TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10nMAssay Description:Inhibition of human FPP synthase expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails
Article
BindingDB Entry DOI: 10.7270/Q2F76CD8PubMedDrugBank
MMDB
PDB
3D Structure (crystal)
BindingDB Entry DOI: 10.7270/Q2F76CD8PubMedDrugBank
MMDB
PDB
3D Structure (crystal)
Affinity DataIC50: 9.03nMAssay Description:Inhibition of human FPP synthase expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
Affinity DataIC50: 16.1nMAssay Description:Inhibition of human FPP synthase expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Ability to inhibit binding of [3H]WIN-35428 to dopamine transporter in rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
Affinity DataIC50: 28.1nMAssay Description:Inhibition of human FPP synthase expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Ability to inhibit binding of [3H]WIN-35428 to dopamine transporter in rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 89nMAssay Description:Ability to inhibit binding of [3H]WIN-35428 to dopamine transporter in rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 95nMAssay Description:Ability to inhibit binding of [3H]WIN-35428 to dopamine transporter in rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 118nMAssay Description:Ability to inhibit binding of [3H]WIN-35428 to dopamine transporter in rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 118nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 276nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
Affinity DataIC50: 388nMAssay Description:Inhibition of human FPP synthase expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 650nMAssay Description:Ability to inhibit binding of [3H]WIN-35428 to dopamine transporter in rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 750nMAssay Description:Ability to inhibit binding of [3H]WIN-35428 to dopamine transporter in rat caudate putamenMore data for this Ligand-Target Pair
Affinity DataIC50: 883nMAssay Description:Inhibition of human FPP synthase expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.13E+3nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Ability to inhibit binding of [3H]WIN-35428 to dopamine transporter in rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
Affinity DataIC50: 3.07E+3nMAssay Description:Inhibition of human FPP synthase expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 4.50E+3nMAssay Description:Displacement of [3H]WIN-35428 from Dopamine transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Ability to inhibit binding of [3H]WIN-35428 to dopamine transporter in rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Ability to inhibit binding of [3H]paroxetine to Serotonin transporter in rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Ability to inhibit binding of [3H]paroxetine to Serotonin transporter in rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Ability to inhibit binding of [3H]paroxetine to Serotonin transporter in rat caudate putamenMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Universit£ di Ferrara
Curated by ChEMBL
Universit£ di Ferrara
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Ability to inhibit binding of [3H]paroxetine to Serotonin transporter in rat caudate putamenMore data for this Ligand-Target Pair