Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]-raclopride from human D2 receptor expressed in HEK cells incubated for 1 hr by Cheng-Prusoff analysis based microbeta scintillat...More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]-raclopride from recombinant human D2 receptor expressed in HEK293 cells measured after 1 hr by microbeta scintillation counting ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 2.80nMAssay Description:Displacement of [3H]-ketanserin from recombinant human 5HT2A receptor expressed in HEK293 cells measured after 1.5 hrs by microbeta scintillation cou...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 2.80nMAssay Description:Displacement of [3H]ketanserin from human 5HT2A receptor expressed in HEK293 cells incubated for 1.5 hrs by Cheng-Prusoff analysis based microbeta sc...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 3.60nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Displacement of [3H]-raclopride from human D2 receptor expressed in HEK cells incubated for 1 hr by Cheng-Prusoff analysis based microbeta scintillat...More data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Displacement of [3H]-raclopride from recombinant human D2 receptor expressed in HEK293 cells measured after 1 hr by microbeta scintillation counting ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:Displacement of [3H]-ketanserin from recombinant human 5HT2A receptor expressed in HEK293 cells measured after 1.5 hrs by microbeta scintillation cou...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:Displacement of [3H]ketanserin from human 5HT2A receptor expressed in HEK293 cells incubated for 1.5 hrs by Cheng-Prusoff analysis based microbeta sc...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 4.80nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Displacement of [3H]-LSD from recombinant human 5HT6 receptor expressed in HEK293 cells measured after 1 hr by microbeta scintillation counting analy...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Displacement of [3H]LSD from human 5-HT6 receptor expressed in HEK cells incubated for 1 hr by Cheng-Prusoff analysis based microbeta scintillation c...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue incubated for 60 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue incubated for 60 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Displacement of [3H]-5-CT from recombinant human 5HT7 receptor expressed in HEK293 cells measured after 1 hr by microbeta scintillation counting anal...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Displacement of [3H]-5-CT from human 5HT7 receptor expressed in HEK cells incubated for 1 hr by Cheng-Prusoff analysis based microbeta scintillation ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Displacement of [3H]-ketanserin from recombinant human 5HT2A receptor expressed in HEK293 cells measured after 1.5 hrs by microbeta scintillation cou...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 28nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue incubated for 60 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue incubated for 60 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue incubated for 60 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 34nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue incubated for 60 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 41nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 42nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 42nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Displacement of [3H]-raclopride from recombinant human D2 receptor expressed in HEK293 cells measured after 1 hr by microbeta scintillation counting ...More data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Displacement of [3H]-raclopride from human D2 receptor expressed in HEK cells incubated for 1 hr by Cheng-Prusoff analysis based microbeta scintillat...More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 47nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Displacement of [3H]-8-OH-DPAT from recombinant human 5HT1A receptor expressed in CHO cell membranes measured after 60 mins by microbeta scintillatio...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 52nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in CHO-K1 cell membranes incubated for 60 mins by microbeta scintillation counting...More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University of Warsaw
Curated by ChEMBL
Medical University of Warsaw
Curated by ChEMBL
Affinity DataKi: 52nMAssay Description:Displacement of [3H]-citalopram from SERT in rat cortex tissue incubated for 60 mins by microbeta scintillation counting methodMore data for this Ligand-Target Pair
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