Compile Data Set for Download or QSAR
Found 72 with Last Name = 'kull' and Initial = 'fc'
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040317(CHEMBL262756 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)copy SMILEScopy InChI
Affinity DataIC50: 0.00100nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040307(1-naphthyl(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Ph...)copy SMILEScopy InChI
Affinity DataIC50: 0.00100nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040299(CHEMBL410783 | cyclopropylbenzene(CO)His-Trp-Ala-V...)copy SMILEScopy InChI
Affinity DataIC50: 0.0300nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040325(CHEMBL268386 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)copy SMILEScopy InChI
Affinity DataIC50: 0.0380nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040299(CHEMBL410783 | cyclopropylbenzene(CO)His-Trp-Ala-V...)copy SMILEScopy InChI
Affinity DataIC50: 0.0490nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040307(1-naphthyl(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Ph...)copy SMILEScopy InChI
Affinity DataIC50: 0.0500nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040301(4-OHPhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)copy SMILEScopy InChI
Affinity DataIC50: 0.0500nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040312(2-tetrahydronaphthyl(CO)His-Trp-Ala-Val-DAla-His-D...)copy SMILEScopy InChI
Affinity DataIC50: 0.0790nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040308(2-aminoPhCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040310(3-CF3PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi...)copy SMILEScopy InChI
Affinity DataIC50: 0.160nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040315((CH3)2PhC(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Phe...)copy SMILEScopy InChI
Affinity DataIC50: 0.180nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040315((CH3)2PhC(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Phe...)copy SMILEScopy InChI
Affinity DataIC50: 0.180nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040317(CHEMBL262756 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)copy SMILEScopy InChI
Affinity DataIC50: 0.220nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040301(4-OHPhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)copy SMILEScopy InChI
Affinity DataIC50: 0.230nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040312(2-tetrahydronaphthyl(CO)His-Trp-Ala-Val-DAla-His-D...)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040320(CHEMBL264122 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)copy SMILEScopy InChI
Affinity DataIC50: 0.330nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50407275(CHEMBL2112786)copy SMILEScopy InChI
Affinity DataIC50: 0.490nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040316(3-isoquinolyl(CO)His-Trp-Ala-Val-DAla-His-DPro(psi...)copy SMILEScopy InChI
Affinity DataIC50: 0.570nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040324(CHEMBL266516 | PhCH2CH2(CO)His-(BzthAla)-Ala-Val-D...)copy SMILEScopy InChI
Affinity DataIC50: 0.75nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040310(3-CF3PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50407276(CHEMBL2111952)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50407276(CHEMBL2111952)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50407273(CHEMBL2111953)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040314((CH3)2PhCCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50407273(CHEMBL2111953)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040323(CHEMBL265736 | phenothiazoneCH2CH2(CO)His-Trp-Ala-...)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040308(2-aminoPhCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040298(CHEMBL386478 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50407277(CHEMBL2112785)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50407277(CHEMBL2112785)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040319(4-CF3PhCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Ph...)copy SMILEScopy InChI
Affinity DataIC50: 3.70nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040298(CHEMBL386478 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040304(CHEMBL267943 | PhCH2CH2(CO)ThiAla-Trp-Ala-Val-DAla...)copy SMILEScopy InChI
Affinity DataIC50: 5.60nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040304(CHEMBL267943 | PhCH2CH2(CO)ThiAla-Trp-Ala-Val-DAla...)copy SMILEScopy InChI
Affinity DataIC50: 5.60nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040321(CHEMBL385805 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)copy SMILEScopy InChI
Affinity DataIC50: 7.30nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040321(CHEMBL385805 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)copy SMILEScopy InChI
Affinity DataIC50: 7.30nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50453525(CHEMBL2370862)copy SMILEScopy InChI
Affinity DataIC50: 7.70nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040305(3-CF3PhCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Ph...)copy SMILEScopy InChI
Affinity DataIC50: 8.40nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040314((CH3)2PhCCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040306(2-CF3PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040302(CHEMBL415455 | PhCH2CH2(CO)His-Trp-Ala-Val-Sar-His...)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040302(CHEMBL415455 | PhCH2CH2(CO)His-Trp-Ala-Val-Sar-His...)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM32362(5-[[3-methoxy-4-[(4-methoxyphenyl)methoxy]phenyl]m...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant human GST-tagged CFMS kinase catalytic domain using biotin-EAIYAPFAKKK-NH2 as substrate after 40 mins by NXT scintillation ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC32TBPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50407274(CHEMBL2111954)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50407274(CHEMBL2111954)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]-Gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040303(CHEMBL383984 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)copy SMILEScopy InChI
Affinity DataIC50: 140nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040303(CHEMBL383984 | PhCH2CH2(CO)His-Trp-Ala-Val-DAla-Hi...)copy SMILEScopy InChI
Affinity DataIC50: 140nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetGastrin-releasing peptide receptor(MOUSE)
Burroughs Wellcome Company

Curated by ChEMBL
LigandPNGBDBM50040318(CHEMBL386476 | PhCH2CH2(CO)His-Trp-Ala-(psi)Val-DA...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]-gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ST7NXNPubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM32362(5-[[3-methoxy-4-[(4-methoxyphenyl)methoxy]phenyl]m...)copy SMILEScopy InChI
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of recombinant human His-tagged B-RAF after 60 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC32TBPubMed
TargetProto-oncogene tyrosine-protein kinase LCK(Mus musculus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM32362(5-[[3-methoxy-4-[(4-methoxyphenyl)methoxy]phenyl]m...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mouse LCKMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC32TBPubMed
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