Compile Data Set for Download or QSAR
Found 24 with Last Name = 'iovenitti' and Initial = 'g'
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50354489(CHEMBL1836680)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Inhibition of human wild type full length N-terminal GST/6His-tagged SRC (M1 to L536 residues) expressed in baculovirus infected Sf9 cells using src ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2RMGPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50436584(CHEMBL2397802)copy SMILEScopy InChI
Affinity DataKi:  60nMAssay Description:Inhibition of human wild type full length N-terminal GST/6His-tagged SRC (M1 to L536 residues) expressed in baculovirus infected Sf9 cells using src ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2RMGPubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50515526(CHEMBL4452230)copy SMILEScopy InChI
Affinity DataKi:  120nMAssay Description:Inhibition of recombinant full length N-terminal His6 tagged human FYN expressed in baculovirus infected sf21 cells using KVEKIGEGTYGVVYK as substrat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85CHNPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50102903(CHEMBL3394092)copy SMILEScopy InChI
Affinity DataKi:  120nMAssay Description:Inhibition of human wild type full length N-terminal GST/6His-tagged ABL (P118 to S535 residues) expressed in Sf9 cells using abltide as substrate af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2RMGPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50102903(CHEMBL3394092)copy SMILEScopy InChI
Affinity DataKi:  130nMAssay Description:Inhibition of human wild type full length N-terminal GST/6His-tagged SRC (M1 to L536 residues) expressed in baculovirus infected Sf9 cells using src ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2RMGPubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50089575(CHEMBL3578214)copy SMILEScopy InChI
Affinity DataKi:  160nMAssay Description:Inhibition of recombinant full length N-terminal His6 tagged human FYN expressed in baculovirus infected sf21 cells using KVEKIGEGTYGVVYK as substrat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85CHNPubMed
TargetTyrosine-protein kinase Blk(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50515526(CHEMBL4452230)copy SMILEScopy InChI
Affinity DataKi:  170nMAssay Description:Inhibition of BLK (unknown origin) using KVEKIGEGTYGVVYK as substrate in presence of [gamma33P]ATP as substrate in presence of [gamma33P]ATP by scint...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85CHNPubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50515526(CHEMBL4452230)copy SMILEScopy InChI
Affinity DataKi:  190nMAssay Description:Inhibition of LYN (unknown origin) using KVEKIGEGTYGVVYK as substrate in presence of [gamma33P]ATP as substrate in presence of [gamma33P]ATP by scint...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85CHNPubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50089575(CHEMBL3578214)copy SMILEScopy InChI
Affinity DataKi:  190nMAssay Description:Inhibition of LYN (unknown origin) using KVEKIGEGTYGVVYK as substrate in presence of [gamma33P]ATP as substrate in presence of [gamma33P]ATP by scint...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85CHNPubMed
TargetTyrosine-protein kinase Blk(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50089575(CHEMBL3578214)copy SMILEScopy InChI
Affinity DataKi:  190nMAssay Description:Inhibition of BLK (unknown origin) using KVEKIGEGTYGVVYK as substrate in presence of [gamma33P]ATP as substrate in presence of [gamma33P]ATP by scint...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B85CHNPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50354486(CHEMBL411043)copy SMILEScopy InChI
Affinity DataKi:  370nMAssay Description:Inhibition of human wild type full length N-terminal GST/6His-tagged ABL (P118 to S535 residues) expressed in Sf9 cells using abltide as substrate af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2RMGPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50224368(1-(2-chloro-2-phenylethyl)-N-(3-chlorophenyl)-6-(m...)copy SMILEScopy InChI
Affinity DataKi:  600nMAssay Description:Inhibition of human wild type full length N-terminal GST/6His-tagged ABL (P118 to S535 residues) expressed in Sf9 cells using abltide as substrate af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2RMGPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50436584(CHEMBL2397802)copy SMILEScopy InChI
Affinity DataKi:  610nMAssay Description:Inhibition of human wild type full length N-terminal GST/6His-tagged ABL (P118 to S535 residues) expressed in Sf9 cells using abltide as substrate af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2RMGPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50224368(1-(2-chloro-2-phenylethyl)-N-(3-chlorophenyl)-6-(m...)copy SMILEScopy InChI
Affinity DataKi:  720nMAssay Description:Inhibition of human wild type full length N-terminal GST/6His-tagged SRC (M1 to L536 residues) expressed in baculovirus infected Sf9 cells using src ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2RMGPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50354489(CHEMBL1836680)copy SMILEScopy InChI
Affinity DataKi:  1.07E+3nMAssay Description:Inhibition of human wild type full length N-terminal GST/6His-tagged ABL (P118 to S535 residues) expressed in Sf9 cells using abltide as substrate af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2RMGPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50354486(CHEMBL411043)copy SMILEScopy InChI
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of human wild type full length N-terminal GST/6His-tagged SRC (M1 to L536 residues) expressed in baculovirus infected Sf9 cells using src ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2RMGPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50238530(CHEMBL4087882)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human wild type full length N-terminal GST/6His-tagged SRC (M1 to L536 residues) expressed in baculovirus infected Sf9 cells using src ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2RMGPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50238533(CHEMBL4060917)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human wild type full length N-terminal GST/6His-tagged ABL (P118 to S535 residues) expressed in Sf9 cells using abltide as substrate af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2RMGPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50238531(CHEMBL2407628)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human wild type full length N-terminal GST/6His-tagged ABL (P118 to S535 residues) expressed in Sf9 cells using abltide as substrate af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2RMGPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50238532(CHEMBL4084427)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human wild type full length N-terminal GST/6His-tagged ABL (P118 to S535 residues) expressed in Sf9 cells using abltide as substrate af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2RMGPubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50238530(CHEMBL4087882)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human wild type full length N-terminal GST/6His-tagged ABL (P118 to S535 residues) expressed in Sf9 cells using abltide as substrate af...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2RMGPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50238533(CHEMBL4060917)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human wild type full length N-terminal GST/6His-tagged SRC (M1 to L536 residues) expressed in baculovirus infected Sf9 cells using src ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2RMGPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50238532(CHEMBL4084427)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human wild type full length N-terminal GST/6His-tagged SRC (M1 to L536 residues) expressed in baculovirus infected Sf9 cells using src ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2RMGPubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50238531(CHEMBL2407628)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human kidney reninMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2RMGPubMed