Compile Data Set for Download or QSAR
Found 156 with Last Name = 'kwarcinski' and Initial = 'fe'
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50119568(CHEMBL3617738)copy SMILEScopy InChI
Affinity DataKi:  70nMAssay Description:Inhibition of c-Src (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TTZPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50119569(CHEMBL3617733)copy SMILEScopy InChI
Affinity DataKi:  90nMAssay Description:Inhibition of c-Src (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TTZPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50119569(CHEMBL3617733)copy SMILEScopy InChI
Affinity DataKi:  120nMAssay Description:Inhibition of c-Src C277S, C483S, S496S mutant (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TTZPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50119567(CHEMBL3617740)copy SMILEScopy InChI
Affinity DataKi:  130nMAssay Description:Inhibition of c-Src (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TTZPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50119578(CHEMBL3617734)copy SMILEScopy InChI
Affinity DataKi:  140nMAssay Description:Inhibition of c-Src (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TTZPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50119570(CHEMBL3617731)copy SMILEScopy InChI
Affinity DataKi:  200nMAssay Description:Inhibition of c-Src C277S, C483S, S496S mutant (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TTZPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50119576(CHEMBL3617736)copy SMILEScopy InChI
Affinity DataKi:  230nMAssay Description:Inhibition of c-Src (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TTZPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50119568(CHEMBL3617738)copy SMILEScopy InChI
Affinity DataKi:  260nMAssay Description:Inhibition of c-Src E280G mutant (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TTZPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50119575(CHEMBL3617737)copy SMILEScopy InChI
Affinity DataKi:  330nMAssay Description:Inhibition of c-Src (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TTZPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50119579(CHEMBL3617730)copy SMILEScopy InChI
Affinity DataKi:  360nMAssay Description:Inhibition of c-Src (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TTZPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50119574(CHEMBL3617739)copy SMILEScopy InChI
Affinity DataKi:  370nMAssay Description:Inhibition of c-Src (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TTZPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50119566(CHEMBL3617732)copy SMILEScopy InChI
Affinity DataKi:  400nMAssay Description:Inhibition of c-Src (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TTZPubMed
TargetTyrosine-protein kinase Yes(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50119566(CHEMBL3617732)copy SMILEScopy InChI
Affinity DataKi:  470nMAssay Description:Inhibition of c-Yes (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TTZPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50119577(CHEMBL3617735)copy SMILEScopy InChI
Affinity DataKi:  480nMAssay Description:Inhibition of c-Src (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TTZPubMed
TargetTyrosine-protein kinase Yes(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50119568(CHEMBL3617738)copy SMILEScopy InChI
Affinity DataKi:  610nMAssay Description:Inhibition of c-Yes (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TTZPubMed
TargetTyrosine-protein kinase HCK(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50119568(CHEMBL3617738)copy SMILEScopy InChI
Affinity DataKi:  730nMAssay Description:Inhibition of Hck (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TTZPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50119568(CHEMBL3617738)copy SMILEScopy InChI
Affinity DataKi:  730nMAssay Description:Inhibition of c-Abl (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TTZPubMed
TargetTyrosine-protein kinase Yes(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50119567(CHEMBL3617740)copy SMILEScopy InChI
Affinity DataKi:  800nMAssay Description:Inhibition of c-Yes (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TTZPubMed
TargetTyrosine-protein kinase HCK(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50119566(CHEMBL3617732)copy SMILEScopy InChI
Affinity DataKi:  980nMAssay Description:Inhibition of Hck (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TTZPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50119566(CHEMBL3617732)copy SMILEScopy InChI
Affinity DataKi:  980nMAssay Description:Inhibition of c-Abl (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TTZPubMed
TargetTyrosine-protein kinase HCK(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50119567(CHEMBL3617740)copy SMILEScopy InChI
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of Hck (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TTZPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50119567(CHEMBL3617740)copy SMILEScopy InChI
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of c-Abl (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TTZPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50119571(CHEMBL3617729)copy SMILEScopy InChI
Affinity DataKi:  1.60E+5nMAssay Description:Inhibition of c-Src C277S, C483S, S496S mutant (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TTZPubMed
TargetTyrosine-protein kinase HCK(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50119571(CHEMBL3617729)copy SMILEScopy InChI
Affinity DataKi: >1.25E+6nMAssay Description:Inhibition of Hck (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TTZPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50119571(CHEMBL3617729)copy SMILEScopy InChI
Affinity DataKi: >1.25E+6nMAssay Description:Inhibition of c-Abl (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2833TTZPubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559236(CHEMBL4796519)copy SMILES
Affinity DataIC50: 7nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559235(CHEMBL4760126)copy SMILES
Affinity DataIC50: 13nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559233(CHEMBL4753926)copy SMILES
Affinity DataIC50: 14nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559225(CHEMBL4763132)copy SMILES
Affinity DataIC50: 18nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50354565(CHEMBL1836719)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50354559(CHEMBL1836724)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559226(CHEMBL4754748)copy SMILES
Affinity DataIC50: 27nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559243(CHEMBL4794509)copy SMILES
Affinity DataIC50: 28nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559224(CHEMBL4788024)copy SMILES
Affinity DataIC50: 33nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559222(CHEMBL4752776)copy SMILES
Affinity DataIC50: 34nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559222(CHEMBL4752776)copy SMILES
Affinity DataIC50: 34nMAssay Description:Inhibition of human STK17B in presence of ATP at Km levelMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50354540(CHEMBL1836717)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559237(CHEMBL4747753)copy SMILES
Affinity DataIC50: 35nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559232(CHEMBL4740090)copy SMILES
Affinity DataIC50: 37nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50354541(CHEMBL1836714)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559230(CHEMBL4783516)copy SMILES
Affinity DataIC50: 40nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559244(CHEMBL4753625)copy SMILES
Affinity DataIC50: 41nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559229(CHEMBL4745018)copy SMILES
Affinity DataIC50: 49nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559247(CHEMBL4789685)copy SMILES
Affinity DataIC50: 49nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559245(CHEMBL4740604)copy SMILES
Affinity DataIC50: 49nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559242(CHEMBL4748440)copy SMILES
Affinity DataIC50: 59nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559228(CHEMBL4788886)copy SMILES
Affinity DataIC50: 60nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559241(CHEMBL4739879)copy SMILES
Affinity DataIC50: 62nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559231(CHEMBL4792541)copy SMILES
Affinity DataIC50: 63nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
TargetSerine/threonine-protein kinase 17B(Homo sapiens (Human))TBA
LigandPNGBDBM50559227(CHEMBL4748561)copy SMILES
Affinity DataIC50: 74nMAssay Description:Inhibition of N-terminal His-tagged STK17B kinase domain (25 to 329 residues) (unknown origin) expressed in Escherichia coli incubated for 90 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB85J2PubMed
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