TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Nagoya University School of Medicine
Curated by ChEMBL
Nagoya University School of Medicine
Curated by ChEMBL
Affinity DataKi: 2.27E+4nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake (PAH: 5 uM, indoxyl sulfate:500 uM) in S2 human-OAT1 expressing cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Homo sapiens (Human))
Nagoya University School of Medicine
Curated by ChEMBL
Nagoya University School of Medicine
Curated by ChEMBL
Affinity DataKi: 2.30E+4nMAssay Description:TP_TRANSPORTER: uptake&inhibition of PAH in OAT1-S2 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Nagoya University School of Medicine
Curated by ChEMBL
Nagoya University School of Medicine
Curated by ChEMBL
Affinity DataKi: 1.69E+5nMAssay Description:TP_TRANSPORTER: inhibition of E1S uptake (E1S: 5 uM, indoxyl sulfate:500 uM) in S2 cells expressing human-OAT3More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 8(Homo sapiens (Human))
Nagoya University School of Medicine
Curated by ChEMBL
Nagoya University School of Medicine
Curated by ChEMBL
Affinity DataKi: 1.69E+5nMAssay Description:TP_TRANSPORTER: uptake&inhibition of estrone sulfate in OAT3-S2 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 11(Homo sapiens (Human))
Nagoya University School of Medicine
Curated by ChEMBL
Nagoya University School of Medicine
Curated by ChEMBL
Affinity DataKi: 1.81E+5nMAssay Description:TP_TRANSPORTER: uptake&inhibition of estrone sulfate in OAT4-S2 cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 11(Homo sapiens (Human))
Nagoya University School of Medicine
Curated by ChEMBL
Nagoya University School of Medicine
Curated by ChEMBL
Affinity DataKi: 1.81E+5nMAssay Description:TP_TRANSPORTER: inhibition of E1S uptake (E1S: 5 uM, indoxyl sulfate:500 uM) in S2 cells expressing human-OAT4More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 52nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 60nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 74nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 100nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 110nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 210nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 300nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 340nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 360nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 460nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 580nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 710nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 780nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 800nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 820nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 830nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 920nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 990nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 1.40E+3nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 1.40E+3nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 1.70E+3nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 3.60E+3nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 3.60E+3nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 4.10E+3nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 4.40E+3nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 4.60E+3nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 4.80E+3nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 8.10E+3nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 9.60E+3nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fussed PPARdelta expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fussed PPARgamma expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 41nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 29nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 15nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 8.80nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 5nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataEC50: 7.60nMAssay Description:Agonist activity at Gal4-fussed PPARalpha expressed in human HEK293 cells by reporter gene assayMore data for this Ligand-Target Pair