Compile Data Set for Download or QSAR
Found 48 with Last Name = 'takayama' and Initial = 'f'
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Nagoya University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50420185(CHEMBL1233636)copy SMILEScopy InChI
Affinity DataKi:  2.27E+4nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake (PAH: 5 uM, indoxyl sulfate:500 uM) in S2 human-OAT1 expressing cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23R0V48PubMed
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Nagoya University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50420185(CHEMBL1233636)copy SMILEScopy InChI
Affinity DataKi:  2.30E+4nMAssay Description:TP_TRANSPORTER: uptake&inhibition of PAH in OAT1-S2 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23R0V48PubMed
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Nagoya University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50420185(CHEMBL1233636)copy SMILEScopy InChI
Affinity DataKi:  1.69E+5nMAssay Description:TP_TRANSPORTER: inhibition of E1S uptake (E1S: 5 uM, indoxyl sulfate:500 uM) in S2 cells expressing human-OAT3More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23R0V48PubMed
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Nagoya University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50420185(CHEMBL1233636)copy SMILEScopy InChI
Affinity DataKi:  1.69E+5nMAssay Description:TP_TRANSPORTER: uptake&inhibition of estrone sulfate in OAT3-S2 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23R0V48PubMed
TargetSolute carrier family 22 member 11(Homo sapiens (Human))
Nagoya University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50420185(CHEMBL1233636)copy SMILEScopy InChI
Affinity DataKi:  1.81E+5nMAssay Description:TP_TRANSPORTER: uptake&inhibition of estrone sulfate in OAT4-S2 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23R0V48PubMed
TargetSolute carrier family 22 member 11(Homo sapiens (Human))
Nagoya University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50420185(CHEMBL1233636)copy SMILEScopy InChI
Affinity DataKi:  1.81E+5nMAssay Description:TP_TRANSPORTER: inhibition of E1S uptake (E1S: 5 uM, indoxyl sulfate:500 uM) in S2 cells expressing human-OAT4More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23R0V48PubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344337(CHEMBL1779478 | rac-2-(3-((4-(Benzyloxy)benzamido)...)copy SMILEScopy InChI
Affinity DataEC50:  52nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344338(CHEMBL1779479 | rac-2-(4-Methoxy-3-((4-phenethoxyb...)copy SMILEScopy InChI
Affinity DataEC50:  60nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344339(CHEMBL1779476 | rac-2-(4-Methoxy-3-((3-phenylbenza...)copy SMILEScopy InChI
Affinity DataEC50:  74nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344340(CHEMBL255392 | rac-2-(3-(4-Methylbenzamidomethyl)-...)copy SMILEScopy InChI
Affinity DataEC50:  100nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344333(CHEMBL1779473 | rac-2-(4-Methoxy-3-((4-(trifluorom...)copy SMILEScopy InChI
Affinity DataEC50:  110nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344332(2-(4-methoxy-3-((4-phenoxybenzamido)methyl)benzyl)...)copy SMILEScopy InChI
Affinity DataEC50:  120nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344331(CHEMBL270587 | rac-2-(3-{[(biphenyl-4-carbonyl)-am...)copy SMILEScopy InChI
Affinity DataEC50:  210nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344330((S)-2-(3-((4-(4-Fluorophenoxy)benzamido)methyl)-4-...)copy SMILEScopy InChI
Affinity DataEC50:  300nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344331(CHEMBL270587 | rac-2-(3-{[(biphenyl-4-carbonyl)-am...)copy SMILEScopy InChI
Affinity DataEC50:  340nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344340(CHEMBL255392 | rac-2-(3-(4-Methylbenzamidomethyl)-...)copy SMILEScopy InChI
Affinity DataEC50:  360nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344337(CHEMBL1779478 | rac-2-(3-((4-(Benzyloxy)benzamido)...)copy SMILEScopy InChI
Affinity DataEC50:  460nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344334((S)-2-(3-((4-(4-Chlorophenoxy)benzamido)methyl)-4-...)copy SMILEScopy InChI
Affinity DataEC50:  580nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344339(CHEMBL1779476 | rac-2-(4-Methoxy-3-((3-phenylbenza...)copy SMILEScopy InChI
