-1,1'-binaphth...)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]5CT from human cloned 5HT7B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S182M1PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50513594(CHEMBL4556722)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in Wistar rat brain membrane incubated for 3 hrs by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49V3XPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50513583(CHEMBL4533685)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in Wistar rat brain membrane incubated for 3 hrs by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49V3XPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)copy SMILEScopy InChI
Affinity DataKi:  0.340nMAssay Description:Displacement of [125I]2-Iodomelatonin from human MT2 receptor expressed in HEK293 cells after 120 mins by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC6318PubMedDrugBank
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)copy SMILEScopy InChI
Affinity DataKi:  0.340nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1JWMPubMedDrugBank
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50037242(CHEMBL323332 | N-(2-(5-methoxybenzofuran-3-yl)ethy...)copy SMILEScopy InChI
Affinity DataKi:  0.340nMAssay Description:Displacement of [125I]2-Iodomelatonin from human MT2 receptor expressed in HEK293 cells after 120 mins by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC6318PubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50340329(4-azamelatonin | CHEMBL1760944)copy SMILEScopy InChI
Affinity DataKi:  0.360nMAssay Description:Displacement of [125I]2-Iodomelatonin from human MT2 receptor expressed in HEK293 cells after 120 mins by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC6318PubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50340325(CHEMBL1760945 | N-(2-(6-Methoxy-1H-pyrrolo[2,3-b]p...)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1JWMPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50513613(CHEMBL4567300)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in Wistar rat brain membrane incubated for 3 hrs by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49V3XPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50340327(CHEMBL1760957 | N-(2-(5,6,7,8-Tetrahydro-2-methoxy...)copy SMILEScopy InChI
Affinity DataKi:  0.680nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1JWMPubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50139351(2-(6-cyclohexylpyridin-2-ylthio)-N,N-dimethylethan...)copy SMILEScopy InChI
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]5CT from human cloned 5HT7B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S182M1PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50513577(CHEMBL4445961)copy SMILEScopy InChI
Affinity DataKi:  0.700nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in Wistar rat brain membrane incubated for 3 hrs by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49V3XPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50513611(CHEMBL4452867)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in Wistar rat brain membrane incubated for 3 hrs by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49V3XPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50513606(CHEMBL4547917)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in Wistar rat brain membrane incubated for 3 hrs by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49V3XPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50139841(CHEMBL3763281)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Displacement of [125I]2-Iodomelatonin from human MT2 receptor expressed in HEK293 cells after 120 mins by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC6318PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50500420(CHEMBL3746010)copy SMILEScopy InChI
Affinity DataKi:  1.30nMAssay Description:Displacement of [125I]alpha-bungarotoxin from alpha7 nAchR in rat frontal corticesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TF01CWPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50340338(CHEMBL1760947 | N-(2-(6-Methoxy-1H-pyrrolo[2,3-b]p...)copy SMILEScopy InChI
Affinity DataKi:  1.30nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1JWMPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50139846(CHEMBL3764879)copy SMILEScopy InChI
Affinity DataKi:  1.30nMAssay Description:Displacement of [125I]2-Iodomelatonin from human MT2 receptor expressed in HEK293 cells after 120 mins by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC6318PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50513579(CHEMBL4534225)copy SMILEScopy InChI
Affinity DataKi:  1.40nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in Wistar rat brain membrane incubated for 3 hrs by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49V3XPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50340325(CHEMBL1760945 | N-(2-(6-Methoxy-1H-pyrrolo[2,3-b]p...)copy SMILEScopy InChI
Affinity DataKi:  1.40nMAssay Description:Displacement of 2-[125I]-iodomelatonin from human MT1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1JWMPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50513616(CHEMBL4532801)copy SMILEScopy InChI
Affinity DataKi:  1.40nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in Wistar rat brain membrane incubated for 3 hrs by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49V3XPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50513592(CHEMBL4517968)copy SMILEScopy InChI
Affinity DataKi:  1.5nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in Wistar rat brain membrane incubated for 3 hrs by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49V3XPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50513585(CHEMBL4467924)copy SMILEScopy InChI
Affinity DataKi:  1.5nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in Wistar rat brain membrane incubated for 3 hrs by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49V3XPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50139841(CHEMBL3763281)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Displacement of [125I]2-Iodomelatonin from human MT1 receptor expressed in HEK293 cells after 120 mins by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC6318PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50513584(CHEMBL4583910)copy SMILEScopy InChI
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in Wistar rat brain membrane incubated for 3 hrs by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49V3XPubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50426657(CHEMBL2326199)copy SMILEScopy InChI
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]2-Iodomelatonin from human MT2 receptor expressed in HEK293 cells after 120 mins by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC6318PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50513588(CHEMBL4582749)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in Wistar rat brain membrane incubated for 3 hrs by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49V3XPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50139847(CHEMBL3764765)copy SMILEScopy InChI
Affinity DataKi:  2.20nMAssay Description:Displacement of [125I]2-Iodomelatonin from human MT1 receptor expressed in HEK293 cells after 120 mins by radioligand competition assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC6318PubMed
TargetAmyloid-beta precursor protein [1-42](Homo sapiens (Human))
CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE; UNIVERSITE D''ORLEANS; UNIVERSITE DE TOURS; CENTRE HOSPITALIER REGIONAL UNIVERSITAIRE DE TOURS; INSERM (INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE)

US Patent
LigandPNGBDBM50492518(Florbetapir | US10906900, AV45)copy SMILEScopy InChI
Affinity DataKi:  2.20nMAssay Description:Table 5: Fresh solutions of the test compounds (2.5 mM in DMSO) are diluted in PBS pH7.4, at concentrations between 0.5 nM and 5 μM in the prese...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2BC42NCUS Patent
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50500406(CHEMBL3746146)copy SMILEScopy InChI
Affinity DataKi:  2.30nMAssay Description:Displacement of [125I]alpha-bungarotoxin from alpha7 nAchR in rat frontal corticesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TF01CWPubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50150684((R)-8-(2,6-dimethoxyphenyl)-N,N-dimethylchroman-3-...)copy SMILEScopy InChI
Affinity DataKi:  2.55nMAssay Description:Displacement of [3H]5CT from human cloned 5HT7B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S182M1PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£ d'Orl£ans

Curated by ChEMBL
LigandPNGBDBM50513604(CHEMBL4441856)copy SMILEScopy InChI
Affinity DataKi:  2.80nMAssay Description:Displacement of [125I]-alpha-bungarotoxin from alpha7 nAChR in Wistar rat brain membrane incubated for 3 hrs by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49V3XPubMed
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