TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataKi: 5.60E+3nMAssay Description:Non-competitive inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by mi...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataKi: 6.30E+3nMAssay Description:Non-competitive inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by mi...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataKi: 1.60E+4nMAssay Description:Inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting...More data for this Ligand-Target Pair
TargetAdenosine kinase(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged AK using [2,8-3H]-adenosine as substrate after 20 mins by microbeta counting methodMore data for this Ligand-Target Pair
TargetAdenosine kinase(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human AKMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(RAT)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of CaV1.2 channel in rat tail artery myocytes assessed as reduction in Ba2+ current at -50 mV holding potential by whole-cell patch-clamp ...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 8.70E+3nMAssay Description:Inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting...More data for this Ligand-Target Pair
TargetAdenosine kinase(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 1.36E+4nMAssay Description:Inhibition of recombinant human His-tagged AK using [2,8-3H]-adenosine as substrate after 20 mins by microbeta counting methodMore data for this Ligand-Target Pair
TargetAdenosine kinase(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 1.36E+4nMAssay Description:Inhibition of recombinant human His-tagged AK using [2,8-3H]-adenosine as substrate after 20 mins by microbeta counting methodMore data for this Ligand-Target Pair
TargetAdenosine kinase(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 1.37E+4nMAssay Description:Inhibition of recombinant human His-tagged AK using [2,8-3H]-adenosine as substrate after 20 mins by microbeta counting methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 2.12E+4nMAssay Description:Inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting...More data for this Ligand-Target Pair
TargetAdenosine kinase(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 2.47E+4nMAssay Description:Inhibition of recombinant human His-tagged AK using [2,8-3H]-adenosine as substrate after 20 mins by microbeta counting methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 2.56E+4nMAssay Description:Inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting...More data for this Ligand-Target Pair
TargetAdenosine kinase(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 3.16E+4nMAssay Description:Inhibition of recombinant human His-tagged AK using [2,8-3H]-adenosine as substrate after 20 mins by microbeta counting methodMore data for this Ligand-Target Pair
TargetAdenosine kinase(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 3.22E+4nMAssay Description:Inhibition of recombinant human His-tagged AK using [2,8-3H]-adenosine as substrate after 20 mins by microbeta counting methodMore data for this Ligand-Target Pair
TargetAdenosine kinase(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of recombinant human His-tagged AK using [2,8-3H]-adenosine as substrate after 20 mins by microbeta counting methodMore data for this Ligand-Target Pair
TargetPhosphoethanolamine N-methyltransferase(Plasmodium falciparum)
University of Siena
Curated by ChEMBL
University of Siena
Curated by ChEMBL
Affinity DataIC50: 4.43E+4nMAssay Description:Inhibition of plasmodium falciparum phosphoethanolamine N-methyltransferase expressed in Escherichia coli using phosphoethanolamine as substrate and ...More data for this Ligand-Target Pair
TargetAdenosine kinase(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged AK using [2,8-3H]-adenosine as substrate after 20 mins by microbeta counting methodMore data for this Ligand-Target Pair
TargetAdenosine kinase(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged AK using [2,8-3H]-adenosine as substrate after 20 mins by microbeta counting methodMore data for this Ligand-Target Pair
TargetAdenosine kinase(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged AK using [2,8-3H]-adenosine as substrate after 20 mins by microbeta counting methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting...More data for this Ligand-Target Pair
TargetAdenosine kinase(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged AK using [2,8-3H]-adenosine as substrate after 20 mins by microbeta counting methodMore data for this Ligand-Target Pair
TargetAdenosine kinase(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged AK using [2,8-3H]-adenosine as substrate after 20 mins by microbeta counting methodMore data for this Ligand-Target Pair
TargetAdenosine kinase(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged AK using [2,8-3H]-adenosine as substrate after 20 mins by microbeta counting methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting...More data for this Ligand-Target Pair
TargetAdenosine kinase(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged AK using [2,8-3H]-adenosine as substrate after 20 mins by microbeta counting methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting...More data for this Ligand-Target Pair
TargetAdenosine kinase(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged AK using [2,8-3H]-adenosine as substrate after 20 mins by microbeta counting methodMore data for this Ligand-Target Pair
TargetAdenosine kinase(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged AK using [2,8-3H]-adenosine as substrate after 20 mins by microbeta counting methodMore data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of recombinant human His-tagged GSK3beta using GS-2 peptide as substrate in presence of [33P]gamma-ATP after 15 mins by microbeta counting...More data for this Ligand-Target Pair
TargetAdenosine kinase(Homo sapiens (Human))
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Universit£ degli Studi di Siena via Aldo Moro 2
Curated by ChEMBL
Affinity DataIC50: 5.74E+4nMAssay Description:Inhibition of recombinant human His-tagged AK using [2,8-3H]-adenosine as substrate after 20 mins by microbeta counting methodMore data for this Ligand-Target Pair