Affinity DataEC50:  710nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344338(CHEMBL1779479 | rac-2-(4-Methoxy-3-((4-phenethoxyb...)copy SMILEScopy InChI
Affinity DataEC50:  780nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344335((S)-2-(3-((4-(4-bromophenoxy)benzamido)methyl)-4-m...)copy SMILEScopy InChI
Affinity DataEC50:  800nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344332(2-(4-methoxy-3-((4-phenoxybenzamido)methyl)benzyl)...)copy SMILEScopy InChI
Affinity DataEC50:  820nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344334((S)-2-(3-((4-(4-Chlorophenoxy)benzamido)methyl)-4-...)copy SMILEScopy InChI
Affinity DataEC50:  830nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344330((S)-2-(3-((4-(4-Fluorophenoxy)benzamido)methyl)-4-...)copy SMILEScopy InChI
Affinity DataEC50:  920nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344335((S)-2-(3-((4-(4-bromophenoxy)benzamido)methyl)-4-m...)copy SMILEScopy InChI
Affinity DataEC50:  990nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344337(CHEMBL1779478 | rac-2-(3-((4-(Benzyloxy)benzamido)...)copy SMILEScopy InChI
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344338(CHEMBL1779479 | rac-2-(4-Methoxy-3-((4-phenethoxyb...)copy SMILEScopy InChI
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344341(CHEMBL255593 | rac-2-(3-(benzamidomethyl)-4-methox...)copy SMILEScopy InChI
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344342(CHEMBL1779475 | rac-2-(4-Methoxy-3-((2-phenoxybenz...)copy SMILEScopy InChI
Affinity DataEC50:  3.60E+3nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344343(CHEMBL1779477 | rac-2-(4-Methoxy-3-((2-phenylbenza...)copy SMILEScopy InChI
Affinity DataEC50:  3.60E+3nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344339(CHEMBL1779476 | rac-2-(4-Methoxy-3-((3-phenylbenza...)copy SMILEScopy InChI
Affinity DataEC50:  4.10E+3nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344333(CHEMBL1779473 | rac-2-(4-Methoxy-3-((4-(trifluorom...)copy SMILEScopy InChI
Affinity DataEC50:  4.40E+3nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344336(CHEMBL1779474 | rac-2-(4-Methoxy-3-((3-phenoxybenz...)copy SMILEScopy InChI
Affinity DataEC50:  4.60E+3nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344336(CHEMBL1779474 | rac-2-(4-Methoxy-3-((3-phenoxybenz...)copy SMILEScopy InChI
Affinity DataEC50:  4.80E+3nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344341(CHEMBL255593 | rac-2-(3-(benzamidomethyl)-4-methox...)copy SMILEScopy InChI
Affinity DataEC50:  8.10E+3nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344340(CHEMBL255392 | rac-2-(3-(4-Methylbenzamidomethyl)-...)copy SMILEScopy InChI
Affinity DataEC50:  9.60E+3nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344342(CHEMBL1779475 | rac-2-(4-Methoxy-3-((2-phenoxybenz...)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344343(CHEMBL1779477 | rac-2-(4-Methoxy-3-((2-phenylbenza...)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344341(CHEMBL255593 | rac-2-(3-(benzamidomethyl)-4-methox...)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344342(CHEMBL1779475 | rac-2-(4-Methoxy-3-((2-phenoxybenz...)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344343(CHEMBL1779477 | rac-2-(4-Methoxy-3-((2-phenylbenza...)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344336(CHEMBL1779474 | rac-2-(4-Methoxy-3-((3-phenoxybenz...)copy SMILEScopy InChI
Affinity DataEC50:  41nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344335((S)-2-(3-((4-(4-bromophenoxy)benzamido)methyl)-4-m...)copy SMILEScopy InChI
Affinity DataEC50:  29nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344334((S)-2-(3-((4-(4-Chlorophenoxy)benzamido)methyl)-4-...)copy SMILEScopy InChI
Affinity DataEC50:  15nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344333(CHEMBL1779473 | rac-2-(4-Methoxy-3-((4-(trifluorom...)copy SMILEScopy InChI
Affinity DataEC50:  12nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344332(2-(4-methoxy-3-((4-phenoxybenzamido)methyl)benzyl)...)copy SMILEScopy InChI
Affinity DataEC50:  8.80nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344330((S)-2-(3-((4-(4-Fluorophenoxy)benzamido)methyl)-4-...)copy SMILEScopy InChI
Affinity DataEC50:  5nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50344331(CHEMBL270587 | rac-2-(3-{[(biphenyl-4-carbonyl)-am...)copy SMILEScopy InChI
Affinity DataEC50:  7.60nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GNCPubMed